Visible‐Light Photoswitchable Benzimidazole Azo‐Arenes as β‐Arrestin2‐Biased Selective Cannabinoid 2 Receptor Agonists
Steinmüller, Sophie A. M., Fender, Julia, Deventer, Marie H., Tutov, Anna, Lorenz, Kristina, Stove, Christophe P., Hislop, James N., Decker, Michael
Published in Angewandte Chemie International Edition (04.12.2023)
Published in Angewandte Chemie International Edition (04.12.2023)
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Assessment of structure-activity relationships and biased agonism at the Mu opioid receptor of novel synthetic opioids using a novel, stable bio-assay platform
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Published in Biochemical pharmacology (01.07.2020)
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In vitro characterization of the pyrazole-carrying synthetic cannabinoid receptor agonist 5F-3,5-AB-PFUPPYCA and its structural analogs
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Published in Forensic science international (01.02.2023)
Published in Forensic science international (01.02.2023)
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Frontispiece: Visible‐Light Photoswitchable Benzimidazole Azo‐Arenes as β‐Arrestin2‐Biased Selective Cannabinoid 2 Receptor Agonists
Steinmüller, Sophie A. M., Fender, Julia, Deventer, Marie H., Tutov, Anna, Lorenz, Kristina, Stove, Christophe P., Hislop, James N., Decker, Michael
Published in Angewandte Chemie International Edition (04.12.2023)
Published in Angewandte Chemie International Edition (04.12.2023)
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Off-target activity of NBOMes and NBOMe analogs at the µ opioid receptor
Deventer, Marie H., Persson, Mattias, Laus, Antonio, Pottie, Eline, Cannaert, Annelies, Tocco, Graziella, Gréen, Henrik, Stove, Christophe P.
Published in Archives of toxicology (01.05.2023)
Published in Archives of toxicology (01.05.2023)
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Cannabinoid receptor activation potential of the next generation, generic ban evading OXIZID synthetic cannabinoid receptor agonists
Deventer, M H, Van Uytfanghe, K, Vinckier, I M J, Reniero, F, Guillou, C, Stove, C P
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Published in Drug testing and analysis (01.09.2022)
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A Fentanyl Hapten-Displaying Lipid Nanoparticle Vaccine that Non-Covalently Encapsulates a TLR7/8 Agonist and T-helper Epitope Induces Protective Anti-Fentanyl Immunity
Zhong, Zifu, Deventer, Marie H, Chen, Yong, Vanhee, Stijn, Lammens, Inés, Deswarte, Kim, Huang, Yi, Ye, Tingting, Wang, Haixiu, Nuhn, Lutz, Vandeputte, Marthe, Gontsarik, Mark, Cui, Xiaole, Sanders, Niek N, Lienenklaus, Stefan, Lambrecht, Bart N, Stove, Christophe P, Baptista, Antonio P, de Geest, Bruno
Published in Angewandte Chemie International Edition (23.10.2024)
Published in Angewandte Chemie International Edition (23.10.2024)
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Waxy- or Putty-Like Materials as a Novel Drug Preparation for Synthetic Cannabinoid Receptor Agonists: Detection in Prisons and In Vitro Cannabinoid Receptor Activity
Timmerman, Axelle, Deventer, Marie H, Andrews, Rachael, Reid, Robert, Marland, Victoria, Edwards, Darren, Pudney, Christopher R, Nic Daéid, Niamh, Stove, Christophe P, Norman, Caitlyn
Published in Drug testing and analysis (15.10.2024)
Published in Drug testing and analysis (15.10.2024)
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Dual-Acting Small Molecules: Subtype-Selective Cannabinoid Receptor 2 Agonist/Butyrylcholinesterase Inhibitor Hybrids Show Neuroprotection in an Alzheimer’s Disease Mouse Model
Spatz, Philipp, Steinmüller, Sophie A. M., Tutov, Anna, Poeta, Eleonora, Morilleau, Axelle, Carles, Allison, Deventer, Marie H., Hofmann, Julian, Stove, Christophe P., Monti, Barbara, Maurice, Tangui, Decker, Michael
Published in Journal of medicinal chemistry (11.05.2023)
Published in Journal of medicinal chemistry (11.05.2023)
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In vitro cannabinoid activity profiling of generic ban-evading brominated synthetic cannabinoid receptor agonists and their analogs
Deventer, Marie H, Persson, Mattias, Norman, Caitlyn, Liu, Huiling, Connolly, Matthew J, Daéid, Niamh Nic, McKenzie, Craig, Gréen, Henrik, Stove, Christophe P
Published in Drug testing and analysis (01.06.2024)
Published in Drug testing and analysis (01.06.2024)
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Detection in seized samples, analytical characterization, and in vitro metabolism of the newly emerged 5-bromo-indazole-3-carboxamide synthetic cannabinoid receptor agonists
Norman, Caitlyn, Webling, Kristin, Kyslychenko, Oleksandra, Reid, Robert, Krotulski, Alex J, Farrell, Ryan, Deventer, Marie H, Liu, Huiling, Connolly, Matthew J, Guillou, Claude, Vinckier, Inge M J, Logan, Barry K, NicDaéid, Niamh, McKenzie, Craig, Stove, Christophe P, Gréen, Henrik
Published in Drug testing and analysis (01.09.2024)
Published in Drug testing and analysis (01.09.2024)
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In vitro cannabinoid receptor activity, metabolism, and detection in seized samples of CH‐PIATA, a new indole‐3‐acetamide synthetic cannabinoid
Norman, Caitlyn, Deventer, Marie H., Dremann, Olivia, Reid, Robert, Van Uytfanghe, Katleen, Guillou, Claude, Vinckier, Inge M. J., Nic Daéid, Niamh, Krotulski, Alex, Stove, Christophe P.
Published in Drug testing and analysis (01.04.2024)
Published in Drug testing and analysis (01.04.2024)
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Structure-activity relationships of valine, tert-leucine, and phenylalanine amino acid-derived synthetic cannabinoid receptor agonists related to ADB-BUTINACA, APP-BUTINACA, and ADB-P7AICA
Sparkes, Eric, Cairns, Elizabeth A., Kevin, Richard C., Lai, Felcia, Grafinger, Katharina Elisabeth, Chen, Shuli, Deventer, Marie H., Ellison, Ross, Boyd, Rochelle, Martin, Lewis J., McGregor, Iain S., Gerona, Roy R., Hibbs, David E., Auwaerter, Volker, Glass, Michelle, Stove, Christophe, Banister, Samuel D.
Published in MedChemComm (23.02.2022)
Published in MedChemComm (23.02.2022)
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NNL-3: A Synthetic Intermediate or a New Class of Hydroxybenzotriazole Esters with Cannabinoid Receptor Activity?
Ametovski, Adam, Cairns, Elizabeth A, Grafinger, Katharina Elisabeth, Cannaert, Annelies, Deventer, Marie H, Chen, Shuli, Wu, Xinyi, Shepperson, Caitlin E, Lai, Felcia, Ellison, Ross, Gerona, Roy, Blakey, Karen, Kevin, Richard, McGregor, Iain S, Hibbs, David E, Glass, Michelle, Stove, Christophe, Auwärter, Volker, Banister, Samuel D
Published in ACS chemical neuroscience (03.11.2021)
Published in ACS chemical neuroscience (03.11.2021)
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Development of an Indole-Amide-Based Photoswitchable Cannabinoid Receptor Subtype 1 (CB1R) “Cis-On” Agonist
Rodríguez-Soacha, Diego A., Steinmüller, Sophie A. M., Işbilir, Ali, Fender, Julia, Deventer, Marie H., Ramírez, Yesid A., Tutov, Anna, Sotriffer, Christoph, Stove, Christophe P., Lorenz, Kristina, Lohse, Martin J., Hislop, James N., Decker, Michael
Published in ACS chemical neuroscience (17.08.2022)
Published in ACS chemical neuroscience (17.08.2022)
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Frontispiz: Mit sichtbarem Licht schaltbare Benzimidazol‐Azo‐Arene wirken als β‐Arrestin2 funktionell selektive Cannabinoid‐Rezeptor 2 Agonisten
Steinmüller, Sophie A. M., Fender, Julia, Deventer, Marie H., Tutov, Anna, Lorenz, Kristina, Stove, Christophe P., Hislop, James N., Decker, Michael
Published in Angewandte Chemie (04.12.2023)
Published in Angewandte Chemie (04.12.2023)
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Mit sichtbarem Licht schaltbare Benzimidazol‐Azo‐Arene wirken als β‐Arrestin2 funktionell selektive Cannabinoid‐Rezeptor 2 Agonisten
Steinmüller, Sophie A. M., Fender, Julia, Deventer, Marie H., Tutov, Anna, Lorenz, Kristina, Stove, Christophe P., Hislop, James N., Decker, Michael
Published in Angewandte Chemie (04.12.2023)
Published in Angewandte Chemie (04.12.2023)
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Journal Article
Dual-Acting Small Molecules: Subtype-Selective Cannabinoid Receptor 2 Agonist/Butyrylcholinesterase Inhibitor Hybrids Show Neuroprotection in an Alzheimer?s Disease Mouse Model
Spatz, Philipp, Steinmueller, Sophie A. M., Tutov, Anna, Poeta, Eleonora, Morilleau, Axelle, Carles, Allison, Deventer, Marie H., Hofmann, Julian, Stove, Christophe P., Monti, Barbara, Maurice, Tangui, Decker, Michael
Published in Journal of medicinal chemistry (11.05.2023)
Published in Journal of medicinal chemistry (11.05.2023)
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