Design, Synthesis, and Pharmacological Evaluation of Bis-2-(5-phenylacetamido-1,2,4-thiadiazol-2-yl)ethyl Sulfide 3 (BPTES) Analogs as Glutaminase Inhibitors
Shukla, Krupa, Ferraris, Dana V., Thomas, Ajit G., Stathis, Marigo, Duvall, Bridget, Delahanty, Greg, Alt, Jesse, Rais, Rana, Rojas, Camilo, Gao, Ping, Xiang, Yan, Dang, Chi V., Slusher, Barbara S., Tsukamoto, Takashi
Published in Journal of medicinal chemistry (13.12.2012)
Published in Journal of medicinal chemistry (13.12.2012)
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Design, Synthesis, and Pharmacological Evaluation of Fluorinated Tetrahydrouridine Derivatives as Inhibitors of Cytidine Deaminase
Ferraris, Dana, Duvall, Bridget, Delahanty, Greg, Mistry, Bipin, Alt, Jesse, Rojas, Camilo, Rowbottom, Christopher, Sanders, Kristen, Schuck, Edgar, Huang, Kuan-Chun, Redkar, Sanjeev, Slusher, Barbara B, Tsukamoto, Takashi
Published in Journal of medicinal chemistry (27.03.2014)
Published in Journal of medicinal chemistry (27.03.2014)
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Peptidomimetics of Arg-Phe-NH2 as small molecule agonists of Mas-related gene C (MrgC) receptors
Hin, Niyada, Alt, Jesse, Zimmermann, Sarah C., Delahanty, Greg, Ferraris, Dana V., Rojas, Camilo, Li, Fengxian, Liu, Qin, Dong, Xinzhong, Slusher, Barbara S., Tsukamoto, Takashi
Published in Bioorganic & medicinal chemistry (01.11.2014)
Published in Bioorganic & medicinal chemistry (01.11.2014)
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Peptidomimetics of Arg-Phe-NH sub(2) as small molecule agonists of Mas-related gene C (MrgC) receptors
Hin, Niyada, Alt, Jesse, Zimmermann, Sarah C, Delahanty, Greg, Ferraris, Dana V, Rojas, Camilo, Li, Fengxian, Liu, Qin, Dong, Xinzhong, Slusher, Barbara S, Tsukamoto, Takashi
Published in Bioorganic & medicinal chemistry (01.11.2014)
Published in Bioorganic & medicinal chemistry (01.11.2014)
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Design, Synthesis, and Pharmacological Evaluation of Glutamate Carboxypeptidase II (GCPII) Inhibitors Based on Thioalkylbenzoic Acid Scaffolds
Stoermer, Doris, Vitharana, Dilrukshi, Hin, Niyada, Delahanty, Greg, Duvall, Bridget, Ferraris, Dana V, Grella, Brian S, Hoover, Randall, Rojas, Camilo, Shanholtz, Megan K, Smith, Kyle P, Stathis, Marigo, Wu, Ying, Wozniak, Krystyna M, Slusher, Barbara S, Tsukamoto, Takashi
Published in Journal of medicinal chemistry (28.06.2012)
Published in Journal of medicinal chemistry (28.06.2012)
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Journal Article
Design, synthesis, and pharmacological evaluation of bis-2-(5-phenylacetamido-1,2,4-thiadiazol-2-yl)ethyl sulfide (BPTES) analogs as glutaminase inhibitors
Shukla, Krupa, Ferraris, Dana V., Thomas, Ajit G., Stathis, Marigo, Duvall, Bridget, Delahanty, Greg, Alt, Jesse, Rais, Rana, Rojas, Camilo, Gao, Ping, Xiang, Yan, Dang, Chi V., Slusher, Barbara S., Tsukamoto, Takashi
Published in Journal of medicinal chemistry (30.11.2012)
Published in Journal of medicinal chemistry (30.11.2012)
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The discovery and structure–activity relationships of indole-based inhibitors of glutamate carboxypeptidase II
Grella, Brian, Adams, Jessica, Berry, James F., Delahanty, Greg, Ferraris, Dana V., Majer, Pavel, Ni, Chiyou, Shukla, Krupa, Shuler, Scott A., Slusher, Barbara S., Stathis, Marigo, Tsukamoto, Takashi
Published in Bioorganic & medicinal chemistry letters (15.12.2010)
Published in Bioorganic & medicinal chemistry letters (15.12.2010)
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Structural Optimization of Thiol-Based Inhibitors of Glutamate Carboxypeptidase II by Modification of the P1‘ Side Chain
Majer, Pavel, Hin, Bunda, Stoermer, Doris, Adams, Jessica, Xu, Weizheng, Duvall, Bridget R, Delahanty, Greg, Liu, Qun, Stathis, Marigo J, Wozniak, Krystyna M, Slusher, Barbara S, Tsukamoto, Takashi
Published in Journal of medicinal chemistry (18.05.2006)
Published in Journal of medicinal chemistry (18.05.2006)
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Journal Article
Synthesis and Biological Evaluation of Thiol-Based Inhibitors of Glutamate Carboxypeptidase II: Discovery of an Orally Active GCP II Inhibitor
Majer, Pavel, Jackson, Paul F, Delahanty, Greg, Grella, Brian S, Ko, Yao-Sen, Li, Weixing, Liu, Qun, Maclin, Keith M, Poláková, Jana, Shaffer, Kathryn A, Stoermer, Doris, Vitharana, Dilrukshi, Wang, Eric Yanjun, Zakrzewski, Anthony, Rojas, Camilo, Slusher, Barbara S, Wozniak, Krystyna M, Burak, Eric, Limsakun, Tharin, Tsukamoto, Takashi
Published in Journal of medicinal chemistry (08.05.2003)
Published in Journal of medicinal chemistry (08.05.2003)
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