Locked 2′-Deoxy-2′,4′-Difluororibo Modified Nucleic Acids: Thermal Stability, Structural Studies, and siRNA Activity
Martínez-Montero, Saúl, Deleavey, Glen F, Martín-Pintado, Nerea, Fakhoury, Johans F, González, Carlos, Damha, Masad J
Published in ACS chemical biology (18.09.2015)
Published in ACS chemical biology (18.09.2015)
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Synergistic effects between analogs of DNA and RNA improve the potency of siRNA-mediated gene silencing
Deleavey, Glen F, Watts, Jonathan K, Alain, Tommy, Robert, Francis, Kalota, Anna, Aishwarya, Veenu, Pelletier, Jerry, Gewirtz, Alan M, Sonenberg, Nahum, Damha, Masad J
Published in Nucleic acids research (01.07.2010)
Published in Nucleic acids research (01.07.2010)
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Synthesis and Properties of 2′-Deoxy-2′,4′-difluoroarabinose-Modified Nucleic Acids
Martínez-Montero, Saúl, Deleavey, Glen F, Dierker-Viik, Arden, Lindovska, Petra, Ilina, Tatiana, Portella, Guillem, Orozco, Modesto, Parniak, Michael A, González, Carlos, Damha, Masad J
Published in Journal of organic chemistry (20.03.2015)
Published in Journal of organic chemistry (20.03.2015)
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Journal Article
Click conjugated polymeric immuno-nanoparticles for targeted siRNA and antisense oligonucleotide delivery
Chan, Dianna P.Y, Deleavey, Glen F, Owen, Shawn C, Damha, Masad J, Shoichet, Molly S
Published in Biomaterials (01.11.2013)
Published in Biomaterials (01.11.2013)
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Antisense 2′-Deoxy, 2′-Fluoroarabino Nucleic Acid (2′F-ANA) Oligonucleotides: In Vitro Gymnotic Silencers of Gene Expression Whose Potency Is Enhanced by Fatty Acids
Souleimanian, Naira, Deleavey, Glen F, Soifer, Harris, Wang, Sijian, Tiemann, Katrin, Damha, Masad J, Stein, Cy A
Published in Molecular therapy. Nucleic acids (2012)
Published in Molecular therapy. Nucleic acids (2012)
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Phenylpyrrolocytosine as an Unobtrusive Base Modification for Monitoring Activity and Cellular Trafficking of siRNA
Wahba, Alexander S, Azizi, Fereshteh, Deleavey, Glen F, Brown, Claire, Robert, Francis, Carrier, Marilyn, Kalota, Anna, Gewirtz, Alan M, Pelletier, Jerry, Hudson, Robert H. E, Damha, Masad J
Published in ACS chemical biology (16.09.2011)
Published in ACS chemical biology (16.09.2011)
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Chemically modified siRNA: tools and applications
Watts, Jonathan K., Deleavey, Glen F., Damha, Masad J.
Published in Drug discovery today (01.10.2008)
Published in Drug discovery today (01.10.2008)
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Dramatic Effect of Furanose C2′ Substitution on Structure and Stability: Directing the Folding of the Human Telomeric Quadruplex with a Single Fluorine Atom
Martín-Pintado, Nerea, Yahyaee-Anzahaee, Maryam, Deleavey, Glen F, Portella, Guillem, Orozco, Modesto, Damha, Masad J, González, Carlos
Published in Journal of the American Chemical Society (10.04.2013)
Published in Journal of the American Chemical Society (10.04.2013)
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Journal Article
Rigid 2 ',4 '-Difluororibonucleosides: Synthesis, Conformational Analysis, and Incorporation into Nascent RNA by HCV Polymerase
Martinez-Montero, Saul, Deleavey, Glen F., Kulkarni, Anupriya, Martin-Pintado, Nerea, Lindovska, Petra, Thomson, Michael, Gonzalez, Carlos, Goette, Matthias, Damha, Masad J.
Published in Journal of organic chemistry (20.06.2014)
Published in Journal of organic chemistry (20.06.2014)
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Allele-Selective Inhibition of Mutant Huntingtin Expression with Antisense Oligonucleotides Targeting the Expanded CAG Repeat
Gagnon, Keith T, Pendergraff, Hannah M, Deleavey, Glen F, Swayze, Eric E, Potier, Pierre, Randolph, John, Roesch, Eric B, Chattopadhyaya, Jyoti, Damha, Masad J, Bennett, C. Frank, Montaillier, Christophe, Lemaitre, Marc, Corey, David R
Published in Biochemistry (Easton) (30.11.2010)
Published in Biochemistry (Easton) (30.11.2010)
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Journal Article
siRNA nanocarriers based on methacrylic acid copolymers
Felber, Arnaud E., Castagner, Bastien, Elsabahy, Mahmoud, Deleavey, Glen F., Damha, Masad J., Leroux, Jean-Christophe
Published in Journal of controlled release (30.05.2011)
Published in Journal of controlled release (30.05.2011)
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Conference Proceeding
The interactions of amphiphilic antisense oligonucleotides with serum proteins and their effects on in vitro silencing activity
Felber, Arnaud E, Bayó-Puxan, Núria, Deleavey, Glen F, Castagner, Bastien, Damha, Masad J, Leroux, Jean-Christophe
Published in Biomaterials (01.09.2012)
Published in Biomaterials (01.09.2012)
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Journal Article
Nucleotide Sugar Pucker Preference Mitigates Excision by HIV‑1 RT
Yamada, Ken, Wahba, Alexander S, Bernatchez, Jean A, Ilina, Tatiana, Martínez-Montero, Saúl, Habibian, Maryam, Deleavey, Glen F, Götte, Matthias, Parniak, Michael A, Damha, Masad J
Published in ACS chemical biology (18.09.2015)
Published in ACS chemical biology (18.09.2015)
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Journal Article
Arabinonucleic Acids: 2′-Stereoisomeric Modulators of siRNA Activity
Anzahaee, Maryam Yahyaee, Deleavey, Glen F., Le, Phuong Uyen, Fakhoury, Johans, Petrecca, Kevin, Damha, Masad J.
Published in Nucleic acid therapeutics (01.10.2014)
Published in Nucleic acid therapeutics (01.10.2014)
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Journal Article
Chemical modification of siRNA
Deleavey, Glen F, Watts, Jonathan K, Damha, Masad J
Published in Current protocols in nucleic acid chemistry (01.12.2009)
Published in Current protocols in nucleic acid chemistry (01.12.2009)
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