Quantification of Accurate Composition and Total Abundance of Homologous Proteins by Conserved-Plus-Surrogate Peptide Approach: Quantification of UDP Glucuronosyltransferases in Human Tissues
Ahire, Deepak, Patel, Mitesh, Deshmukh, Sujal V, Prasad, Bhagwat
Published in Drug metabolism and disposition (01.03.2023)
Published in Drug metabolism and disposition (01.03.2023)
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The discovery of 6-amino nicotinamides as potent and selective histone deacetylase inhibitors
Hamblett, Christopher L., Methot, Joey L., Mampreian, Dawn M., Sloman, David L., Stanton, Matthew G., Kral, Astrid M., Fleming, Judith C., Cruz, Jonathan C., Chenard, Melissa, Ozerova, Nicole, Hitz, Anna M., Wang, Hongmei, Deshmukh, Sujal V., Nazef, Naim, Harsch, Andreas, Hughes, Bethany, Dahlberg, William K., Szewczak, Alex A., Middleton, Richard E., Mosley, Ralph T., Secrist, J. Paul, Miller, Thomas A.
Published in Bioorganic & medicinal chemistry letters (01.10.2007)
Published in Bioorganic & medicinal chemistry letters (01.10.2007)
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Evaluation of JAK3 Biology in Autoimmune Disease Using a Highly Selective, Irreversible JAK3 Inhibitor
Elwood, Fiona, Witter, David J, Piesvaux, Jennifer, Kraybill, Brian, Bays, Nathan, Alpert, Carla, Goldenblatt, Peter, Qu, Yujie, Ivanovska, Irena, Lee, Hyun-Hee, Chiu, Chi-Sung, Tang, Hao, Scott, Mark E, Deshmukh, Sujal V, Zielstorff, Mark, Byford, Alan, Chakravarthy, Kalyan, Dorosh, Lauren, Rivkin, Alexey, Klappenbach, Joel, Pan, Bo-Sheng, Kariv, Ilona, Dinsmore, Christopher, Slipetz, Deborah, Dandliker, Peter J
Published in The Journal of pharmacology and experimental therapeutics (01.05.2017)
Published in The Journal of pharmacology and experimental therapeutics (01.05.2017)
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The Discovery of 3‑((4-Chloro-3-methoxyphenyl)amino)-1-((3R,4S)‑4-cyanotetrahydro‑2H‑pyran-3-yl)‑1H‑pyrazole-4-carboxamide, a Highly Ligand Efficient and Efficacious Janus Kinase 1 Selective Inhibitor with Favorable Pharmacokinetic Properties
Siu, Tony, Brubaker, Jason, Fuller, Peter, Torres, Luis, Zeng, Hongbo, Close, Joshua, Mampreian, Dawn M., Shi, Feng, Liu, Duan, Fradera, Xavier, Johnson, Kevin, Bays, Nathan, Kadic, Elma, He, Fang, Goldenblatt, Peter, Shaffer, Lynsey, Patel, Sangita B., Lesburg, Charles A., Alpert, Carla, Dorosh, Lauren, Deshmukh, Sujal V., Yu, Hongshi, Klappenbach, Joel, Elwood, Fiona, Dinsmore, Christopher J., Fernandez, Rafael, Moy, Lily, Young, Jonathan R.
Published in Journal of medicinal chemistry (14.12.2017)
Published in Journal of medicinal chemistry (14.12.2017)
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Structure-based design and development of (benz)imidazole pyridones as JAK1-selective kinase inhibitors
Simov, Vladimir, Deshmukh, Sujal V., Dinsmore, Christopher J., Elwood, Fiona, Fernandez, Rafael B., Garcia, Yudith, Gibeau, Craig, Gunaydin, Hakan, Jung, Joon, Katz, Jason D., Kraybill, Brian, Lapointe, Blair, Patel, Sangita B., Siu, Tony, Su, Hua, Young, Jonathan R.
Published in Bioorganic & medicinal chemistry letters (01.04.2016)
Published in Bioorganic & medicinal chemistry letters (01.04.2016)
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Journal Article
MK-2461, a Novel Multitargeted Kinase Inhibitor, Preferentially Inhibits the Activated c-Met Receptor
PAN, Bo-Sheng, CHAN, Grace K. Y, JEWELL, James P, KARIV, Ilona, KATZ, Jason D, KUNII, Kaiko, WEI LU, LUTTERBACH, Bart A, PAWELETZ, Cloud P, XIANLU QU, REILLY, John F, SZEWCZAK, Alexander A, CHENARD, Melissa, QINWEN ZENG, KOHL, Nancy E, DINSMORE, Christopher J, CHI, An, DAVIS, Lenora J, DESHMUKH, Sujal V, GIBBS, Jackson B, GIL, Susana, GAOZHEN HANG, HATCH, Harold
Published in Cancer research (Chicago, Ill.) (15.02.2010)
Published in Cancer research (Chicago, Ill.) (15.02.2010)
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Discovery of 1‑[3-(1-Methyl‑1H‑pyrazol-4-yl)-5-oxo‑5H‑benzo[4,5]cyclohepta[1,2‑b]pyridin-7-yl]‑N‑(pyridin-2-ylmethyl)methanesulfonamide (MK-8033): A Specific c‑Met/Ron Dual Kinase Inhibitor with Preferential Affinity for the Activated State of c‑Met
Northrup, Alan B, Katcher, Matthew H, Altman, Michael D, Chenard, Melissa, Daniels, Matthew H, Deshmukh, Sujal V, Falcone, Danielle, Guerin, David J, Hatch, Harold, Li, Chaomin, Lu, Wei, Lutterbach, Bart, Allison, Timothy J, Patel, Sangita B, Reilly, John F, Reutershan, Michael, Rickert, Keith W, Rosenstein, Craig, Soisson, Stephen M, Szewczak, Alexander A, Walker, Deborah, Wilson, Kevin, Young, Jonathan R, Pan, Bo-Sheng, Dinsmore, Christopher J
Published in Journal of medicinal chemistry (28.03.2013)
Published in Journal of medicinal chemistry (28.03.2013)
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Discovery of a 5H-Benzo[4,5]cyclohepta[1,2-b]pyridin-5-one (MK-2461) Inhibitor of c-Met Kinase for the Treatment of Cancer
Katz, Jason D, Jewell, James P, Guerin, David J, Lim, Jongwon, Dinsmore, Christopher J, Deshmukh, Sujal V, Pan, Bo-Sheng, Marshall, C. Gary, Lu, Wei, Altman, Michael D, Dahlberg, William K, Davis, Lenora, Falcone, Danielle, Gabarda, Ana E, Hang, Gaozhen, Hatch, Harold, Holmes, Rachael, Kunii, Kaiko, Lumb, Kevin J, Lutterbach, Bart, Mathvink, Robert, Nazef, Naim, Patel, Sangita B, Qu, Xianlu, Reilly, John F, Rickert, Keith W, Rosenstein, Craig, Soisson, Stephen M, Spencer, Kerrie B, Szewczak, Alexander A, Walker, Deborah, Wang, Wenxian, Young, Jonathan, Zeng, Qinwen
Published in Journal of medicinal chemistry (23.06.2011)
Published in Journal of medicinal chemistry (23.06.2011)
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Potent benzoazepinone γ-secretase modulators with improved bioavailability
Methot, Joey L., Fischer, Christian, Li, Chaomin, Rivkin, Alexey, Ahearn, Sean P., Brown, William Colby, Kattar, Sam, Kelley, Elizabeth, Mampreian, Dawn M., Schell, Adam, Rosenau, Andrew, Zhou, Hua, Ball, Richard, Deshmukh, Sujal V., Jeliazkova-Mecheva, Valentina V., Diaz, Damaris, Moy, Lily Y., Kenific, Candia M., Moxham, Chris, Shah, Sanjiv, Nuthall, Hugh, Szewczak, Alexander A., Hill, Armetta, Hughes, Bethany, Smotrov, Nadya, Munoz, Benito, Miller, Thomas A., Shearman, Mark S.
Published in Bioorganic & medicinal chemistry letters (01.09.2015)
Published in Bioorganic & medicinal chemistry letters (01.09.2015)
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Direct determination of the ratio of unbound fraction in plasma to unbound fraction in microsomal system ( fu p/ fu mic) for refined prediction of phase I mediated metabolic hepatic clearance
Deshmukh, Sujal V., Harsch, Andreas
Published in Journal of pharmacological and toxicological methods (2011)
Published in Journal of pharmacological and toxicological methods (2011)
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Journal Article
Discovery of novel triazolobenzazepinones as γ-secretase modulators with central Aβ42 lowering in rodents and rhesus monkeys
Fischer, Christian, Zultanski, Susan L., Zhou, Hua, Methot, Joey L., Shah, Sanjiv, Hayashi, Ikuo, Hughes, Bethany L., Moxham, Christopher M., Bays, Nathan W., Smotrov, Nadya, Hill, Armetta D., Pan, Bo-Sheng, Wu, Zhenhua, Moy, Lily Y., Tanga, Flobert, Kenific, Candia, Cruz, Jonathan C., Walker, Deborah, Bouthillette, Melanie, Nikov, George N., Deshmukh, Sujal V., Jeliazkova-Mecheva, Valentina V., Diaz, Damaris, Michener, Maria S., Cook, Jacquelynn J., Munoz, Benito, Shearman, Mark S.
Published in Bioorganic & medicinal chemistry letters (01.09.2015)
Published in Bioorganic & medicinal chemistry letters (01.09.2015)
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siRNA-Mediated Knockdown of P450 Oxidoreductase in Rats: A Tool to Reduce Metabolism by CYPs and Increase Exposure of High Clearance Compounds
Burke, Rob S., Somasuntharam, Inthirai, Rearden, Paul, Brown, Duncan, Deshmukh, Sujal V., DiPietro, Martha A., DiMuzio, Jillian, Eisenhandler, Roy, Fauty, Scott E., Gibson, Christopher, Gindy, Marian E., Hamilton, Kelly A., Knemeyer, Ian, Koeplinger, Kenneth A., Kwon, Hae Won, Lifsted, Traci Q., Menzel, Karsten, Patel, Mihir, Pudvah, Nicole, Rudd, Deanne Jackson, Seitzer, Jessica, Strapps, Walter R., Prueksaritanont, Thomayant, Thompson, Charles D., Hochman, Jerome H., Carr, Brian A.
Published in Pharmaceutical research (01.12.2014)
Published in Pharmaceutical research (01.12.2014)
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Design of novel histone deacetylase inhibitors
Siliphaivanh, Phieng, Harrington, Paul, Witter, David J., Otte, Karin, Tempest, Paul, Kattar, Sam, Kral, Astrid M., Fleming, Judith C., Deshmukh, Sujal V., Harsch, Andreas, Secrist, Paul J., Miller, Thomas A.
Published in Bioorganic & medicinal chemistry letters (15.08.2007)
Published in Bioorganic & medicinal chemistry letters (15.08.2007)
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Journal Article
Methadone metabolism by human placenta
Nanovskaya, Tatiana N., Deshmukh, Sujal V., Nekhayeva, Ilona A., Zharikova, Olga L., Hankins, Gary D.V., Ahmed, Mahmoud S.
Published in Biochemical pharmacology (01.08.2004)
Published in Biochemical pharmacology (01.08.2004)
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Journal Article
The effect of methadone and buprenorphine on human placental aromatase
Zharikova, Olga L., Deshmukh, Sujal V., Nanovskaya, Tatiana N., Hankins, Gary D.V., Ahmed, Mahmoud S.
Published in Biochemical pharmacology (14.04.2006)
Published in Biochemical pharmacology (14.04.2006)
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