Direct Preparation of Amides from Amine Hydrochloride Salts and Orthoesters: A Synthetic and Mechanistic Perspective
Di Grandi, Martin J., Bennett, Caitlin, Cagino, Kristen, Muccini, Arnold, Suraci, Corey, Saba, Shahrokh
Published in Synthetic communications (17.11.2015)
Published in Synthetic communications (17.11.2015)
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Journal Article
Thiourea inhibitors of herpesviruses. Part 3: Inhibitors of varicella zoster virus
Di Grandi, Martin J, Curran, Kevin J, Feigelson, Gregg, Prashad, Amar, Ross, Adma A, Visalli, Robert, Fairhurst, Jeanette, Feld, Boris, Bloom, Jonathan D
Published in Bioorganic & medicinal chemistry letters (16.08.2004)
Published in Bioorganic & medicinal chemistry letters (16.08.2004)
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Journal Article
Novel pyrazolopyrimidines as highly potent B-Raf inhibitors
Di Grandi, Martin J., Berger, Dan M., Hopper, Darrin W., Zhang, Chunchun, Dutia, Minu, Dunnick, Alejandro L., Torres, Nancy, Levin, Jeremy I., Diamantidis, George, Zapf, Christoph W., Bloom, Jonathan D., Hu, YongBo, Powell, Dennis, Wojciechowicz, Donald, Collins, Karen, Frommer, Eileen
Published in Bioorganic & medicinal chemistry letters (15.12.2009)
Published in Bioorganic & medicinal chemistry letters (15.12.2009)
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Journal Article
Synthesis of competent nucleophiles for delivering the A ring of taxol
Di Grandi, Martin J, Jung, David K, Krol, Walter J, Danishefsky, Samuel J
Published in Journal of organic chemistry (01.08.1993)
Published in Journal of organic chemistry (01.08.1993)
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Journal Article
Total Synthesis of Baccatin III and Taxol
Danishefsky, Samuel J, Masters, John J, Young, Wendy B, Link, J. T, Snyder, Lawrence B, Magee, Thomas V, Jung, David K, Isaacs, Richard C. A, Bornmann, William G, Alaimo, Cheryl A, Coburn, Craig A, Di Grandi, Martin J
Published in Journal of the American Chemical Society (27.03.1996)
Published in Journal of the American Chemical Society (27.03.1996)
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Journal Article
Pyrimido[1,2-b]-1,2,4,5-tetrazin-6-ones as HCMV protease inhibitors: A new class of heterocycles with flavin-like redox properties
DI GRANDI, Martin J, CURRAN, Kevin J, BAUM, Ellen Z, BEBERNITZ, Geraldine, ELLESTAD, George A, DING, Wei-Dong, LANG, Stanley A, ROSSI, Miriam, BLOOMS, Jonathan D
Published in Bioorganic & medicinal chemistry letters (20.10.2003)
Published in Bioorganic & medicinal chemistry letters (20.10.2003)
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Journal Article
Synthesis of an enantiomerically pure intermediate containing the CD substructure of taxol
Isaacs, Richard C. A, Di Grandi, Martin J, Danishefsky, Samuel J
Published in Journal of organic chemistry (01.07.1993)
Published in Journal of organic chemistry (01.07.1993)
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Journal Article
Degradative routes to electrophilic CD-substructures of taxol
Di Grandi, Martin J, Coburn, Craig A, Isaacs, Richard C. A, Danishefsky, Samuel J
Published in Journal of organic chemistry (01.12.1993)
Published in Journal of organic chemistry (01.12.1993)
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Journal Article
The calculation and synthesis of a template molecule
Wilson, Stephen R., Tam, Wai K., Di Grandi, Martin J., Cui, Weili
Published in Tetrahedron (23.04.1993)
Published in Tetrahedron (23.04.1993)
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Journal Article
Thiourea Inhibitors of Herpesviruses. Part 3. Inhibitors of Varicella Zoster Virus
Di Grandi, Martin J., Curran, Kevin J., Feigelson, Gregg, Prashad, Amar, Ross, Adma A., Visalli, Robert, Fairhurst, Jeanette, Feld, Boris, Bloom, Jonathan D.
Published in ChemInform (07.12.2004)
Published in ChemInform (07.12.2004)
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Journal Article
Pyrimido[1,2-b]-1,2,4,5-tetrazin-6-ones as HCMV Protease Inhibitors: A New Class of Heterocycles with Flavin-Like Redox Properties
Di Grandi, Martin J., Curran, Kevin J., Baum, Ellen Z., Bebernitz, Geraldine, Ellestad, George A., Ding, Wei-Dong, Lang, Stanley A., Rossi, Miriam, Bloom, Jonathan D.
Published in ChemInform (20.01.2004)
Published in ChemInform (20.01.2004)
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Journal Article