Design, Synthesis, Molecular Docking, and Preliminary Pharmacological Screening of some New Benzo[d]thiazol-2-ylamino Containing Chromen-2- one Derivatives with Atypical Antipsychotic Profile
Gawai, Ashish A, Biyani, Kailash R, Das, Sanjib, Tapadiya, Ganesh G, Mokale, Santosh N, Dhawale, Sachin A
Published in Current computer-aided drug design (01.01.2023)
Published in Current computer-aided drug design (01.01.2023)
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Natural polymers as potential P-glycoprotein inhibitors: Pre-ADMET profile and computational analysis as a proof of concept to fight multidrug resistance in cancer
Gandla, Kumaraswamy, Islam, Fahadul, Zehravi, Mehrukh, Karunakaran, Anandakumar, Sharma, Indu, Haque, M. Akiful, Kumar, Sanjay, Pratyush, Kumar, Dhawale, Sachin A., Nainu, Firzan, Khan, Sharuk L., Islam, Md Rezaul, Al-Mugren, Kholoud Saad, Siddiqui, Falak A., Emran, Talha Bin, Khandaker, Mayeen Uddin
Published in Heliyon (01.09.2023)
Published in Heliyon (01.09.2023)
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The Design, Synthesis, and Evaluation of Diaminopimelic Acid Derivatives as Potential dapF Inhibitors Preventing Lysine Biosynthesis for Antibacterial Activity
Shaikh, Mohd Sayeed, Kale, Mayura A., Muralidharan, V., Venkatachalam, T., Ali, Syed Sarfaraz, Islam, Fahadul, Khan, Sharuk L., Siddiqui, Falak A., Urmee, Humaira, Tapadiya, Ganesh G., Dhawale, Sachin A., Ming, Long Chiau, Ibrahim, Ibrahim Abdel Aziz, Alzahrani, Abdullah R., Sarker, Md. Moklesur Rahman, Azlina, Mohd Fahami Nur
Published in Antibiotics (Basel) (01.01.2023)
Published in Antibiotics (Basel) (01.01.2023)
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Molecular docking and molecular dynamic simulation-based phytoconstituents against SARS-CoV-2 with dual inhibition of the primary protease targets
Dhawale, Sachin A, Mahajan, Sadhana, Pandit, Madhuri, Gawale, Sachin, Ghodke, Mangesh, Tapadiya, Ganesh
Published in Natural product research (22.03.2024)
Published in Natural product research (22.03.2024)
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Dual targeting in prostate cancer with phytoconstituents as a potent lead: a computational approach for novel drug discovery
Dhawale, Sachin A., Bhosle, Pallavi, Mahajan, Sadhana, Patil, Geetanjali, Gawale, Sachin, Ghodke, Mangesh, Tapadiya, Ganesh, Ansari, Azim
Published in Journal of biomolecular structure & dynamics (30.08.2023)
Published in Journal of biomolecular structure & dynamics (30.08.2023)
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Green synthesis of silver nanoparticles mediated Azadirachta indica extract and study of their characterization, molecular docking, and antibacterial activity
Gawai, Ashish A., Kharat, Amol R., Chorge, Shivani S., Dhawale, Sachin A.
Published in Journal of molecular recognition (01.10.2023)
Published in Journal of molecular recognition (01.10.2023)
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Synthesis, antiproliferative activity and insilco studies of substituted 2-((N-benzyl-5-bromo-2-methoxyphenyl) sulfonamide) glycinamide derivatives
Gaikwad, Dattatray D., Dhawale, Sachin A., Pawar, Chandrakant D., Pansare, Dattatraya N., Pawar, Umakant D., Zine, Ashok M.
Published in Synthetic communications (01.09.2024)
Published in Synthetic communications (01.09.2024)
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Novel Pyrazole‐Chalcone Hybrids: Synthesis and Computational Insights Against Breast Cancer
Dabhade, Pratap S., Dabhade, Manjushri P., Rathod, Lala S., Dhawale, Sachin A., More, Shweta A., Chaudhari, Somdatta Y., Mokale, Santosh N.
Published in Chemistry & biodiversity (01.07.2024)
Published in Chemistry & biodiversity (01.07.2024)
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Exploring the potential of small molecules of dual c-Met and VEGFR inhibitors for advances and future drug discovery in cancer therapy
Dhawale, Sachin A., Deokar, Arundhati V., Firdous, Momin Aaliya, Pandit, Madhuri, Chaudhari, Minal Y., Salve, Sameer B., Khandgaonkar, Madhuri, Parwe, Mahesh, Khalse, Rupesh, Dake, Shruti G., Chatse, Siddharth H., Tapadiya, Ganesh G.
Published in Future journal of pharmaceutical sciences (01.12.2024)
Published in Future journal of pharmaceutical sciences (01.12.2024)
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Synthesis and Pharmacological Evaluation of Some Amide Functionalized 1H‐Benzo[d]imidazole‐2‐thiol Derivatives as Antimicrobial Agents
Singu, Padma S., Kanugala, Sirisha, Dhawale, Sachin A., Kumar, C. Ganesh, Kumbhare, Ravindra M.
Published in ChemistrySelect (Weinheim) (09.01.2020)
Published in ChemistrySelect (Weinheim) (09.01.2020)
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Journal Article
Synthesis and Pharmacological Evaluation of Some Amide Functionalized 1 H ‐Benzo[ d ]imidazole‐2‐thiol Derivatives as Antimicrobial Agents
Singu, Padma S., Kanugala, Sirisha, Dhawale, Sachin A., Kumar, C. Ganesh, Kumbhare, Ravindra M.
Published in ChemistrySelect (Weinheim) (09.01.2020)
Published in ChemistrySelect (Weinheim) (09.01.2020)
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Journal Article
The Design, Synthesis, and Evaluation of Diaminopimelic Acid Derivatives as Potential dap F Inhibitors Preventing Lysine Biosynthesis for Antibacterial Activity
Shaikh, Mohd Sayeed, Kale, Mayura A, Muralidharan, V, Venkatachalam, T, Ali, Syed Sarfaraz, Islam, Fahadul, Khan, Sharuk L, Siddiqui, Falak A, Urmee, Humaira, Tapadiya, Ganesh G, Dhawale, Sachin A, Ming, Long Chiau, Ibrahim, Ibrahim Abdel Aziz, Alzahrani, Abdullah R, Sarker, Md Moklesur Rahman, Azlina, Mohd Fahami Nur
Published in Antibiotics (Basel) (28.12.2022)
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Published in Antibiotics (Basel) (28.12.2022)
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