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Arginase inhibitors and methods of use thereof
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Year of Publication 22.12.2023
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Synthesis and KCNQ2 opener activity of N-(1-benzo[1,3]dioxol-5-yl-ethyl, N-[1-(2,3-dihydro-benzofuran-5-yl)-ethyl, and N-[1-(2,3-dihydro-1 H-indol-5-yl)-ethyl acrylamides
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Published in Bioorganic & medicinal chemistry letters (06.09.2004)
Published in Bioorganic & medicinal chemistry letters (06.09.2004)
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Novel 3‘,6‘-Anhydro and N12,N13-Bridged Glycosylated Fluoroindolo[2,3-a]carbazoles as Topoisomerase I Inhibitors. Fluorine as a Leaving Group from sp3 Carbon
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Published in Organic letters (31.03.2005)
Published in Organic letters (31.03.2005)
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Journal Article
Novel 3‘,6‘-Anhydro and N12,N13-Bridged Glycosylated Fluoroindolo[2,3- a ]carbazoles as Topoisomerase I Inhibitors. Fluorine as a Leaving Group from sp 3 Carbon
Saulnier, Mark G., Langley, David R., Frennesson, David B., Long, Byron H., Huang, Stella, Gao, Qi, Wu, Dedong, Fairchild, Craig R., Ruediger, Edward, Zimmermann, Kurt, St. Laurent, Denis R., Balasubramanian, Balu N., Vyas, Dolatrai M.
Published in Organic letters (01.03.2005)
Published in Organic letters (01.03.2005)
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Arginase inhibitors and methods of use thereof
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Year of Publication 23.08.2022
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Year of Publication 23.08.2022
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ARGINASE INHIBITORS AND METHODS OF USE THEREOF
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Year of Publication 23.06.2022
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Year of Publication 23.06.2022
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Identification of a potent and selective 5-HT(6) antagonist: one-step synthesis of (E)-3-(benzenesulfonyl)-2- (methylsulfanyl)pyrido[1,2-a]pyrimidin-4-ylidenamine from 2-(benzenesulfonyl)-3,3-bis(methylsulfanyl)acrylonitrile
Wu, Yong-Jin, He, Huan, Hu, Shuanghua, Huang, Yazhong, Scola, Paul M, Grant-Young, Katharine, Bertekap, Robert L, Wu, Dedong, Gao, Qi, Li, Yi, Klakouski, Cheryl, Westphal, Ryan S
Published in Journal of medicinal chemistry (06.11.2003)
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Published in Journal of medicinal chemistry (06.11.2003)
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Identification of a Potent and Selective 5-HT 6 Antagonist: One-Step Synthesis of ( E )-3-(Benzenesulfonyl)-2- (methylsulfanyl)pyrido[1,2- a ]pyrimidin- 4-ylidenamine from 2-(Benzenesulfonyl)-3,3- bis(methylsulfanyl)acrylonitrile
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(S)-N-[1-(4-Cyclopropylmethyl-3,4-dihydro-2H-benzooxazin-6-yl)-ethyl]-3-(2-fluoro-phenyl)-acrylamide is a potent and efficacious KCNQ2 opener which inhibits induced hyperexcitability of rat hippocampal neurons
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Synthesis and KCNQ2 opener activity of N-1-benzo[1,3]dioxol-5-yl-ethyl, N-[1-(2,3-dihydro-benzofuran-5-yl)-ethyl, and N-[1-(2,3-dihydro-1H-indol-5-yl)-ethyl acrylamides
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Published in Bioorganic & medicinal chemistry letters (2004)
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