Conjugate Additions of Amines to Maleimides via Cooperative Catalysis
Uno, Brice E., Deibler, Kristine K., Villa, Carlos, Raghuraman, Arjun, Scheidt, Karl A.
Published in Advanced synthesis & catalysis (17.04.2018)
Published in Advanced synthesis & catalysis (17.04.2018)
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Journal Article
Design and structural validation of peptide-drug conjugate ligands of the kappa-opioid receptor
Muratspahić, Edin, Deibler, Kristine, Han, Jianming, Tomašević, Nataša, Jadhav, Kirtikumar B, Olivé-Marti, Aina-Leonor, Hochrainer, Nadine, Hellinger, Roland, Koehbach, Johannes, Fay, Jonathan F, Rahman, Mohammad Homaidur, Hegazy, Lamees, Craven, Timothy W, Varga, Balazs R, Bhardwaj, Gaurav, Appourchaux, Kevin, Majumdar, Susruta, Muttenthaler, Markus, Hosseinzadeh, Parisa, Craik, David J, Spetea, Mariana, Che, Tao, Baker, David, Gruber, Christian W
Published in Nature communications (06.12.2023)
Published in Nature communications (06.12.2023)
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Journal Article
A Chemical Probe Strategy for Interrogating Inhibitor Selectivity Across the MEK Kinase Family
Deibler, Kristine K, Mishra, Rama K, Clutter, Matthew R, Antanasijevic, Aleksandar, Bergan, Raymond, Caffrey, Michael, Scheidt, Karl A
Published in ACS chemical biology (19.05.2017)
Published in ACS chemical biology (19.05.2017)
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Journal Article
Modeling MEK4 Kinase Inhibitors through Perturbed Electrostatic Potential Charges
Mishra, Rama K, Deibler, Kristine K, Clutter, Matthew R, Vagadia, Purav P, O’Connor, Matthew, Schiltz, Gary E, Bergan, Raymond, Scheidt, Karl A
Published in Journal of chemical information and modeling (28.10.2019)
Published in Journal of chemical information and modeling (28.10.2019)
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Journal Article
Rational Design of Highly Potent and Selective Covalent MAP2K7 Inhibitors
Kim, Dalton R., Orr, Meghan J., Kwong, Ada J., Deibler, Kristine K., Munshi, Hasan H., Bridges, Cory Seth, Chen, Taylor Jie, Zhang, Xiaoyu, Lacorazza, H. Daniel, Scheidt, Karl A.
Published in ACS medicinal chemistry letters (11.05.2023)
Published in ACS medicinal chemistry letters (11.05.2023)
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Journal Article
Synthesis and Biological Evaluation of 3‐Arylindazoles as Selective MEK4 Inhibitors
Deibler, Kristine K., Schiltz, Gary E., Clutter, Matthew R., Mishra, Rama K., Vagadia, Purav P., O'Connor, Matthew, George, Mariam Donny, Gordon, Ryan, Fowler, Graham, Bergan, Raymond, Scheidt, Karl A.
Published in ChemMedChem (22.03.2019)
Published in ChemMedChem (22.03.2019)
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Journal Article
Deorphanizing Peptides Using Structure Prediction
Teufel, Felix, Refsgaard, Jan C., Kasimova, Marina A., Deibler, Kristine, Madsen, Christian T., Stahlhut, Carsten, Grønborg, Mads, Winther, Ole, Madsen, Dennis
Published in Journal of chemical information and modeling (08.05.2023)
Published in Journal of chemical information and modeling (08.05.2023)
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Journal Article
An integrated platform approach enables discovery of potent, selective and ligand-competitive cyclic peptides targeting the GIP receptor
Bhushan, Bhaskar, Granata, Daniele, Kaas, Christian S, Kasimova, Marina A, Ren, Qiansheng, Cramer, Christian N, White, Mark D, Hansen, Ann Maria K, Fledelius, Christian, Invernizzi, Gaetano, Deibler, Kristine, Coleman, Oliver D, Zhao, Xin, Qu, Xinping, Liu, Haimo, Zurmühl, Silvana S, Kodra, Janos T, Kawamura, Akane, Münzel, Martin
Published in Chemical science (Cambridge) (16.03.2022)
Published in Chemical science (Cambridge) (16.03.2022)
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