Acetamide Scanning around Bicyclic Thiazoles: SAR at the H3 Receptor
Denonne , Frédéric, Célanire, Sylvain, Christophe, Bernard, Defays, Sabine, Delaunoy, Christel, Delporte, Marie-Laure, Detrait, Eric, Durieu, Véronique, Gillard, Michel, Lamberty, Yves, Lorent, Geneviève, Nicolas, Jean-Marie, Vanbellinghen, Alain, Van Houtvin, Nathalie, Provins, Laurent
Published in ChemMedChem (05.09.2011)
Published in ChemMedChem (05.09.2011)
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Journal Article
Towards the Synthesis of Azoacetylenes
Denonne, Frédéric, Seiler, Paul, Diederich, François
Published in Helvetica chimica acta (01.09.2003)
Published in Helvetica chimica acta (01.09.2003)
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8-Substituted 1,3-dimethyltetrahydropyrazino[2,1-f]purinediones: Water-soluble adenosine receptor antagonists and monoamine oxidase B inhibitors
Brunschweiger, Andreas, Koch, Pierre, Schlenk, Miriam, Rafehi, Muhammad, Radjainia, Hamid, Küppers, Petra, Hinz, Sonja, Pineda, Felipe, Wiese, Michael, Hockemeyer, Jörg, Heer, Jag, Denonne, Frédéric, Müller, Christa E.
Published in Bioorganic & medicinal chemistry (01.11.2016)
Published in Bioorganic & medicinal chemistry (01.11.2016)
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Journal Article
Acetamide Scanning around Bicyclic Thiazoles: SAR at the H 3 Receptor
Denonne , Frédéric, Célanire, Sylvain, Christophe, Bernard, Defays, Sabine, Delaunoy, Christel, Delporte, Marie‐Laure, Detrait, Eric, Durieu, Véronique, Gillard, Michel, Lamberty, Yves, Lorent, Geneviève, Nicolas, Jean‐Marie, Vanbellinghen, Alain, Van Houtvin, Nathalie, Provins, Laurent
Published in ChemMedChem (05.09.2011)
Published in ChemMedChem (05.09.2011)
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Journal Article
Lead Optimization of Thiazolo[5,4-c]piperidines: 3-Cyclobutoxy Linker as a Key Spacer for H3R Inverse Agonists
Provins, Laurent, Denonne, Frédéric, Célanire, Sylvain, Christophe, Bernard, Defays, Sabine, Delaunoy, Christel, Delporte, Marie-Laure, Demaude, Thierry, Durieu, Véronique, Gillard, Michel, Hubert, Delphine, Lamberty, Yves, Lorent, Geneviève, Valade, Anne, Vanbellinghen, Alain, Van houtvin, Nathalie
Published in ChemMedChem (01.12.2012)
Published in ChemMedChem (01.12.2012)
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Journal Article
Phenyl‐oxazoles, a New Family of Inverse Agonists at the H 3 Histamine Receptor
Denonne, Frédéric, Atienzar, Franck, Célanire, Sylvain, Christophe, Bernard, Delannois, Frédérique, Delaunoy, Christel, Delporte, Marie‐Laure, Durieu, Véronique, Gillard, Michel, Lallemand, Bénédicte, Lamberty, Yves, Lorent, Geneviève, Vanbellinghen, Alain, Van houtvin, Nathalie, Verbois, Valérie, Provins, Laurent
Published in ChemMedChem (01.02.2010)
Published in ChemMedChem (01.02.2010)
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Journal Article
Discovery of new C3aR ligands. Part 1: Arginine derivatives
Denonne, Frédéric, Binet, Sophie, Burton, Maggi, Collart, Philippe, Dipesa, Alan, Ganguly, Tanmoy, Giannaras, Alexander, Kumar, Seema, Lewis, Timothy, Maounis, Florence, Nicolas, Jean-Marie, Mansley, Tamsin, Pasau, Patrick, Preda, Dorin, Stebbins, Karin, Volosov, Alexander, Zou, Dong
Published in Bioorganic & medicinal chemistry letters (15.06.2007)
Published in Bioorganic & medicinal chemistry letters (15.06.2007)
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Journal Article
Studies of palladium-catalyzed coupling reactions for preparation of hindered 3-arylpyrroles relevant to (-)-rhazinilam and its analogues
Ghosez, Léon, Franc, Cécile, Denonne, Frédéric, Cuisinier, Claire, Touillaux, Roland
Published in Canadian journal of chemistry (01.11.2001)
Published in Canadian journal of chemistry (01.11.2001)
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Journal Article
Discovery of a New Class of Non‐imidazole Oxazoline‐Based Histamine H 3 Receptor (H 3 R) Inverse Agonists
Célanire, Sylvain, Wijtmans, Maikel, Christophe, Bernard, Collart, Philippe, de Esch, Iwan, Dassesse, Donald, Delaunoy, Christel, Denonne, Frédéric, Durieu, Véronique, Gelens, Edith, Gillard, Michel, Lallemand, Bénédicte, Lamberty, Yves, Lebon, Florence, Nicolas, Jean‐Marie, Quéré, Luc, Snip, Erwin, Vanbellinghen, Alain, Van houtvin, Nathalie, Verbois, Valérie, Timmerman, Henk, Talaga, Patrice, Leurs, Rob, Provins, Laurent
Published in ChemMedChem (06.07.2009)
Published in ChemMedChem (06.07.2009)
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Journal Article
Discovery of new C3aR ligands. Part 2: Amino-piperidine derivatives
Denonne, Frédéric, Binet, Sophie, Burton, Maggi, Collart, Philippe, Defays, Sabine, Dipesa, Alan, Eckert, Maria, Giannaras, Alexander, Kumar, Seema, Levine, Beth, Nicolas, Jean-Marie, Pasau, Patrick, Pégurier, Cécile, Preda, Dorin, Van houtvin, Nathalie, Volosov, Andrew, Zou, Dong
Published in Bioorganic & medicinal chemistry letters (15.06.2007)
Published in Bioorganic & medicinal chemistry letters (15.06.2007)
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Journal Article
Lead Optimization of Thiazolo[5,4‐ c ]piperidines: 3‐Cyclobutoxy Linker as a Key Spacer for H 3 R Inverse Agonists
Provins, Laurent, Denonne, Frédéric, Célanire, Sylvain, Christophe, Bernard, Defays, Sabine, Delaunoy, Christel, Delporte, Marie‐Laure, Demaude, Thierry, Durieu, Véronique, Gillard, Michel, Hubert, Delphine, Lamberty, Yves, Lorent, Geneviève, Valade, Anne, Vanbellinghen, Alain, Van houtvin, Nathalie
Published in ChemMedChem (01.12.2012)
Published in ChemMedChem (01.12.2012)
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Journal Article
Phenyl-oxazoles, a New Family of Inverse Agonists at the H3 Histamine Receptor
Denonne, Frédéric, Atienzar, Franck, Célanire, Sylvain, Christophe, Bernard, Delannois, Frédérique, Delaunoy, Christel, Delporte, Marie-Laure, Durieu, Véronique, Gillard, Michel, Lallemand, Bénédicte, Lamberty, Yves, Lorent, Geneviève, Vanbellinghen, Alain, Van houtvin, Nathalie, Verbois, Valérie, Provins, Laurent
Published in ChemMedChem (01.02.2010)
Published in ChemMedChem (01.02.2010)
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A general synthesis of 2-formyl-3-arylpyrroles
Franc, Cécile, Denonne, Frédéric, Cuisinier, Claire, Ghose, Léon
Published in Tetrahedron letters (11.06.1999)
Published in Tetrahedron letters (11.06.1999)
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Journal Article
Lead optimization of thiazolo[5,4-c]piperidines: 3-cyclobutoxy linker as a key spacer for H(3)R inverse agonists
Provins, Laurent, Denonne, Frédéric, Célanire, Sylvain, Christophe, Bernard, Defays, Sabine, Delaunoy, Christel, Delporte, Marie-Laure, Demaude, Thierry, Durieu, Véronique, Gillard, Michel, Hubert, Delphine, Lamberty, Yves, Lorent, Geneviève, Valade, Anne, Vanbellinghen, Alain, Van Houtvin, Nathalie
Published in ChemMedChem (01.12.2012)
Published in ChemMedChem (01.12.2012)
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Journal Article
Histamine H3 receptor ligands with a 3-cyclobutoxy motif: a novel and versatile constraint of the classical 3-propoxy linker
Wijtmans, Maikel, Denonne, Frédéric, Célanire, Sylvain, Gillard, Michel, Hulscher, Saskia, Delaunoy, Christel, Van houtvin, Nathalie, Bakker, Remko A., Defays, Sabine, Gérard, Julien, Grooters, Luc, Hubert, Delphine, Timmerman, Henk, Leurs, Rob, Talaga, Patrice, de Esch, Iwan J. P., Provins, Laurent
Published in MedChemComm (01.07.2010)
Published in MedChemComm (01.07.2010)
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Journal Article
Histamine H3 receptor ligands with a 3-cyclobutoxy motif: a novel and versatile constraint of the classical 3-propoxy linkerElectronic supplementary information (ESI) available: Gradient programs, compound purities, pharmacological procedures, computational studies, synthetic procedures and NMR spectra. See DOI: 10.1039/c0md00056f
Wijtmans, Maikel, Denonne, Frédéric, Célanire, Sylvain, Gillard, Michel, Hulscher, Saskia, Delaunoy, Christel, Van houtvin, Nathalie, Bakker, Remko A, Defays, Sabine, Gérard, Julien, Grooters, Luc, Hubert, Delphine, Timmerman, Henk, Leurs, Rob, Talaga, Patrice, de Esch, Iwan J. P, Provins, Laurent
Year of Publication 01.07.2010
Year of Publication 01.07.2010
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Journal Article
Discovery of a New Class of Non-imidazole Oxazoline-Based Histamine H3 Receptor (H3R) Inverse Agonists
Célanire, Sylvain, Wijtmans, Maikel, Christophe, Bernard, Collart, Philippe, de Esch, Iwan, Dassesse, Donald, Delaunoy, Christel, Denonne, Frédéric, Durieu, Véronique, Gelens, Edith, Gillard, Michel, Lallemand, Bénédicte, Lamberty, Yves, Lebon, Florence, Nicolas, Jean-Marie, Quéré, Luc, Snip, Erwin, Vanbellinghen, Alain, Van houtvin, Nathalie, Verbois, Valérie, Timmerman, Henk, Talaga, Patrice, Leurs, Rob, Provins, Laurent
Published in ChemMedChem (06.07.2009)
Published in ChemMedChem (06.07.2009)
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Journal Article
Phenyl-oxazoles, a new family of inverse agonists at the H(3) histamine receptor
Denonne, Frédéric, Atienzar, Franck, Célanire, Sylvain, Christophe, Bernard, Delannois, Frédérique, Delaunoy, Christel, Delporte, Marie-Laure, Durieu, Véronique, Gillard, Michel, Lallemand, Bénédicte, Lamberty, Yves, Lorent, Geneviève, Vanbellinghen, Alain, Van Houtvin, Nathalie, Verbois, Valérie, Provins, Laurent
Published in ChemMedChem (01.02.2010)
Published in ChemMedChem (01.02.2010)
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Journal Article
Discovery of a new class of non-imidazole oxazoline-based histamine H(3) receptor (H(3)R) inverse agonists
Célanire, Sylvain, Wijtmans, Maikel, Christophe, Bernard, Collart, Philippe, de Esch, Iwan, Dassesse, Donald, Delaunoy, Christel, Denonne, Frédéric, Durieu, Véronique, Gelens, Edith, Gillard, Michel, Lallemand, Bénédicte, Lamberty, Yves, Lebon, Florence, Nicolas, Jean-Marie, Quéré, Luc, Snip, Erwin, Vanbellinghen, Alain, Van Houtvin, Nathalie, Verbois, Valérie, Timmerman, Henk, Talaga, Patrice, Leurs, Rob, Provins, Laurent
Published in ChemMedChem (01.07.2009)
Published in ChemMedChem (01.07.2009)
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Journal Article