An improved method for specific and quantitative determination of the clopidogrel active metabolite isomers in human plasma
Tuffal, Gilles, Roy, Sebastien, Lavisse, Melanie, Brasseur, Denis, Schofield, Joe, Delesque Touchard, Nathalie, Savi, Pierre, Bremond, Nicolas, Rouchon, Marie-Claude, Hurbin, Fabrice, Sultan, Eric
Published in Thrombosis and haemostasis (01.04.2011)
Published in Thrombosis and haemostasis (01.04.2011)
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Journal Article
The Active Metabolite of Clopidogrel Disrupts P2Y12 Receptor Oligomers and Partitions Them out of Lipid Rafts
Savi, Pierre, Zachayus, Jean-Luc, Delesque-Touchard, Nathalie, Labouret, Catherine, Hervé, Caroline, Uzabiaga, Marie-Françoise, Pereillo, Jean-Marie, Culouscou, Jean-Michel, Bono, Françoise, Ferrara, Pascual, Herbert, Jean-Marc
Published in Proceedings of the National Academy of Sciences - PNAS (18.07.2006)
Published in Proceedings of the National Academy of Sciences - PNAS (18.07.2006)
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Journal Article
Regulator of G-protein signaling 18 controls both platelet generation and function
Delesque-Touchard, Nathalie, Pendaries, Caroline, Volle-Challier, Cécile, Millet, Laurence, Salel, Véronique, Hervé, Caroline, Pflieger, Anne-Marie, Berthou-Soulie, Laurence, Prades, Catherine, Sorg, Tania, Herbert, Jean-Marc, Savi, Pierre, Bono, Françoise
Published in PloS one (18.11.2014)
Published in PloS one (18.11.2014)
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Journal Article
Gas6 promotes inflammation by enhancing interactions between endothelial cells, platelets, and leukocytes
Tjwa, Marc, Bellido-Martin, Lola, Lin, Yuan, Lutgens, Esther, Plaisance, Stéphane, Bono, Françoise, Delesque-Touchard, Nathalie, Hervé, Caroline, Moura, Rute, Billiau, An D., Aparicio, Cristina, Levi, Marcel, Daemen, Mat, Dewerchin, Mieke, Lupu, Florea, Arnout, Jef, Herbert, Jean-Marc, Waer, Mark, García de Frutos, Pablo, Dahlbäck, Björn, Carmeliet, Peter, Hoylaerts, Marc F., Moons, Lieve
Published in Blood (15.04.2008)
Published in Blood (15.04.2008)
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Journal Article
A new synthetic FGF receptor antagonist inhibits arteriosclerosis in a mouse vein graft model and atherosclerosis in apolipoprotein E-deficient mice
Dol-Gleizes, Frédérique, Delesque-Touchard, Nathalie, Marès, Anne-Marie, Nestor, Anne-Laure, Schaeffer, Paul, Bono, Françoise
Published in PloS one (04.11.2013)
Published in PloS one (04.11.2013)
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Journal Article
The Tyrosine Phosphatase SHP-1 Associates with the sst2 Somatostatin Receptor and Is an Essential Component of sst2-mediated Inhibitory Growth Signaling
Lopez, Frédéric, Estève, Jean-Pierre, Buscail, Louis, Delesque, Nathalie, Saint-Laurent, Nathalie, Théveniau, Magali, Nahmias, Clara, Vaysse, Nicole, Susini, Christiane
Published in The Journal of biological chemistry (26.09.1997)
Published in The Journal of biological chemistry (26.09.1997)
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Journal Article
Characterization of the Antiproliferative Signal Mediated by the Somatostatin Receptor Subtype sst5
Cordelier, Pierre, Esteve, Jean-Pierre, Bousquet, Corinne, Delesque, Nathalie, O'Carroll, Anne-Marie, Schally, Andrew V., Vaysse, Nicole, Susini, Christiane, Buscail, Louis
Published in Proceedings of the National Academy of Sciences - PNAS (19.08.1997)
Published in Proceedings of the National Academy of Sciences - PNAS (19.08.1997)
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Journal Article
sst2 Somatostatin Receptor Mediates Negative Regulation of Insulin Receptor Signaling through the Tyrosine Phosphatase SHP-1
Bousquet, C, Delesque, N, Lopez, F, Saint-Laurent, N, Estève, J P, Bedecs, K, Buscail, L, Vaysse, N, Susini, C
Published in The Journal of biological chemistry (20.03.1998)
Published in The Journal of biological chemistry (20.03.1998)
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Journal Article
Aflibercept exhibits VEGF binding stoichiometry distinct from bevacizumab and does not support formation of immune-like complexes
MacDonald, Douglas A., Martin, Joel, Muthusamy, Kathir K., Luo, Jiann-Kae, Pyles, Erica, Rafique, Ashique, Huang, Tammy, Potocky, Terra, Liu, Yang, Cao, Jingtai, Bono, Françoise, Delesque, Nathalie, Savi, Pierre, Francis, John, Amirkhosravi, Ali, Meyer, Todd, Romano, Carmelo, Glinka, Meredith, Yancopoulos, George D., Stahl, Neil, Wiegand, Stanley J., Papadopoulos, Nicholas
Published in Angiogenesis (London) (01.07.2016)
Published in Angiogenesis (London) (01.07.2016)
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Journal Article
N‑[6-(4-Butanoyl-5-methyl‑1H‑pyrazol-1-yl)pyridazin-3-yl]-5-chloro-1-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]‑1H‑indole-3-carboxamide (SAR216471), a Novel Intravenous and Oral, Reversible, and Directly Acting P2Y12 Antagonist
Boldron, Christophe, Besse, Angélina, Bordes, Marie-Françoise, Tissandié, Stéphanie, Yvon, Xavier, Gau, Benjamin, Badorc, Alain, Rousseaux, Tristan, Barré, Guillaume, Meneyrol, Jérôme, Zech, Gernot, Nazare, Marc, Fossey, Valérie, Pflieger, Anne-Marie, Bonnet-Lignon, Sandrine, Millet, Laurence, Briot, Christophe, Dol, Frédérique, Hérault, Jean-Pascal, Savi, Pierre, Lassalle, Gilbert, Delesque, Nathalie, Herbert, Jean-Marc, Bono, Françoise
Published in Journal of medicinal chemistry (11.09.2014)
Published in Journal of medicinal chemistry (11.09.2014)
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N -[6-(4-Butanoyl-5-methyl-1 H -pyrazol-1-yl)pyridazin-3-yl]-5-chloro-1-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-1 H -indole-3-carboxamide (SAR216471), a Novel Intravenous and Oral, Reversible, and Directly Acting P2Y12 Antagonist
Boldron, Christophe, Besse, Angélina, Bordes, Marie-Françoise, Tissandié, Stéphanie, Yvon, Xavier, Gau, Benjamin, Badorc, Alain, Rousseaux, Tristan, Barré, Guillaume, Meneyrol, Jérôme, Zech, Gernot, Nazare, Marc, Fossey, Valérie, Pflieger, Anne-Marie, Bonnet-Lignon, Sandrine, Millet, Laurence, Briot, Christophe, Dol, Frédérique, Hérault, Jean-Pascal, Savi, Pierre, Lassalle, Gilbert, Delesque, Nathalie, Herbert, Jean-Marc, Bono, Françoise
Published in Journal of medicinal chemistry (11.09.2014)
Published in Journal of medicinal chemistry (11.09.2014)
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A novel inhibitor of p75-neurotrophin receptor improves functional outcomes in two models of traumatic brain injury
Delbary-Gossart, Sandrine, Lee, Sangmi, Baroni, Marco, Lamarche, Isabelle, Arnone, Michele, Canolle, Benoit, Lin, Amity, Sacramento, Jeffrey, Salegio, Ernesto A, Castel, Marie-Noelle, Delesque-Touchard, Nathalie, Alam, Antoine, Laboudie, Patricia, Ferzaz, Badia, Savi, Pierre, Herbert, Jean-Marc, Manley, Geoffrey T, Ferguson, Adam R, Bresnahan, Jacqueline C, Bono, Françoise, Beattie, Michael S
Published in Brain (London, England : 1878) (01.06.2016)
Published in Brain (London, England : 1878) (01.06.2016)
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VEGF-R2 and neuropilin-1 are involved in VEGF-A-induced differentiation of human bone marrow progenitor cells
Fons, Pierre, Herault, Jean-Pascal, Delesque, Nathalie, Tuyaret, Joēl, Bono, Françoise, Herbert, Jean-Marc
Published in Journal of cellular physiology (01.09.2004)
Published in Journal of cellular physiology (01.09.2004)
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Journal Article
Stimulation of Tyrosine Phosphatase and Inhibition of Cell Proliferation by Somatostatin Analogues: Mediation by Human Somatostatin Receptor Subtypes SSTR1 and SSTR2
Buscail, Louis, Delesque, Nathalie, Esteve, Jean-Pierre, Saint-Laurent, Nathalie, Prats, Herve, Clerc, Pascal, Robberecht, Patrick, Bell, Graeme I., Liebow, Charles, Schally, Andrew V., Vaysse, Nicole, Susini, Christiane
Published in Proceedings of the National Academy of Sciences - PNAS (15.03.1994)
Published in Proceedings of the National Academy of Sciences - PNAS (15.03.1994)
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sst2 somatostatin receptor expression reverses tumorigenicity of human pancreatic cancer cells
DELESQUE, N, BUSCAIL, L, ESTEVE, J.-P, SAINT-LAURENT, N, MÜLLER, C, WECKBECKER, G, BRUNS, C, VAYSSE, N, SUSINI, C
Published in Cancer research (Chicago, Ill.) (01.03.1997)
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Published in Cancer research (Chicago, Ill.) (01.03.1997)
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Abstract CT206: EVT801, a novel selective VEGFR-3 inhibitor targeting tumor angiogenesis, started enrollment for its phase I first-in-human study
Gomez roca, Carlos, Cassier, Philippe, Mandron, Marie, Estrabaut, Myriam, Delesque-Touchard, Nathalie, Smith, Adam C., Klawitter, Amy, Gentry, Leesa, Fons, Pierre, Paillasse, Michael R., Davenne, Lise, Fitzgerald, Michael, Garner, James, Delord, Jean-Pierre
Published in Cancer research (Chicago, Ill.) (15.06.2022)
Published in Cancer research (Chicago, Ill.) (15.06.2022)
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DERIVATIVES OF N- [( 1H - PYRAZOL - 1 - YL) ARYL] - 1H - INDOLE OR 1H - INDAZOLE - 3 - CARBOXAMIDE, THEIR PREPARATION AND THEIR USE AS P2Y12 ANTAGONISTS
LASSALLE, GILBERT, BOLDRON, CHRISTOPHE, FOSSEY, VALERIE, YVON, XAVIER, BADORC, ALAIN, DELESQUE, NATHALIE
Year of Publication 26.02.2019
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Year of Publication 26.02.2019
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