The development of β-selective glycosylation reactions with benzyl substituted 2-deoxy-1,4-dithio-D-erythro-pentofuranosides: enabling practical multi-gram syntheses of 4'-Thio-2'-deoxycytidine (T-dCyd) and 5-aza-4'-thio-2'-deoxycytidine (aza-T-dCyd) to support clinical development
Wishka, Donn G., Lopez, Omar D., Rudchenko, Vladimir F., Huang, Guangfei, Bahde, Robert, Kumar, Vineet, Denysenko, Sergiy M., Zhang, Lianhao, Zhang, Mianji, Teicher, Beverly A., Morris, Joel
Published in Nucleosides, nucleotides & nucleic acids (01.01.2021)
Published in Nucleosides, nucleotides & nucleic acids (01.01.2021)
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