Blockade of EIF5A hypusination limits colorectal cancer growth by inhibiting MYC elongation
Coni, Sonia, Serrao, Silvia Maria, Yurtsever, Zuleyha Nihan, Di Magno, Laura, Bordone, Rosa, Bertani, Camilla, Licursi, Valerio, Ianniello, Zaira, Infante, Paola, Moretti, Marta, Petroni, Marialaura, Guerrieri, Francesca, Fatica, Alessandro, Macone, Alberto, De Smaele, Enrico, Di Marcotullio, Lucia, Giannini, Giuseppe, Maroder, Marella, Agostinelli, Enzo, Canettieri, Gianluca
Published in Cell death & disease (10.12.2020)
Published in Cell death & disease (10.12.2020)
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Journal Article
Non-canonical Hedgehog/AMPK-Mediated Control of Polyamine Metabolism Supports Neuronal and Medulloblastoma Cell Growth
D’Amico, Davide, Antonucci, Laura, Di Magno, Laura, Coni, Sonia, Sdruscia, Giulia, Macone, Alberto, Miele, Evelina, Infante, Paola, Di Marcotullio, Lucia, De Smaele, Enrico, Ferretti, Elisabetta, Ciapponi, Laura, Giangaspero, Felice, Yates, John R., Agostinelli, Enzo, Cardinali, Beatrice, Screpanti, Isabella, Gulino, Alberto, Canettieri, Gianluca
Published in Developmental cell (12.10.2015)
Published in Developmental cell (12.10.2015)
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Journal Article
coactivator CRTC1 promotes cell proliferation and transformation via AP-1
Canettieri, Gianluca, Coni, Sonia, Della Guardia, Michele, Nocerino, Valentina, Antonucci, Laura, Di Magno, Laura, Screaton, Robert, Screpanti, Isabella, Giannini, Giuseppe, Gulino, Alberto
Published in Proceedings of the National Academy of Sciences - PNAS (03.02.2009)
Published in Proceedings of the National Academy of Sciences - PNAS (03.02.2009)
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Journal Article
The Mechanism of Action of Biguanides: New Answers to a Complex Question
Di Magno, Laura, Di Pastena, Fiorella, Bordone, Rosa, Coni, Sonia, Canettieri, Gianluca
Published in Cancers (30.06.2022)
Published in Cancers (30.06.2022)
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Journal Article
ERAP1 promotes Hedgehog-dependent tumorigenesis by controlling USP47-mediated degradation of βTrCP
Bufalieri, Francesca, Infante, Paola, Bernardi, Flavia, Caimano, Miriam, Romania, Paolo, Moretti, Marta, Lospinoso Severini, Ludovica, Talbot, Julie, Melaiu, Ombretta, Tanori, Mirella, Di Magno, Laura, Bellavia, Diana, Capalbo, Carlo, Puget, Stéphanie, De Smaele, Enrico, Canettieri, Gianluca, Guardavaccaro, Daniele, Busino, Luca, Peschiaroli, Angelo, Pazzaglia, Simonetta, Giannini, Giuseppe, Melino, Gerry, Locatelli, Franco, Gulino, Alberto, Ayrault, Olivier, Fruci, Doriana, Di Marcotullio, Lucia
Published in Nature communications (24.07.2019)
Published in Nature communications (24.07.2019)
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Journal Article
Phenformin Inhibits Hedgehog-Dependent Tumor Growth through a Complex I-Independent Redox/Corepressor Module
Di Magno, Laura, Manni, Simona, Di Pastena, Fiorella, Coni, Sonia, Macone, Alberto, Cairoli, Sara, Sambucci, Manolo, Infante, Paola, Moretti, Marta, Petroni, Marialaura, Nicoletti, Carmine, Capalbo, Carlo, De Smaele, Enrico, Di Marcotullio, Lucia, Giannini, Giuseppe, Battistini, Luca, Goffredo, Bianca Maria, Iorio, Egidio, Agostinelli, Enzo, Maroder, Marella, Canettieri, Gianluca
Published in Cell reports (Cambridge) (11.02.2020)
Published in Cell reports (Cambridge) (11.02.2020)
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Journal Article
Selective targeting of HDAC1/2 elicits anticancer effects through Gli1 acetylation in preclinical models of SHH Medulloblastoma
Coni, Sonia, Mancuso, Anna Barbara, Di Magno, Laura, Sdruscia, Giulia, Manni, Simona, Serrao, Silvia Maria, Rotili, Dante, Spiombi, Eleonora, Bufalieri, Francesca, Petroni, Marialaura, Kusio-Kobialka, Monika, De Smaele, Enrico, Ferretti, Elisabetta, Capalbo, Carlo, Mai, Antonello, Niewiadomski, Pawel, Screpanti, Isabella, Di Marcotullio, Lucia, Canettieri, Gianluca
Published in Scientific reports (09.03.2017)
Published in Scientific reports (09.03.2017)
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Journal Article
Gli2 acetylation at lysine 757 regulates hedgehog-dependent transcriptional output by preventing its promoter occupancy
Coni, Sonia, Antonucci, Laura, D'Amico, Davide, Di Magno, Laura, Infante, Paola, De Smaele, Enrico, Giannini, Giuseppe, Di Marcotullio, Lucia, Screpanti, Isabella, Gulino, Alberto, Canettieri, Gianluca
Published in PloS one (06.06.2013)
Published in PloS one (06.06.2013)
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Journal Article
Sulfonamide Inhibitors of β‐Catenin Signaling as Anticancer Agents with Different Output on c‐MYC
Di Magno, Laura, Di Pastena, Fiorella, Puxeddu, Michela, La Regina, Giuseppe, Coluccia, Antonio, Ciogli, Alessia, Manetto, Simone, Maroder, Marella, Canettieri, Gianluca, Silvestri, Romano, Nalli, Marianna
Published in ChemMedChem (03.12.2020)
Published in ChemMedChem (03.12.2020)
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Journal Article
Determination of Acetylation of the Gli Transcription Factors
Coni, Sonia, Di Magno, Laura, Canettieri, Gianluca
Published in Methods in molecular biology (Clifton, N.J.) (01.01.2015)
Published in Methods in molecular biology (Clifton, N.J.) (01.01.2015)
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Journal Article
KCTD15 inhibits the Hedgehog pathway in Medulloblastoma cells by increasing protein levels of the oncosuppressor KCASH2
Spiombi, Eleonora, Angrisani, Annapaola, Fonte, Simone, De Feudis, Giuseppina, Fabretti, Francesca, Cucchi, Danilo, Izzo, Mariapaola, Infante, Paola, Miele, Evelina, Po, Agnese, Di Magno, Laura, Magliozzi, Roberto, Guardavaccaro, Daniele, Maroder, Marella, Canettieri, Gianluca, Giannini, Giuseppe, Ferretti, Elisabetta, Gulino, Alberto, Di Marcotullio, Lucia, Moretti, Marta, De Smaele, Enrico
Published in Oncogenesis (New York, NY) (04.11.2019)
Published in Oncogenesis (New York, NY) (04.11.2019)
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Journal Article
Partial Truncation of the C-Terminal Domain of PTCH1 in Cancer Enhances Autophagy and Metabolic Adaptability
Caballero-Ruiz, Begoña, Gkotsi, Danai S, Ollerton, Hattie, Morales-Alcala, Cintli C, Bordone, Rosa, Jenkins, Georgia M L, Di Magno, Laura, Canettieri, Gianluca, Riobo-Del Galdo, Natalia A
Published in Cancers (06.01.2023)
Published in Cancers (06.01.2023)
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Journal Article
Opposite Effect of Thyroid Hormones on Oxidative Stress and on Mitochondrial Respiration in COVID-19 Patients
De Vitis, Claudia, Capalbo, Carlo, Torsello, Alessandra, Napoli, Christian, Salvati, Valentina, Loffredo, Chiara, Blandino, Giovanni, Piaggio, Giulia, Auciello, Francesca Romana, Pelliccia, Flaminia, Salerno, Gerardo, Simmaco, Maurizio, Di Magno, Laura, Canettieri, Gianluca, Coluzzi, Flaminia, Mancini, Rita, Rocco, Monica, Sciacchitano, Salvatore
Published in Antioxidants (01.10.2022)
Published in Antioxidants (01.10.2022)
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Journal Article
Enzymatic Spermine Metabolites Induce Apoptosis Associated with Increase of p53, caspase-3 and miR-34a in Both Neuroblastoma Cells, SJNKP and the N-Myc-Amplified Form IMR5
Kanamori, Yuta, Finotti, Alessia, Di Magno, Laura, Canettieri, Gianluca, Tahara, Tomoaki, Timeus, Fabio, Greco, Antonio, Tirassa, Paola, Gasparello, Jessica, Fino, Pasquale, Di Liegro, Carlo Maria, Proia, Patrizia, Schiera, Gabriella, Di Liegro, Italia, Gambari, Roberto, Agostinelli, Enzo
Published in Cells (Basel, Switzerland) (31.07.2021)
Published in Cells (Basel, Switzerland) (31.07.2021)
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Journal Article
Combined inhibition of polyamine metabolism and eIF5A hypusination suppresses colorectal cancer growth through a converging effect on MYC translation
Coni, Sonia, Bordone, Rosa, Ivy, Devon Michael, Yurtsever, Zuleyha Nihan, Di Magno, Laura, D'Amico, Rodrigo, Cesaro, Bianca, Fatica, Alessandro, Belardinilli, Francesca, Bufalieri, Francesca, Maroder, Marella, De Smaele, Enrico, Di Marcotullio, Lucia, Giannini, Giuseppe, Agostinelli, Enzo, Canettieri, Gianluca
Published in Cancer letters (10.04.2023)
Published in Cancer letters (10.04.2023)
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Journal Article
Discovery of novel human lactate dehydrogenase inhibitors: Structure-based virtual screening studies and biological assessment
Di Magno, Laura, Coluccia, Antonio, Bufano, Marianna, Ripa, Silvia, La Regina, Giuseppe, Nalli, Marianna, Di Pastena, Fiorella, Canettieri, Gianluca, Silvestri, Romano, Frati, Luigi
Published in European journal of medicinal chemistry (05.10.2022)
Published in European journal of medicinal chemistry (05.10.2022)
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Journal Article
Human duodenal submucosal glands contain a defined stem/progenitor subpopulation with liver-specific regenerative potential
Cardinale, Vincenzo, Carpino, Guido, Overi, Diletta, Safarikia, Samira, Zhang, Wencheng, Kanke, Matt, Franchitto, Antonio, Costantini, Daniele, Riccioni, Olga, Nevi, Lorenzo, Chiappetta, Michele, Onori, Paolo, Franchitto, Matteo, Bini, Simone, Hung, Yu-Han, Lai, Quirino, Zizzari, Ilaria, Nuti, Marianna, Nicoletti, Carmine, Checquolo, Saula, Di Magno, Laura, Giuli, Maria Valeria, Rossi, Massimo, Sethupathy, Praveen, Reid, Lola M., Alvaro, Domenico, Gaudio, Eugenio
Published in Journal of hepatology (01.01.2023)
Published in Journal of hepatology (01.01.2023)
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Journal Article
4-(3-Phenyl-4-(3,4,5-trimethoxybenzoyl)-1 H -pyrrol-1-yl)benzenesulfonamide, a Novel Carbonic Anhydrase and Wnt/β-Catenin Signaling Pathway Dual-Targeting Inhibitor with Potent Activity against Multidrug Resistant Cancer Cells
Masci, Domiziana, Puxeddu, Michela, Di Magno, Laura, D'Ambrosio, Michele, Parisi, Anastasia, Nalli, Marianna, Bai, Ruoli, Coluccia, Antonio, Sciò, Pietro, Orlando, Viviana, D'Angelo, Sara, Biagioni, Stefano, Urbani, Andrea, Hamel, Ernest, Nocentini, Alessio, Filiberti, Serena, Turati, Marta, Ronca, Roberto, Kopecka, Joanna, Riganti, Chiara, Fionda, Cinzia, Bordone, Rosa, Della Rocca, Giorgia, Canettieri, Gianluca, Supuran, Claudiu T, Silvestri, Romano, La Regina, Giuseppe
Published in Journal of medicinal chemistry (09.11.2023)
Published in Journal of medicinal chemistry (09.11.2023)
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Journal Article
4‑(3-Phenyl-4-(3,4,5-trimethoxybenzoyl)‑1H‑pyrrol-1-yl)benzenesulfonamide, a Novel Carbonic Anhydrase and Wnt/β-Catenin Signaling Pathway Dual-Targeting Inhibitor with Potent Activity against Multidrug Resistant Cancer Cells
Masci, Domiziana, Puxeddu, Michela, Di Magno, Laura, D’Ambrosio, Michele, Parisi, Anastasia, Nalli, Marianna, Bai, Ruoli, Coluccia, Antonio, Sciò, Pietro, Orlando, Viviana, D’Angelo, Sara, Biagioni, Stefano, Urbani, Andrea, Hamel, Ernest, Nocentini, Alessio, Filiberti, Serena, Turati, Marta, Ronca, Roberto, Kopecka, Joanna, Riganti, Chiara, Fionda, Cinzia, Bordone, Rosa, Della Rocca, Giorgia, Canettieri, Gianluca, Supuran, Claudiu T., Silvestri, Romano, La Regina, Giuseppe
Published in Journal of medicinal chemistry (09.11.2023)
Published in Journal of medicinal chemistry (09.11.2023)
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