Novel Class of Benzoic Acid Ester Derivatives as Potent PDE4 Inhibitors for Inhaled Administration in the Treatment of Respiratory Diseases
Armani, Elisabetta, Amari, Gabriele, Rizzi, Andrea, Fanti, Renato De, Ghidini, Eleonora, Capaldi, Carmelida, Carzaniga, Laura, Caruso, Paola, Guala, Matilde, Peretto, Ilaria, La Porta, Elena, Bolzoni, Pier T, Facchinetti, Fabrizio, Carnini, Chiara, Moretto, Nadia, Patacchini, Riccardo, Bassani, Franco, Cenacchi, Valentina, Volta, Roberta, Amadei, Francesco, Capacchi, Silvia, Delcanale, Maurizio, Puccini, Paola, Catinella, Silvia, Civelli, Maurizio, Villetti, Gino
Published in Journal of medicinal chemistry (13.02.2014)
Published in Journal of medicinal chemistry (13.02.2014)
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Journal Article
Pharmacological Actions of a Novel, Potent, Tissue-Selective Benzopyran Estrogen
Galbiati, Elisabetta, Caruso, Paola Lorenza, Amari, Gabriele, Armani, Elisabetta, Ghirardi, Silvia, Delcanale, Maurizio, Civelli, Maurizio
Published in The Journal of pharmacology and experimental therapeutics (01.10.2002)
Published in The Journal of pharmacology and experimental therapeutics (01.10.2002)
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Journal Article
Effects of 3-Phenyl-4-[[4-[2-(1-piperidinyl)ethoxy]phenyl]methyl]- 2H-1-benzopyran-7-ol (CHF 4056), a Novel Nonsteroidal Estrogen Agonist/Antagonist, on Reproductive and Nonreproductive Tissue
Galbiati, Elisabetta, Caruso, Paola Lorenza, Amari, Gabriele, Armani, Elisabetta, Ghirardi, Silvia, Delcanale, Maurizio, Civelli, Maurizio
Published in The Journal of pharmacology and experimental therapeutics (01.03.2002)
Published in The Journal of pharmacology and experimental therapeutics (01.03.2002)
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Journal Article
Optimization of M3 Antagonist–PDE4 Inhibitor (MAPI) Dual Pharmacology Molecules for the Treatment of COPD
Rizzi, Andrea, Amari, Gabriele, Pivetti, Fausto, Delcanale, Maurizio, Amadei, Francesco, Pappani, Alice, Fornasari, Luca, Villetti, Gino, Marchini, Gessica, Pisano, Anna Rita, Pitozzi, Vanessa, Pittelli, Maria Gloria, Trevisani, Marcello, Salvadori, Michela, Cenacchi, Valentina, Fioni, Alessandro, Puccini, Paola, Civelli, Maurizio, Patacchini, Riccardo, Baker-Glenn, Charles, Van de Poël, Hervé, Blackaby, Wesley, Nash, Kevin, Armani, Elisabetta
Published in Journal of medicinal chemistry (24.08.2023)
Published in Journal of medicinal chemistry (24.08.2023)
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Journal Article
Discovery of Clinical Candidate CHF-6366: A Novel Super-soft Dual Pharmacology Muscarinic Antagonist and beta(2) Agonist (MABA) for the Inhaled Treatment of Respiratory Diseases
Carzaniga, Laura, Linney, Ian D., Rizzi, Andrea, Delcanale, Maurizio, Schmidt, Wolfgang, Knight, Christopher K., Pastore, Fiorella, Miglietta, Daniela, Carnini, Chiara, Cesari, Nicola, Riccardi, Benedetta, Mileo, Valentina, Venturi, Luca, Moretti, Elisa, Blackaby, Wesley P., Patacchini, Riccardo, Accetta, Alessandro, Biagetti, Matteo, Bassani, Franco, Tondelli, Marina, Murgo, Annalisa, Battipaglia, Loredana, Villetti, Gino, Puccini, Paola, Catinella, Silvia, Civelli, Maurizio, Rancati, Fabio
Published in Journal of medicinal chemistry (11.08.2022)
Published in Journal of medicinal chemistry (11.08.2022)
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Journal Article
Discovery of a Potent, Selective, and Orally Bioavailable Tool Compound for Probing the Role of Lysophosphatidic Acid Type 2 Receptor Antagonists in Fibrotic Disorders
Armani, Elisabetta, Rizzi, Andrea, Iotti, Nicolò, Saccani, Francesca, Di Lascia, Maria Rosaria, Tigli, Laura, Pappani, Alice, Marchini, Gessica, Murgo, Annalisa, Capelli, Anna Maria, Delcanale, Maurizio, Puccini, Paola, Villetti, Gino, Civelli, Maurizio, Beato, Claudia, Giuliani, Marta, Mundi, Claudia, Murarolli, Francesca, Pagano, Mafalda, Raveglia, Luca F., Remelli, Rosaria, Amari, Gabriele
Published in Journal of medicinal chemistry (27.04.2023)
Published in Journal of medicinal chemistry (27.04.2023)
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Journal Article
Optimization of M 3 Antagonist-PDE4 Inhibitor (MAPI) Dual Pharmacology Molecules for the Treatment of COPD
Rizzi, Andrea, Amari, Gabriele, Pivetti, Fausto, Delcanale, Maurizio, Amadei, Francesco, Pappani, Alice, Fornasari, Luca, Villetti, Gino, Marchini, Gessica, Pisano, Anna Rita, Pitozzi, Vanessa, Pittelli, Maria Gloria, Trevisani, Marcello, Salvadori, Michela, Cenacchi, Valentina, Fioni, Alessandro, Puccini, Paola, Civelli, Maurizio, Patacchini, Riccardo, Baker-Glenn, Charles, Van de Poël, Hervé, Blackaby, Wesley, Nash, Kevin, Armani, Elisabetta
Published in Journal of medicinal chemistry (24.08.2023)
Published in Journal of medicinal chemistry (24.08.2023)
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Journal Article
Discovery of a novel class of inhaled dual pharmacology muscarinic antagonist and beta 2 agonist (MABA) for the treatment of chronic obstructive pulmonary disease (COPD)
Rancati, Fabio, Linney, Ian D., Rizzi, Andrea, Delcanale, Maurizio, Knight, Chris K., Schmidt, Wolfgang, Pastore, Fiorella, Riccardi, Benedetta, Mileo, Valentina, Carnini, Chiara, Cesari, Nicola, Blackaby, Wesley P., Patacchini, Riccardo, Carzaniga, Laura
Published in Bioorganic & medicinal chemistry letters (01.06.2021)
Published in Bioorganic & medicinal chemistry letters (01.06.2021)
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Journal Article
Design, Synthesis, and Biological Characterization of Inhaled p38?/? MAPK Inhibitors for the Treatment of Lung Inflammatory Diseases
Armani, Elisabetta, Capaldi, Carmelida, Bagnacani, Valentina, Saccani, Francesca, Aquino, Giancarlo, Puccini, Paola, Facchinetti, Fabrizio, Martucci, Cataldo, Moretto, Nadia, Villetti, Gino, Patacchini, Riccardo, Civelli, Maurizio, Hurley, Chris, Jennings, Andrew, Alcaraz, Lilian, Bloomfield, Dawn, Briggs, Michael, Daly, Stephen, Panchal, Terry, Russell, Vince, Wicks, Sharon, Finch, Harry, Fitzgerald, Mary, Fox, Craig, Delcanale, Maurizio
Published in Journal of medicinal chemistry (26.05.2022)
Published in Journal of medicinal chemistry (26.05.2022)
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Journal Article
Discovery of a novel class of inhaled dual pharmacology muscarinic antagonist and β2 agonist (MABA) for the treatment of chronic obstructive pulmonary disease (COPD)
Rancati, Fabio, Linney, Ian D., Rizzi, Andrea, Delcanale, Maurizio, Knight, Chris K., Schmidt, Wolfgang, Pastore, Fiorella, Riccardi, Benedetta, Mileo, Valentina, Carnini, Chiara, Cesari, Nicola, Blackaby, Wesley P., Patacchini, Riccardo, Carzaniga, Laura
Published in Bioorganic & medicinal chemistry letters (01.06.2021)
Published in Bioorganic & medicinal chemistry letters (01.06.2021)
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Journal Article
Discovery of Clinical Candidate CHF-6366: A Novel Super-soft Dual Pharmacology Muscarinic Antagonist and β2 Agonist (MABA) for the Inhaled Treatment of Respiratory Diseases
Carzaniga, Laura, Linney, Ian D., Rizzi, Andrea, Delcanale, Maurizio, Schmidt, Wolfgang, Knight, Christopher K., Pastore, Fiorella, Miglietta, Daniela, Carnini, Chiara, Cesari, Nicola, Riccardi, Benedetta, Mileo, Valentina, Venturi, Luca, Moretti, Elisa, Blackaby, Wesley P., Patacchini, Riccardo, Accetta, Alessandro, Biagetti, Matteo, Bassani, Franco, Tondelli, Marina, Murgo, Annalisa, Battipaglia, Loredana, Villetti, Gino, Puccini, Paola, Catinella, Silvia, Civelli, Maurizio, Rancati, Fabio
Published in Journal of medicinal chemistry (11.08.2022)
Published in Journal of medicinal chemistry (11.08.2022)
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Journal Article
Discovery of M-3 Antagonist-PDE4 Inhibitor Dual Pharmacology Molecules for the Treatment of Chronic Obstructive Pulmonary Disease
Armani, Elisabetta, Rizzi, Andrea, Capaldi, Carmelida, De Fanti, Renato, Delcanale, Maurizio, Villetti, Gino, Marchini, Gessica, Pisano, Anna Rita, Pitozzi, Vanessa, Pittelli, Maria Gloria, Trevisani, Marcello, Salvadori, Michela, Cenacchi, Valentina, Puccini, Paola, Amadei, Francesco, Pappani, Alice, Civelli, Maurizio, Patacchini, Riccardo, Baker-Glenn, Charles A. G., Van de Poel, Herve, Blackaby, Wesley P., Nash, Kevin, Amari, Gabriele
Published in Journal of medicinal chemistry (08.07.2021)
Published in Journal of medicinal chemistry (08.07.2021)
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Journal Article
CHF6001 I: a novel highly potent and selective phosphodiesterase 4 inhibitor with robust anti-inflammatory activity and suitable for topical pulmonary administration
Moretto, Nadia, Caruso, Paola, Bosco, Raffaella, Marchini, Gessica, Pastore, Fiorella, Armani, Elisabetta, Amari, Gabriele, Rizzi, Andrea, Ghidini, Eleonora, De Fanti, Renato, Capaldi, Carmelida, Carzaniga, Laura, Hirsch, Emilio, Buccellati, Carola, Sala, Angelo, Carnini, Chiara, Patacchini, Riccardo, Delcanale, Maurizio, Civelli, Maurizio, Villetti, Gino, Facchinetti, Fabrizio
Published in The Journal of pharmacology and experimental therapeutics (01.03.2015)
Published in The Journal of pharmacology and experimental therapeutics (01.03.2015)
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Journal Article
Discovery of Clinical Candidate CHF-6366: A Novel Super-soft Dual Pharmacology Muscarinic Antagonist and β 2 Agonist (MABA) for the Inhaled Treatment of Respiratory Diseases
Carzaniga, Laura, Linney, Ian D., Rizzi, Andrea, Delcanale, Maurizio, Schmidt, Wolfgang, Knight, Christopher K., Pastore, Fiorella, Miglietta, Daniela, Carnini, Chiara, Cesari, Nicola, Riccardi, Benedetta, Mileo, Valentina, Venturi, Luca, Moretti, Elisa, Blackaby, Wesley P., Patacchini, Riccardo, Accetta, Alessandro, Biagetti, Matteo, Bassani, Franco, Tondelli, Marina, Murgo, Annalisa, Battipaglia, Loredana, Villetti, Gino, Puccini, Paola, Catinella, Silvia, Civelli, Maurizio, Rancati, Fabio
Published in Journal of medicinal chemistry (11.08.2022)
Published in Journal of medicinal chemistry (11.08.2022)
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Journal Article
Design, Synthesis, and Biological Characterization of Inhaled p38α/β MAPK Inhibitors for the Treatment of Lung Inflammatory Diseases
Armani, Elisabetta, Capaldi, Carmelida, Bagnacani, Valentina, Saccani, Francesca, Aquino, Giancarlo, Puccini, Paola, Facchinetti, Fabrizio, Martucci, Cataldo, Moretto, Nadia, Villetti, Gino, Patacchini, Riccardo, Civelli, Maurizio, Hurley, Chris, Jennings, Andrew, Alcaraz, Lilian, Bloomfield, Dawn, Briggs, Michael, Daly, Stephen, Panchal, Terry, Russell, Vince, Wicks, Sharon, Finch, Harry, Fitzgerald, Mary, Fox, Craig, Delcanale, Maurizio
Published in Journal of medicinal chemistry (26.05.2022)
Published in Journal of medicinal chemistry (26.05.2022)
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Journal Article
Discovery of M3 Antagonist-PDE4 Inhibitor Dual Pharmacology Molecules for the Treatment of Chronic Obstructive Pulmonary Disease
Armani, Elisabetta, Rizzi, Andrea, Capaldi, Carmelida, De Fanti, Renato, Delcanale, Maurizio, Villetti, Gino, Marchini, Gessica, Pisano, Anna Rita, Pitozzi, Vanessa, Pittelli, Maria Gloria, Trevisani, Marcello, Salvadori, Michela, Cenacchi, Valentina, Puccini, Paola, Amadei, Francesco, Pappani, Alice, Civelli, Maurizio, Patacchini, Riccardo, Baker-Glenn, Charles A.G, Van de Poël, Hervé, Blackaby, Wesley P, Nash, Kevin, Amari, Gabriele
Published in Journal of medicinal chemistry (08.07.2021)
Published in Journal of medicinal chemistry (08.07.2021)
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Journal Article
Discovery and Optimization of Thiazolidinyl and Pyrrolidinyl Derivatives as Inhaled PDE4 Inhibitors for Respiratory Diseases
Carzaniga, Laura, Amari, Gabriele, Rizzi, Andrea, Capaldi, Carmelida, De Fanti, Renato, Ghidini, Eleonora, Villetti, Gino, Carnini, Chiara, Moretto, Nadia, Facchinetti, Fabrizio, Caruso, Paola, Marchini, Gessica, Battipaglia, Loredana, Patacchini, Riccardo, Cenacchi, Valentina, Volta, Roberta, Amadei, Francesco, Pappani, Alice, Capacchi, Silvia, Bagnacani, Valentina, Delcanale, Maurizio, Puccini, Paola, Catinella, Silvia, Civelli, Maurizio, Armani, Elisabetta
Published in Journal of medicinal chemistry (28.12.2017)
Published in Journal of medicinal chemistry (28.12.2017)
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Journal Article
Erythroid differentiation ability of butyric acid analogues: Identification of basal chemical structures of new inducers of foetal haemoglobin
Bianchi, Nicoletta, Chiarabelli, Cristiano, Zuccato, Cristina, Lampronti, Ilaria, Borgatti, Monica, Amari, Gabriele, Delcanale, Maurizio, Chiavilli, Francesco, Prus, Eugenia, Fibach, Eitan, Gambari, Roberto
Published in European journal of pharmacology (05.04.2015)
Published in European journal of pharmacology (05.04.2015)
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Journal Article