Deep cavitands featuring functional acetal-based walls
Degardin, Melissa, Busseron, Eric, Kim, Dang-A., Ajami, Dariush, Rebek, Julius
Published in Chemical communications (Cambridge, England) (01.01.2012)
Published in Chemical communications (Cambridge, England) (01.01.2012)
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Journal Article
Natural-like Replication of an Unnatural Base Pair for the Expansion of the Genetic Alphabet and Biotechnology Applications
Li, Lingjun, Degardin, Mélissa, Lavergne, Thomas, Malyshev, Denis A, Dhami, Kirandeep, Ordoukhanian, Phillip, Romesberg, Floyd E
Published in Journal of the American Chemical Society (22.01.2014)
Published in Journal of the American Chemical Society (22.01.2014)
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Journal Article
Expanding the Scope of Replicable Unnatural DNA: Stepwise Optimization of a Predominantly Hydrophobic Base Pair
Lavergne, Thomas, Degardin, Mélissa, Malyshev, Denis A, Quach, Henry T, Dhami, Kirandeep, Ordoukhanian, Phillip, Romesberg, Floyd E
Published in Journal of the American Chemical Society (10.04.2013)
Published in Journal of the American Chemical Society (10.04.2013)
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Journal Article
Synthesis and recognition studies with a ditopic, photoswitchable deep cavitand
Busseron, Eric, Lux, Jacques, Degardin, Mélissa, Rebek, Jr, Julius
Published in Chemical communications (Cambridge, England) (25.05.2013)
Published in Chemical communications (Cambridge, England) (25.05.2013)
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Journal Article
Impact of Multimeric Ferrocene‐containing Cyclodecapeptide Scaffold on Host‐Guest Interactions at a β‐Cyclodextrin Covered Surface
Sanchez Perez, Enrique, Toor, Ritu, Bruyat, Pierrick, Cepeda, Céline, Degardin, Mélissa, Dejeu, Jérôme, Boturyn, Didier, Coche‐Guérente, Liliane
Published in Chemphyschem (04.11.2021)
Published in Chemphyschem (04.11.2021)
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Journal Article
Radiotheranostic Agent 64Cu-cyclam-RAFT-c(-RGDfK-)4 for Management of Peritoneal Metastasis in Ovarian Cancer
Jin, Zhao-Hui, Tsuji, Atsushi B., Degardin, Mélissa, Sugyo, Aya, Obara, Satoshi, Wakizaka, Hidekatsu, Nagatsu, Kotaro, Hu, Kuan, Zhang, Ming-Rong, Dumy, Pascal, Boturyn, Didier, Higashi, Tatsuya
Published in Clinical cancer research (01.12.2020)
Published in Clinical cancer research (01.12.2020)
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Journal Article
Multiplexed Imaging Reveals the Spatial Relationship of the Extracellular Acidity-Targeting pHLIP with Necrosis, Hypoxia, and the Integrin-Targeting cRGD Peptide
Jin, Zhao-Hui, Tsuji, Atsushi B, Degardin, Mélissa, Dumy, Pascal, Boturyn, Didier, Higashi, Tatsuya
Published in Cells (Basel, Switzerland) (01.11.2022)
Published in Cells (Basel, Switzerland) (01.11.2022)
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Journal Article
From Peptide Aptamers to Inhibitors of FUR, Bacterial Transcriptional Regulator of Iron Homeostasis and Virulence
Mathieu, Sophie, Cissé, Cheickna, Vitale, Sylvia, Ahmadova, Aynur, Degardin, Mélissa, Pérard, Julien, Colas, Pierre, Miras, Roger, Boturyn, Didier, Covès, Jacques, Crouzy, Serge, Michaud-Soret, Isabelle
Published in ACS chemical biology (16.09.2016)
Published in ACS chemical biology (16.09.2016)
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Journal Article
Heparan sulfate co-immobilized with cRGD ligands and BMP2 on biomimetic platforms promotes BMP2-mediated osteogenic differentiation
Sefkow-Werner, Julius, Machillot, Paul, Sales, Adria, Castro-Ramirez, Elaine, Degardin, Melissa, Boturyn, Didier, Cavalcanti-Adam, Elisabetta Ada, Albiges-Rizo, Corinne, Picart, Catherine, Migliorini, Elisa
Published in Acta biomaterialia (15.09.2020)
Published in Acta biomaterialia (15.09.2020)
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Journal Article
Uniform intratumoral distribution of radioactivity produced using two different radioagents, 64Cu-cyclam-RAFT-c(-RGDfK-)4 and 64Cu-ATSM, improves therapeutic efficacy in a small animal tumor model
Jin, Zhao-Hui, Tsuji, Atsushi B., Degardin, Mélissa, Sugyo, Aya, Yoshii, Yukie, Nagatsu, Kotaro, Zhang, Ming-Rong, Fujibayashi, Yasuhisa, Dumy, Pascal, Boturyn, Didier, Higashi, Tatsuya
Published in EJNMMI research (19.06.2018)
Published in EJNMMI research (19.06.2018)
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Journal Article
N-substituted bis- C-alkyloxadiazolones as dual effectors: Efficient intermediates to amidoximes or amidines and prodrug candidates of potent antimalarials
Degardin, Mélissa, Wein, Sharon, Durand, Thierry, Escale, Roger, Vial, Henry, Vo-Hoang, Yen
Published in Bioorganic & medicinal chemistry letters (01.09.2009)
Published in Bioorganic & medicinal chemistry letters (01.09.2009)
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Journal Article
Development of the First Oral Bioprecursors of Bis-alkylguanidine Antimalarial Drugs
Degardin, Mélissa, Wein, Sharon, Duckert, Jean-Frédéric, Maynadier, Marjorie, Guy, Alexandre, Durand, Thierry, Escale, Roger, Vial, Henri, Vo-Hoang, Yen
Published in ChemMedChem (01.02.2014)
Published in ChemMedChem (01.02.2014)
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Journal Article
Heparan sulfate co-immobilized with cRGD ligands and BMP2 on biomimetic platforms promotes BMP2-me diate d osteogenic differentiation
Sefkow-Werner, Julius, Machillot, Paul, Sales, Adrià, Castro-Ramirez, Elaine, Degardin, Melissa, Boturyn, Didier, Cavalcanti-Adam, Elisabetta Ada, Albiges-Rizo, Corinne, Picart, Catherine, Migliorini, Elisa
Published in Acta biomaterialia (2020)
Published in Acta biomaterialia (2020)
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Journal Article
Multivalency: influence of the residence time and the retraction rate on rupture forces measured by AFM
Bacharouche, Jalal, Degardin, Mélissa, Jierry, Loïc, Carteret, Cédric, Lavalle, Philippe, Hemmerlé, Joseph, Senger, Bernard, Auzély-Velty, Rachel, Boulmedais, Fouzia, Boturyn, Didier, Coche-Guérente, Liliane, Schaaf, Pierre, Francius, Grégory
Published in Journal of materials chemistry. B, Materials for biology and medicine (07.03.2015)
Published in Journal of materials chemistry. B, Materials for biology and medicine (07.03.2015)
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Journal Article
alpha V beta 3 Integrin-Targeted Radionuclide Therapy with 64Cu-cyclam-RAFT-c(-RGDfK-)4
Jin, Zhao-Hui, Furukawa, Takako, Degardin, Melissa, Sugyo, Aya, Tsuji, Atsushi B, Yamasaki, Tomoteru, Kawamura, Kazunori, Fujibayashi, Yasuhisa, Zhang, Ming-Rong, Boturyn, Didier, Dumy, Pascal, Saga, Tsuneo
Published in Molecular cancer therapeutics (15.09.2016)
Published in Molecular cancer therapeutics (15.09.2016)
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Journal Article
Evaluation of Bis-Alkylamidoxime O-Alkylsulfonates as Orally Available Antimalarials
Degardin, Mélissa, Wein, Sharon, Gouni, Smitha, Tran Van Ba, Christophe, Duckert, Jean-Frédéric, Durand, Thierry, Escale, Roger, Vial, Henri, Vo-Hoang, Yen
Published in ChemMedChem (01.06.2012)
Published in ChemMedChem (01.06.2012)
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Journal Article
Rational design of peptide derivatives for inhibition of MyD88‐mediated toll‐like receptor signaling in human peripheral blood mononuclear cells and epithelial cells exposed to Francisella tularensis
Ryan, Daniel A., Degardin, Melissa, Alam, Shahabuddin, Kissner, Teri L., Hale, Martha, Cameron, Michael D., Rebek, Mitra, Ajami, Dariush, Saikh, Kamal U., Rebek, Julius
Published in Chemical biology & drug design (01.12.2017)
Published in Chemical biology & drug design (01.12.2017)
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Journal Article
Deep cavitands featuring functional acetal-based wallsElectronic supplementary information (ESI) available: Synthetic procedures and characterization data for compounds 2-5, 7, 10-13, NMR spectra of the studied host-guest systems, VT-NMR and NOESY experiments. See DOI: 10.1039/c2cc36517k
Degardin, Melissa, Busseron, Eric, Kim, Dang-A, Ajami, Dariush, Rebek, Julius
Year of Publication 12.11.2012
Year of Publication 12.11.2012
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Journal Article
Structure-Based Design and Synthesis of a Small Molecule that Exhibits Anti-inflammatory Activity by Inhibition of MyD88-mediated Signaling to Bacterial Toxin Exposure
Alam, Shahabuddin, Javor, Sacha, Degardin, Melissa, Ajami, Dariush, Rebek, Mitra, Kissner, Teri L., Waag, David M., Rebek Jr, Julius, Saikh, Kamal U.
Published in Chemical biology & drug design (01.08.2015)
Published in Chemical biology & drug design (01.08.2015)
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Journal Article
Correction: Multivalency: influence of the residence time and the retraction rate on rupture forces measured by AFM
Bacharouche, Jalal, Degardin, Mélissa, Jierry, Loïc, Carteret, Cédric, Lavalle, Philippe, Hemmerlé, Joseph, Senger, Bernard, Auzély-Velty, Rachel, Boulmedais, Fouzia, Boturyn, Didier, Coche-Guérente, Liliane, Schaaf, Pierre, Francius, Grégory
Published in Journal of materials chemistry. B, Materials for biology and medicine (21.04.2015)
Published in Journal of materials chemistry. B, Materials for biology and medicine (21.04.2015)
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Journal Article