GLP-1 receptor activated insulin secretion from pancreatic β-cells: mechanism and glucose dependence
Meloni, A. R., DeYoung, M. B., Lowe, C., Parkes, D. G.
Published in Diabetes, obesity & metabolism (01.01.2013)
Published in Diabetes, obesity & metabolism (01.01.2013)
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Journal Article
A First-Time-in-Human Study of GSK2636771, a Phosphoinositide 3 Kinase Beta-Selective Inhibitor, in Patients with Advanced Solid Tumors
Mateo, Joaquin, Ganji, Gopinath, Lemech, Charlotte, Burris, Howard A, Han, Sae-Won, Swales, Karen, Decordova, Shaun, DeYoung, M Phillip, Smith, Deborah A, Kalyana-Sundaram, Shanker, Wu, Jiuhua, Motwani, Monica, Kumar, Rakesh, Tolson, Jerry M, Rha, Sun Young, Chung, Hyun Cheol, Eder, Joseph P, Sharma, Sunil, Bang, Yung-Jue, Infante, Jeffrey R, Yan, Li, de Bono, Johann S, Arkenau, Hendrik-Tobias
Published in Clinical cancer research (01.10.2017)
Published in Clinical cancer research (01.10.2017)
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Journal Article
Negative feedback control of HIF-1 through REDD1-regulated ROS suppresses tumorigenesis
Horak, Peter, Crawford, Andrew R, Vadysirisack, Douangsone D, Nash, Zachary M, DeYoung, M. Phillip, Sgroi, Dennis, Ellisen, Leif W
Published in Proceedings of the National Academy of Sciences - PNAS (09.03.2010)
Published in Proceedings of the National Academy of Sciences - PNAS (09.03.2010)
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Journal Article
Characterization of GSK2334470, a novel and highly specific inhibitor of PDK1
Najafov, Ayaz, Sommer, Eeva M, Axten, Jeffrey M, Deyoung, M Phillip, Alessi, Dario R
Published in Biochemical journal (15.01.2011)
Published in Biochemical journal (15.01.2011)
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Journal Article
A phase Ib study of GSK3052230, an FGF ligand trap in combination with pemetrexed and cisplatin in patients with malignant pleural mesothelioma
van Brummelen, Emilie M. J., Levchenko, Evgeny, Dómine, Manuel, Fennell, Dean A., Kindler, Hedy L., Viteri, Santiago, Gadgeel, Shirish, López, Pilar Garrido, Kostorov, Vladimir, Morgensztern, Daniel, Orlov, Sergey, Zauderer, Marjorie G., Vansteenkiste, Johan F., Baker-Neblett, Katherine, Vasquez, James, Wang, Xiaowei, Bellovin, David I., Schellens, Jan H. M., Yan, Li, Mitrica, Ionel, DeYoung, M. Phillip, Trigo, José
Published in Investigational new drugs (01.04.2020)
Published in Investigational new drugs (01.04.2020)
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Journal Article
An open-label phase IB study to evaluate GSK3052230 in combination with paclitaxel and carboplatin, or docetaxel, in FGFR1-amplified non-small cell lung cancer
Morgensztern, Daniel, Karaseva, Nina, Felip, Enriqueta, Delgado, Ignacio, Burdaeva, Olga, Dómine, Manuel, Lara, Primo, Paik, Paul K., Lassen, Ulrik, Orlov, Sergey, Trigo, José, Shomova, Marina, Baker-Neblett, Katherine, Vasquez, James, Wang, Xiaowei, Yan, Li, Mitrica, Ionel, DeYoung, M. Phillip, Garrido, Pilar
Published in Lung cancer (Amsterdam, Netherlands) (01.10.2019)
Published in Lung cancer (Amsterdam, Netherlands) (01.10.2019)
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Journal Article
Inter-examination precision of magnitude-based MRI for estimation of segmental hepatic proton density fat fraction in obese subjects
Negrete, Lindsey M., Middleton, Michael S., Clark, Lisa, Wolfson, Tanya, Gamst, Anthony C., Lam, Jessica, Changchien, Chris, Deyoung-Dominguez, Ivan M., Hamilton, Gavin, Loomba, Rohit, Schwimmer, Jeffrey, Sirlin, Claude B.
Published in Journal of magnetic resonance imaging (01.05.2014)
Published in Journal of magnetic resonance imaging (01.05.2014)
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Journal Article
Long-Range Inhibitor-Induced Conformational Regulation of Human IRE1α Endoribonuclease Activity
Concha, Nestor O, Smallwood, Angela, Bonnette, William, Totoritis, Rachel, Zhang, Guofeng, Federowicz, Kelly, Yang, Jingsong, Qi, Hongwei, Chen, Stephanie, Campobasso, Nino, Choudhry, Anthony E, Shuster, Leanna E, Evans, Karen A, Ralph, Jeff, Sweitzer, Sharon, Heerding, Dirk A, Buser, Carolyn A, Su, Dai-Shi, DeYoung, M Phillip
Published in Molecular pharmacology (01.12.2015)
Published in Molecular pharmacology (01.12.2015)
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Journal Article
Early Animal Origin of BACE1 APP/Aβ Proteolytic Function
Langeland, James A, Baumann, Lillian, DeYoung, Eva M, Varella, Raphaela Angelina, Mwenda, Nkatha, Aguirre, Alejandro, Moore, D Blaine
Published in Biology (Basel, Switzerland) (01.05.2024)
Published in Biology (Basel, Switzerland) (01.05.2024)
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Journal Article
Inhibition of FGF/FGFR autocrine signaling in mesothelioma with the FGF ligand trap, FP-1039/GSK3052230
Blackwell, Christina, Sherk, Christian, Fricko, Maggie, Ganji, Gopinath, Barnette, Mary, Hoang, Bao, Tunstead, James, Skedzielewski, Tina, Alsaid, Hasan, Jucker, Beat M, Minthorn, Elisabeth, Kumar, Rakesh, DeYoung, M Phillip
Published in Oncotarget (28.06.2016)
Published in Oncotarget (28.06.2016)
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Journal Article
The Stomatin/Prohibitin/Flotillin/HflK/C Domain of Flotillin-1 Contains Distinct Sequences That Direct Plasma Membrane Localization and Protein Interactions in 3T3-L1 Adipocytes
Liu, Jun, DeYoung, Stephanie M., Zhang, Mei, Dold, Lisa H., Saltiel, Alan R.
Published in The Journal of biological chemistry (22.04.2005)
Published in The Journal of biological chemistry (22.04.2005)
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Journal Article
Prophylactic use of anti-emetic medications reduced nausea and vomiting associated with exenatide treatment: a retrospective analysis of an open-label, parallel-group, single-dose study in healthy subjects
Ellero, C., Han, J., Bhavsar, S., Cirincione, B. B., DeYoung, M. B., Gray, A. L., Yushmanova, I., Anderson, P. W.
Published in Diabetic medicine (01.10.2010)
Published in Diabetic medicine (01.10.2010)
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Journal Article
Activating Inducible T-cell Costimulator Yields Antitumor Activity Alone and in Combination with Anti-PD-1 Checkpoint Blockade
Yadavilli, Sapna, Waight, Jeremy D., Brett, Sara, Bi, Meixia, Zhang, Tianqian, Liu, Yao-Bin, Ellis, Catherine, Turner, David C., Hahn, Ashleigh, Shi, Hong, Seestaller-Wehr, Laura, Jing, Junping, Xie, Qing, Shaik, Jafar Sadik, Ji, Xiao, Gagnon, Robert, Fieles, William, Hook, Laura, Grant, Steven, Hopley, Stephanie, DeYoung, M. Phillip, Blackwell, Christina, Chisamore, Michael, Biddlecombe, Robert, Figueroa, David J., Hopson, Christopher B., Srinivasan, Roopa, Smothers, James, Maio, Michele, Rischin, Danny, Olive, Daniel, Paul, Elaine, Mayes, Patrick A., Hoos, Axel, Ballas, Marc
Published in Cancer research communications (16.08.2023)
Published in Cancer research communications (16.08.2023)
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Journal Article
Changes in integrin expression during adipocyte differentiation
Liu, Jun, DeYoung, Stephanie M., Zhang, Ming, Zhang, Mei, Cheng, Alan, Saltiel, Alan R.
Published in Cell metabolism (01.09.2005)
Published in Cell metabolism (01.09.2005)
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Journal Article
The Roles of Cbl-b and c-Cbl in Insulin-stimulated Glucose Transport
Liu, Jun, DeYoung, Stephanie M., Hwang, Joseph B., O'Leary, Erin E., Saltiel, Alan R.
Published in The Journal of biological chemistry (19.09.2003)
Published in The Journal of biological chemistry (19.09.2003)
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Journal Article
The effects of exenatide bid on metabolic control, medication use and hospitalization in patients with type 2 diabetes mellitus in clinical practice: a systematic review
Best, J. H., Lavillotti, K., DeYoung, M. B., Garrison, L. P.
Published in Diabetes, obesity & metabolism (01.05.2012)
Published in Diabetes, obesity & metabolism (01.05.2012)
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Journal Article