Inhibitors of the Cancer Target Ribonucleotide Reductase, Past and Present
Huff, Sarah E., Winter, Jordan M., Dealwis, Chris G.
Published in Biomolecules (Basel, Switzerland) (10.06.2022)
Published in Biomolecules (Basel, Switzerland) (10.06.2022)
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Journal Article
Structure-guided design of anti-cancer ribonucleotide reductase inhibitors
Misko, Tessianna A., Liu, Yi-Ting, Harris, Michael E., Oleinick, Nancy L., Pink, John, Lee, Hsueh-Yun, Dealwis, Chris G.
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2019)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2019)
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Journal Article
Crystal Structure of the Anthrax Drug Target, Bacillus anthracis Dihydrofolate Reductase
Bennett, Brad C, Xu, Hai, Simmerman, Richard F, Lee, Richard E, Dealwis, Chris G
Published in Journal of medicinal chemistry (06.09.2007)
Published in Journal of medicinal chemistry (06.09.2007)
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Journal Article
Definition of fatty acid transport protein-2 (FATP2) structure facilitates identification of small molecule inhibitors for the treatment of diabetic complications
Kumar, Mukesh, Gaivin, Robert J., Khan, Shenaz, Fedorov, Yuriy, Adams, Drew J., Zhao, Weiyang, Lee, Hsueh-Yun, Dai, Xinghong, Dealwis, Chris G., Schelling, Jeffrey R.
Published in International journal of biological macromolecules (31.07.2023)
Published in International journal of biological macromolecules (31.07.2023)
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Journal Article
Targeting the Large Subunit of Human Ribonucleotide Reductase for Cancer Chemotherapy
Wijerathna, Sanath R, Ahmad, Md Faiz, Xu, Hai, Fairman, James W, Zhang, Andrew, Kaushal, Prem Singh, Wan, Qun, Kiser, Jianying, Dealwis, Chris G
Published in Pharmaceuticals (13.10.2011)
Published in Pharmaceuticals (13.10.2011)
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Journal Article
Book Review
Structure-Guided Synthesis and Mechanistic Studies Reveal Sweetspots on Naphthyl Salicyl Hydrazone Scaffold as Non-Nucleosidic Competitive, Reversible Inhibitors of Human Ribonucleotide Reductase
Huff, Sarah E, Mohammed, Faiz Ahmad, Yang, Mu, Agrawal, Prashansa, Pink, John, Harris, Michael E, Dealwis, Chris G, Viswanathan, Rajesh
Published in Journal of medicinal chemistry (08.02.2018)
Published in Journal of medicinal chemistry (08.02.2018)
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Journal Article
Capturing the Catalytic Proton of Dihydrofolate Reductase: Implications for General Acid–Base Catalysis
Wan, Qun, Bennett, Brad C, Wymore, Troy, Li, Zhihong, Wilson, Mark A, Brooks, Charles L, Langan, Paul, Kovalevsky, Andrey, Dealwis, Chris G
Published in ACS catalysis (07.05.2021)
Published in ACS catalysis (07.05.2021)
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Journal Article
Nucleoside Analogue Triphosphates Allosterically Regulate Human Ribonucleotide Reductase and Identify Chemical Determinants That Drive Substrate Specificity
Knappenberger, Andrew J, Ahmad, Md. Faiz, Viswanathan, Rajesh, Dealwis, Chris G, Harris, Michael E
Published in Biochemistry (Easton) (18.10.2016)
Published in Biochemistry (Easton) (18.10.2016)
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Journal Article
Inhibition of yeast ribonucleotide reductase by Sml1 depends on the allosteric state of the enzyme
Misko, Tessianna A., Wijerathna, Sanath R., Radivoyevitch, Tomas, Berdis, Anthony J., Ahmad, Md. Faiz, Harris, Michael E., Dealwis, Chris G.
Published in FEBS letters (01.06.2016)
Published in FEBS letters (01.06.2016)
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Journal Article
The Structural Basis for the Allosteric Regulation of Ribonucleotide Reductase
Ahmad, Md. Faiz, Dealwis, Chris G.
Published in Progress in Molecular Biology and Translational Science (2013)
Published in Progress in Molecular Biology and Translational Science (2013)
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Book Chapter
Reference
Journal Article
Crystallographic analysis of reversible metal binding observed in a mutant (Asp153 .fwdarw. Gly) of Escherichia coli alkaline phosphatase
Dealwis, Chris G, Brennan, Catherine, Christianson, Kris, Mandecki, Wlodek, Abad-Zapatero, Cele
Published in Biochemistry (Easton) (01.10.1995)
Published in Biochemistry (Easton) (01.10.1995)
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Journal Article
Sml1p Is a Dimer in Solution: Characterization of Denaturation and Renaturation of Recombinant Sml1p
Gupta, Vibha, Peterson, Cynthia B, Dice, Lezlee T, Uchiki, Tomoaki, Racca, Joseph, Guo, Jun-tao, Xu, Ying, Hettich, Robert, Zhao, Xiaolan, Rothstein, Rodney, Dealwis, Chris G
Published in Biochemistry (Easton) (06.07.2004)
Published in Biochemistry (Easton) (06.07.2004)
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Journal Article
Preliminary neutron diffraction studies of Escherichia coli dihydrofolate reductase bound to the anticancer drug methotrexate
Bennett, Brad C., Meilleur, Flora, Myles, Dean A. A., Howell, Elizabeth E., Dealwis, Chris G.
Published in Acta crystallographica. Section D, Biological crystallography. (01.05.2005)
Published in Acta crystallographica. Section D, Biological crystallography. (01.05.2005)
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Journal Article