Design, synthesis and biological evaluation of chrysin benzimidazole derivatives as potential anticancer agents
Wang, Zhe, Deng, Xiangping, Xiong, Shujuan, Xiong, Runde, Liu, Juan, Zou, Liu, Lei, Xiaoyong, Cao, Xuan, Xie, Zhizhong, Chen, Yanming, Liu, Yunmei, Zheng, Xing, Tang, Guotao
Published in Natural product research (17.12.2018)
Published in Natural product research (17.12.2018)
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Discovery of novel covalent selective estrogen receptor degraders against endocrine-resistant breast cancer
Wang, Yubo, Min, Jian, Deng, Xiangping, Feng, Tian, Hu, Hebing, Guo, Xinyi, Cheng, Yan, Xie, Baohua, Yang, Yu, Chen, Chun-Chi, Guo, Rey-Ting, Dong, Chune, Zhou, Hai-Bing
Published in Acta pharmaceutica Sinica. B (01.12.2023)
Published in Acta pharmaceutica Sinica. B (01.12.2023)
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Design, synthesis and biological evaluation of tryptamine salicylic acid derivatives as potential antitumor agents
Xiong, Runde, He, Dongxiu, Deng, Xiangping, Liu, Juan, Lei, Xiaoyong, Xie, Zhizhong, Cao, Xuan, Chen, Yanming, Peng, Junmei, Tang, Guotao
Published in MedChemComm (01.04.2019)
Published in MedChemComm (01.04.2019)
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FS-7 inhibits MGC-803 cells growth in vitro and in vivo via down-regulating glycolysis
Deng, Xiangping, Li, Zhongli, Xiong, Runde, Liu, Juan, Liu, Renbo, Peng, Junmei, Chen, Yanming, Lei, Xiaoyong, Cao, Xuan, Zheng, Xing, Xie, Zhizhong, Tang, Guotao
Published in Biomedicine & pharmacotherapy (01.01.2019)
Published in Biomedicine & pharmacotherapy (01.01.2019)
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pH regulators and their inhibitors in tumor microenvironment
Liao, Senyi, Wu, Guang, Xie, Zhizhong, Lei, Xiaoyong, Yang, Xiaoyan, Huang, Sheng, Deng, Xiangping, Wang, Zhe, Tang, Guotao
Published in European journal of medicinal chemistry (05.03.2024)
Published in European journal of medicinal chemistry (05.03.2024)
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Journal Article
Discovery of Novel Bicyclic Phenylselenyl-Containing Hybrids: An Orally Bioavailable, Potential, and Multiacting Class of Estrogen Receptor Modulators against Endocrine-Resistant Breast Cancer
Deng, Xiangping, Xie, Baohua, Li, Qiuzi, Xiao, Yuan, Hu, Zhiye, Deng, Xiaofei, Fang, Pingping, Dong, Chune, Zhou, Hai-Bing, Huang, Jian
Published in Journal of medicinal chemistry (09.06.2022)
Published in Journal of medicinal chemistry (09.06.2022)
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Journal Article
Application of wireless measurement technology in hydraulic turbine test
Deng, Xiangping, Wang, Xiuling, Liu, Zhiyuan
Published in IOP conference series. Earth and environmental science (01.09.2022)
Published in IOP conference series. Earth and environmental science (01.09.2022)
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Journal Article
Discovery of a Novel Class of PROTACs as Potent and Selective Estrogen Receptor α Degraders to Overcome Endocrine-Resistant Breast Cancer In Vitro and In Vivo
Xie, Baohua, Yin, Zhinang, Hu, Zhiye, Lv, Junhui, Du, Chuanqian, Deng, Xiangping, Huang, Yuan, Li, Qiuzi, Huang, Jian, Liang, Kaiwei, Zhou, Hai-Bing, Dong, Chune
Published in Journal of medicinal chemistry (25.05.2023)
Published in Journal of medicinal chemistry (25.05.2023)
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Journal Article
Identification of Novel Dual-Target Estrogen Receptor α Degraders with Tubulin Inhibitory Activity for the Treatment of Endocrine-Resistant Breast Cancer
Deng, Xiangping, Deng, Xiaofei, Ning, Wentao, Xin, Lilan, Li, Qiuzi, Hu, Zhiye, Xie, Baohua, Liang, Kaiwei, Min, Chang, Dong, Chune, Huang, Jian, Zhou, Hai-Bing
Published in Journal of medicinal chemistry (24.08.2023)
Published in Journal of medicinal chemistry (24.08.2023)
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Journal Article
Discovery of Novel ERα and Aromatase Dual-Targeting PROTAC Degraders to Overcome Endocrine-Resistant Breast Cancer
Xin, Lilan, Wang, Chao, Cheng, Yan, Wang, Hongli, Guo, Xinyi, Deng, Xiaofei, Deng, Xiangping, Xie, Baohua, Hu, Hankun, Min, Chang, Dong, Chune, Zhou, Hai-Bing
Published in Journal of medicinal chemistry (29.05.2024)
Published in Journal of medicinal chemistry (29.05.2024)
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Journal Article
A novel selective estrogen receptor degrader induces cell cycle arrest in breast cancer via ERα degradation and the autophagy-lysosome pathway
Zhou, Jiawei, Shen, Rong, Liu, Jing, Deng, Xiangping, Xin, Lilan, Zhou, Hai-Bing, Huang, Jian
Published in Bioorganic & medicinal chemistry (15.03.2023)
Published in Bioorganic & medicinal chemistry (15.03.2023)
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Journal Article
A pH-sensitive prodrug strategy to co-deliver DOX and TOS in TPGS nanomicelles for tumor therapy
Xiong, Shujuan, Wang, Zhe, Liu, Juan, Deng, Xiangping, Xiong, Runde, Cao, Xuan, Xie, Zhizhong, Lei, Xiaoyong, Chen, Yanming, Tang, Guotao
Published in Colloids and surfaces, B, Biointerfaces (01.01.2019)
Published in Colloids and surfaces, B, Biointerfaces (01.01.2019)
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Small-molecule modulators of tumor immune microenvironment
Zhang, Jing, Yu, Jia, Liu, Meijing, Xie, Zhizhong, Lei, Xiaoyong, Yang, Xiaoyan, Huang, Sheng, Deng, Xiangping, Wang, Zhe, Tang, Guotao
Published in Bioorganic chemistry (01.04.2024)
Published in Bioorganic chemistry (01.04.2024)
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Corrigendum to “Structure-guided identification of novel dual-targeting estrogen receptor α degraders with aromatase inhibitory activity for the treatment of endocrine-resistant breast cancer” [Eur. J. Med. Chem. 253 (2023) 115328]
Xin, Lilan, Min, Jian, Hu, Hebing, Li, Yuanyuan, Du, Chuanqian, Xie, Baohua, Cheng, Yan, Deng, Xiaofei, Deng, Xiangping, Shen, Kang, Huang, Jian, Chen, Chun-Chi, Guo, Rey-Ting, Dong, Chune, Zhou, Hai-Bing
Published in European journal of medicinal chemistry (05.10.2024)
Published in European journal of medicinal chemistry (05.10.2024)
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Journal Article
Recent advances in pyruvate dehydrogenase kinase inhibitors: Structures, inhibitory mechanisms and biological activities
Li, Yiyang, Xie, Zhizhong, Lei, Xiaoyong, Yang, Xiaoyan, Huang, Sheng, Yuan, Weixi, Deng, Xiangping, Wang, Zhe, Tang, Guotao
Published in Bioorganic chemistry (01.03.2024)
Published in Bioorganic chemistry (01.03.2024)
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Journal Article
Structure-guided identification of novel dual-targeting estrogen receptor α degraders with aromatase inhibitory activity for the treatment of endocrine-resistant breast cancer
Xin, Lilan, Min, Jian, Hu, Hebing, Li, Yuanyuan, Du, Chuanqian, Xie, Baohua, Cheng, Yan, Deng, Xiaofei, Deng, Xiangping, Shen, Kang, Huang, Jian, Chen, Chun-Chi, Guo, Rey-Ting, Dong, Chune, Zhou, Hai-Bing
Published in European journal of medicinal chemistry (05.05.2023)
Published in European journal of medicinal chemistry (05.05.2023)
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Journal Article
FB-15 inhibits MGC-803 cells growth by regulating energy metabolism
Deng, Xiangping, Pi, Yiyuan, Li, Zhongli, Xiong, Runde, Liu, Juan, Zhao, Jingduo, Xie, Zhizhong, Lei, Xiaoyong, Tang, Guotao
Published in Chemico-biological interactions (25.08.2020)
Published in Chemico-biological interactions (25.08.2020)
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Discovery of a Potential Multi-Target Anti-Tumor Agent via Structural Modification on Flavonoid
Deng, Xiangping, Zou, Yang, Liu, Renbo, Peng, Yijiao, Ouyang, Chenglin, Peng, Junmei, Lei, Xiaoyong, Xie, Zhizhong, Li, Chong, Tang, Guotao
Published in Polycyclic aromatic compounds (07.02.2023)
Published in Polycyclic aromatic compounds (07.02.2023)
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