Application of Azamulin to Determine the Contribution of CYP3A4/5 to Drug Metabolic Clearance Using Human Hepatocytes
Chanteux, Hugues, Rosa, Maria, Delatour, Claude, Nicolaï, Johan, Gillent, Eric, Dell’Aiera, Sylvie, Ungell, Anna-Lena
Published in Drug metabolism and disposition (01.09.2020)
Published in Drug metabolism and disposition (01.09.2020)
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(-)- N -3-Benzylphenobarbital Is Superior to Omeprazole and (+)- N -3-Benzylnirvanol as a CYP2C19 Inhibitor in Suspended Human Hepatocytes
Cuypers, Marie-Lynn, Chanteux, Hugues, Gillent, Eric, Bonnaillie, Pierre, Saunders, Kenneth, Beckers, Claire, Delatour, Claude, Dell'Aiera, Sylvie, Ungell, Anna-Lena, Nicolaï, Johan
Published in Drug metabolism and disposition (01.11.2020)
Published in Drug metabolism and disposition (01.11.2020)
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Assessment of cytochrome P450 (1A2, 2B6, 2C9 and 3A4) induction in cryopreserved human hepatocytes cultured in 48-well plates using the cocktail strategy
Gerin, Brigitte, Dell'Aiera, Sylvie, Richert, Lysiane, Smith, Steven, Chanteux, Hugues
Published in Xenobiotica (01.04.2013)
Published in Xenobiotica (01.04.2013)
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Discovery and Characterization of a Novel Series of Chloropyrimidines as Covalent Inhibitors of the Kinase MSK1
Hall, Adrian, Abendroth, Jan, Bolejack, Madison J., Ceska, Tom, Dell’Aiera, Sylvie, Ellis, Victoria, Fox, David, François, Cyril, Muruthi, Muigai M., Prével, Camille, Poullennec, Karine, Romanov, Sergei, Valade, Anne, Vanbellinghen, Alain, Yano, Jason, Geraerts, Martine
Published in ACS medicinal chemistry letters (14.07.2022)
Published in ACS medicinal chemistry letters (14.07.2022)
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Off-line solid phase extraction and liquid chromatography-tandem mass spectrometry method for the quantitation of brivaracetam acid metabolites: Method validation and application to in vitro metabolism assays
Bourgogne, Emmanuel, Culot, Benoit, Dell'Aiera, Sylvie, Chanteux, Hugues, Stockis, Armel, Nicolas, Jean-Marie
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (01.06.2018)
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (01.06.2018)
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