Discovery of 2-amino-heteroaryl-benzothiazole-6-anilides as potent p56(lck) inhibitors
Das, Jagabandhu, Moquin, Robert V, Lin, James, Liu, Chunjian, Doweyko, Arthur M, DeFex, Henry F, Fang, Qiong, Pang, Suhong, Pitt, Sidney, Shen, Ding Ren, Schieven, Gary L, Barrish, Joel C, Wityak, John
Published in Bioorganic & medicinal chemistry letters (04.08.2003)
Published in Bioorganic & medicinal chemistry letters (04.08.2003)
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Journal Article
Molecular design, synthesis, and structure-Activity relationships leading to the potent and selective p56(lck) inhibitor BMS-243117
Das, Jagabandhu, Lin, James, Moquin, Robert V, Shen, Zhongqi, Spergel, Steven H, Wityak, John, Doweyko, Arthur M, DeFex, Henry F, Fang, Qiong, Pang, Suhong, Pitt, Sidney, Shen, Ding Ren, Schieven, Gary L, Barrish, Joel C
Published in Bioorganic & medicinal chemistry letters (07.07.2003)
Published in Bioorganic & medicinal chemistry letters (07.07.2003)
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Journal Article
Molecular design, synthesis, and structure-activity relationships leading to the potent and selective p56lck inhibitor BMS-243117
DAS, Jagabandhu, LIN, James, PITT, Sidney, DING REN SHEN, SCHIEVEN, Gary L, BARRISH, Joel C, MOQUIN, Robert V, ZHONGQI SHEN, SPERGEL, Steven H, WITYAK, John, DOWEYKO, Arthur M, DEFEX, Henry F, QIONG FANG, SUHONG PANG
Published in Bioorganic & medicinal chemistry letters (01.07.2003)
Published in Bioorganic & medicinal chemistry letters (01.07.2003)
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Journal Article
Discovery of 2-amino-heteroaryl-benzothiazole-6-anilides as potent p56lck inhibitors
DAS, Jagabandhu, MOQUIN, Robert V, SCHIEVEN, Gary L, BARRISH, Joel C, WITYAK, John, LIN, James, LIU, Chunjian, DOWEYKO, Arthur M, DEFEX, Henry F, FANG, Qiong, PANG, Suhong, PITT, Sidney, DING REN SHEN
Published in Bioorganic & medicinal chemistry letters (01.08.2003)
Published in Bioorganic & medicinal chemistry letters (01.08.2003)
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Journal Article
The mGluR2 positive allosteric modulator, SAR218645, improves memory and attention deficits in translational models of cognitive symptoms associated with schizophrenia
Griebel, Guy, Pichat, Philippe, Boulay, Denis, Naimoli, Vanessa, Potestio, Lisa, Featherstone, Robert, Sahni, Sukhveen, Defex, Henry, Desvignes, Christophe, Slowinski, Franck, Vigé, Xavier, Bergis, Olivier E, Sher, Rosy, Kosley, Raymond, Kongsamut, Sathapana, Black, Mark D, Varty, Geoffrey B
Published in Scientific reports (13.10.2016)
Published in Scientific reports (13.10.2016)
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Journal Article
Discovery of 2-amino-heteroaryl-benzothiazole-6-anilides as potent p56 lck inhibitors
Das, Jagabandhu, Moquin, Robert V., Lin, James, Liu, Chunjian, Doweyko, Arthur M., DeFex, Henry F., Fang, Qiong, Pang, Suhong, Pitt, Sidney, Shen, Ding Ren, Schieven, Gary L., Barrish, Joel C., Wityak, John
Published in Bioorganic & medicinal chemistry letters (2003)
Published in Bioorganic & medicinal chemistry letters (2003)
Get full text
Journal Article
Molecular design, synthesis, and structure–Activity relationships leading to the potent and selective p56 lck inhibitor BMS-243117
Das, Jagabandhu, Lin, James, Moquin, Robert V., Shen, Zhongqi, Spergel, Steven H., Wityak, John, Doweyko, Arthur M., DeFex, Henry F., Fang, Qiong, Pang, Suhong, Pitt, Sidney, Shen, Ding Ren, Schieven, Gary L., Barrish, Joel C.
Published in Bioorganic & medicinal chemistry letters (2003)
Published in Bioorganic & medicinal chemistry letters (2003)
Get full text
Journal Article