Preclinical Activity of Eltrombopag (SB‐497115), an Oral, Nonpeptide Thrombopoietin Receptor Agonist
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Published in Stem cells (Dayton, Ohio) (01.02.2009)
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Discovery and characterization of a selective, nonpeptidyl thrombopoietin receptor agonist
Erickson-Miller, Connie L., DeLorme, Evelyne, Tian, Shin-Shay, Hopson, Christopher B., Stark, Kenneth, Giampa, Leslie, Valoret, Elizabeth I., Duffy, Kevin J., Luengo, Juan L., Rosen, Jon, Miller, Stephen G., Dillon, Susan B., Lamb, Peter
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Published in Experimental hematology (2005)
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Identification of a Pharmacophore for Thrombopoietic Activity of Small, Non-Peptidyl Molecules. 1. Discovery and Optimization of Salicylaldehyde Thiosemicarbazone Thrombopoietin Mimics
Duffy, Kevin J, Shaw, Anthony N, Delorme, Evelyne, Dillon, Susan B, Erickson-Miller, Connie, Giampa, Leslie, Huang, Yifang, Keenan, Richard M, Lamb, Peter, Liu, Nannan, Miller, Stephen G, Price, Alan T, Rosen, Jon, Smith, Heather, Wiggall, Kenneth J, Zhang, Lihua, Luengo, Juan I
Published in Journal of medicinal chemistry (15.08.2002)
Published in Journal of medicinal chemistry (15.08.2002)
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Identification of a Pharmacophore for Thrombopoietic Activity of Small, Non-Peptidyl Molecules. 2. Rational Design of Naphtho[1,2-d]imidazole Thrombopoietin Mimics
Duffy, Kevin J, Price, Alan T, Delorme, Evelyne, Dillon, Susan B, Duquenne, Celine, Erickson-Miller, Connie, Giampa, Leslie, Huang, Yifang, Keenan, Richard M, Lamb, Peter, Liu, Nannan, Miller, Stephen G, Rosen, Jon, Shaw, Anthony N, Smith, Heather, Wiggall, Kenneth J, Zhang, Lihua, Luengo, Juan I
Published in Journal of medicinal chemistry (15.08.2002)
Published in Journal of medicinal chemistry (15.08.2002)
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Role of glycosylation on the secretion and biological activity of erythropoietin
Delorme, Evelyne, Lorenzini, Tony, Giffin, James, Martin, Frank, Jacobsen, Frederick, Boone, Tom, Elliott, Steve
Published in Biochemistry (Easton) (01.10.1992)
Published in Biochemistry (Easton) (01.10.1992)
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Structural Requirements for Addition of O-Linked Carbohydrate to Recombinant Erythropoietin
Elliott, Steve, Bartley, Tim, Delorme, Evelyne, Derby, Pat, Hunt, Rob, Lorenzini, Tony, Parker, Vann, Rohde, Michael F, Stoney, Ken
Published in Biochemistry (Easton) (01.09.1994)
Published in Biochemistry (Easton) (01.09.1994)
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Discovery of SB-497115, a Small-Molecule Thrombopoietin (TPO) Receptor Agonist for the Treatment of Thrombocytopenia
Luengo, Juan I., Duffy, Kevin J., Shaw, Anthony N., Delorme, Evelyne, Wiggall, Kenneth J., Giampa, Leslie, Liu, Nannan, Smith, Heather, Tian, Shin-Shay, Miller, Stephen G., Keenan, Richard M., Rosen, Jon, Dillon, Susan B., Lamb, Peter, Erickson-Miller, Connie L.
Published in Blood (16.11.2004)
Published in Blood (16.11.2004)
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Determinants of promoter-specific activity by glucocorticoid receptor
Guido, E C, Delorme, E O, Clemm, D L, Stein, R B, Rosen, J, Miner, J N
Published in Molecular endocrinology (Baltimore, Md.) (01.10.1996)
Published in Molecular endocrinology (Baltimore, Md.) (01.10.1996)
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Isolation and characterization of conformation sensitive antierythropoietin monoclonal antibodies : Effect of disulfide bonds and carbohydrate on recombinant human erythropoietin structure
ELLIOTT, S, CHANG, D, DELORME, E, DUNN, C, EGRIE, J, GIFFIN, J, LORENZINI, T, TALBOT, C, HESTERGERG, L
Published in Blood (01.04.1996)
Published in Blood (01.04.1996)
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