Readily Accessible Bicyclononynes for Bioorthogonal Labeling and Three-Dimensional Imaging of Living Cells
Dommerholt, Jan, Schmidt, Samuel, Temming, Rinske, Hendriks, Linda J.A, Rutjes, Floris P.J.T, van Hest, Jan C.M, Lefeber, Dirk J, Friedl, Peter, van Delft, Floris L
Published in Angewandte Chemie (International ed.) (03.12.2010)
Published in Angewandte Chemie (International ed.) (03.12.2010)
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Journal Article
Inducible, Site-Specific Protein Labeling by Tyrosine Oxidation–Strain-Promoted (4 + 2) Cycloaddition
Bruins, Jorick J, Westphal, Adrie H, Albada, Bauke, Wagner, Koen, Bartels, Lina, Spits, Hergen, van Berkel, Willem J. H, van Delft, Floris L
Published in Bioconjugate chemistry (19.04.2017)
Published in Bioconjugate chemistry (19.04.2017)
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Journal Article
High Rates of Quinone‐Alkyne Cycloaddition Reactions are Dictated by Entropic Factors
Damen, Johannes A. M., Escorihuela, Jorge, Zuilhof, Han, Delft, Floris L., Albada, Bauke
Published in Chemistry : a European journal (11.07.2023)
Published in Chemistry : a European journal (11.07.2023)
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Journal Article
Orthogonal, dual protein labelling by tandem cycloaddition of strained alkenes and alkynes to ortho-quinones and azides
Bruins, Jorick J, Blanco-Ania, Daniel, van der Doef, Vincent, van Delft, Floris L, Albada, Bauke
Published in Chemical communications (Cambridge, England) (2018)
Published in Chemical communications (Cambridge, England) (2018)
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Journal Article
Protein Modification by Strain-Promoted Alkyne-Nitrone Cycloaddition
Ning, Xinghai, Temming, Rinske P, Dommerholt, Jan, Guo, Jun, Ania, Daniel B, Debets, Marjoke F, Wolfert, Margreet A, Boons, Geert-Jan, van Delft, Floris L
Published in Angewandte Chemie (International ed.) (12.04.2010)
Published in Angewandte Chemie (International ed.) (12.04.2010)
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Journal Article
Organophosphorus Catalysis to Bypass Phosphine Oxide Waste
van Kalkeren, Henri A., van Delft, Floris L., Rutjes, Floris P. J. T.
Published in ChemSusChem (01.09.2013)
Published in ChemSusChem (01.09.2013)
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Journal Article
Chemoenzymatic Conjugation of Toxic Payloads to the Globally Conserved N‑Glycan of Native mAbs Provides Homogeneous and Highly Efficacious Antibody–Drug Conjugates
van Geel, Remon, Wijdeven, Marloes A, Heesbeen, Ryan, Verkade, Jorge M. M, Wasiel, Anna A, van Berkel, Sander S, van Delft, Floris L
Published in Bioconjugate chemistry (18.11.2015)
Published in Bioconjugate chemistry (18.11.2015)
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Journal Article
Strain-Promoted 1,3-Dipolar Cycloaddition of Cycloalkynes and Organic Azides
Dommerholt, Jan, Rutjes, Floris P. J. T., van Delft, Floris L.
Published in Topics in current chemistry (2016) (01.04.2016)
Published in Topics in current chemistry (2016) (01.04.2016)
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Journal Article
Ultrathin Covalently Bound Organic Layers on Mica: Formation of Atomically Flat Biofunctionalizable Surfaces
Sen, Rickdeb, Gahtory, Digvijay, Carvalho, Rui Rijo, Albada, Bauke, van Delft, Floris L., Zuilhof, Han
Published in Angewandte Chemie (International ed.) (03.04.2017)
Published in Angewandte Chemie (International ed.) (03.04.2017)
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Journal Article
Aza-dibenzocyclooctynes for fast and efficient enzyme PEGylation via copper-free (3+2) cycloaddition
Debets, Marjoke F., van Berkel, Sander S., Schoffelen, Sanne, Rutjes, Floris P. J. T., van Hest, Jan C. M., van Delft, Floris L.
Published in Chemical communications (Cambridge, England) (01.01.2010)
Published in Chemical communications (Cambridge, England) (01.01.2010)
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Journal Article
Radiolabeled CCK/gastrin peptides for imaging and therapy of CCK2 receptor-expressing tumors
Roosenburg, Susan, Laverman, Peter, van Delft, Floris L., Boerman, Otto C.
Published in Amino acids (01.11.2011)
Published in Amino acids (01.11.2011)
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Journal Article
A common sugar-nucleotide-mediated mechanism of inhibition of (glycosamino)glycan biosynthesis, as evidenced by 6F-GalNAc (Ac3)
van Wijk, Xander M, Lawrence, Roger, Thijssen, Victor L, van den Broek, Sebastiaan A, Troost, Ran, van Scherpenzeel, Monique, Naidu, Natasha, Oosterhof, Arie, Griffioen, Arjan W, Lefeber, Dirk J, van Delft, Floris L, van Kuppevelt, Toin H
Published in The FASEB journal (01.07.2015)
Published in The FASEB journal (01.07.2015)
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Journal Article
Targeting aberrant sialylation in cancer cells using a fluorinated sialic acid analog impairs adhesion, migration, and in vivo tumor growth
Büll, Christian, Boltje, Thomas J, Wassink, Melissa, de Graaf, Annemarie M A, van Delft, Floris L, den Brok, Martijn H, Adema, Gosse J
Published in Molecular cancer therapeutics (01.10.2013)
Published in Molecular cancer therapeutics (01.10.2013)
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Journal Article
Enzymatic strategies for (near) clinical development of antibody-drug conjugates
van Berkel, Sander S., van Delft, Floris L.
Published in Drug discovery today. Technologies (01.12.2018)
Published in Drug discovery today. Technologies (01.12.2018)
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Journal Article
Genetic Encoding of a Bicyclo[6.1.0]nonyne-Charged Amino Acid Enables Fast Cellular Protein Imaging by Metal-Free Ligation
Borrmann, Annika, Milles, Sigrid, Plass, Tilman, Dommerholt, Jan, Verkade, Jorge M. M., Wießler, Manfred, Schultz, Carsten, van Hest, Jan C. M., van Delft, Floris L., Lemke, Edward A.
Published in Chembiochem : a European journal of chemical biology (24.09.2012)
Published in Chembiochem : a European journal of chemical biology (24.09.2012)
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Journal Article