Defining and Combating the Mechanisms of Triclosan Resistance in Clinical Isolates of Staphylococcus aureus
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Published in Antimicrobial Agents and Chemotherapy (01.11.2002)
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Published in Antimicrobial Agents and Chemotherapy (01.10.2002)
Published in Antimicrobial Agents and Chemotherapy (01.10.2002)
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Discovery and preclinical development of AR453588 as an anti-diabetic glucokinase activator
Hinklin, Ronald J., Baer, Brian R., Boyd, Steven A., Chicarelli, Mark D., Condroski, Kevin R., DeWolf, Walter E., Fischer, John, Frank, Michele, Hingorani, Gary P., Lee, Patrice A., Neitzel, Nickolas A., Pratt, Scott A., Singh, Ajay, Sullivan, Francis X., Turner, Timothy, Voegtli, Walter C., Wallace, Eli M., Williams, Lance, Aicher, Thomas D.
Published in Bioorganic & medicinal chemistry (01.01.2020)
Published in Bioorganic & medicinal chemistry (01.01.2020)
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Identification of a New Class of Glucokinase Activators through Structure-Based Design
Hinklin, Ronald J, Boyd, Steven A, Chicarelli, Mark J, Condroski, Kevin R, DeWolf, Walter E, Lee, Patrice A, Lee, Waiman, Singh, Ajay, Thomas, Laurie, Voegtli, Walter C, Williams, Lance, Aicher, Thomas D
Published in Journal of medicinal chemistry (10.10.2013)
Published in Journal of medicinal chemistry (10.10.2013)
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Discovery of 2‑Pyridylureas as Glucokinase Activators
Hinklin, Ronald J, Aicher, Thomas D, Anderson, Deborah A, Baer, Brian R, Boyd, Steven A, Condroski, Kevin R, DeWolf, Walter E, Kraser, Christopher F, McVean, Maralee, Rhodes, Susan P, Sturgis, Hillary L, Voegtli, Walter C, Williams, Lance, Houze, Jonathan B
Published in Journal of medicinal chemistry (09.10.2014)
Published in Journal of medicinal chemistry (09.10.2014)
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Characterization of a novel glucokinase activator in rat and mouse models
Lu, Min, Li, Pingping, Bandyopadhyay, Gautam, Lagakos, William, Dewolf, Jr, Walter E, Alford, Taylor, Chicarelli, Mark Joseph, Williams, Lance, Anderson, Deborah A, Baer, Brian R, McVean, Maralee, Conn, Marion, Véniant, Murielle M, Coward, Peter
Published in PloS one (12.02.2014)
Published in PloS one (12.02.2014)
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5‑Alkyl-2-urea-Substituted Pyridines: Identification of Efficacious Glucokinase Activators with Improved Properties
Kohn, Todd J, Du, Xiaohui, Lai, SuJen, Xiong, YuMei, Komorowski, Renee, Veniant, Murielle, Fu, Zice, Jiao, Xianyun, Pattaropong, Vatee, Chow, David, Cardozo, Mario, Jin, Lixia, Conn, Marion, DeWolf, Walter E, Kraser, Christopher F, Hinklin, Ronald J, Boys, Mark L, Medina, Julio C, Houze, Jonathan, Dransfield, Paul, Coward, Peter
Published in ACS medicinal chemistry letters (14.07.2016)
Published in ACS medicinal chemistry letters (14.07.2016)
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Novel Series of Potent Glucokinase Activators Leading to the Discovery of AM-2394
Dransfield, Paul J, Pattaropong, Vatee, Lai, Sujen, Fu, Zice, Kohn, Todd J, Du, Xiaohui, Cheng, Alan, Xiong, Yumei, Komorowski, Renee, Jin, Lixia, Conn, Marion, Tien, Eric, DeWolf, Walter E, Hinklin, Ronald J, Aicher, Thomas D, Kraser, Christopher F, Boyd, Steven A, Voegtli, Walter C, Condroski, Kevin R, Veniant-Ellison, Murielle, Medina, Julio C, Houze, Jonathan, Coward, Peter
Published in ACS medicinal chemistry letters (14.07.2016)
Published in ACS medicinal chemistry letters (14.07.2016)
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Indole Naphthyridinones as Inhibitors of Bacterial Enoyl-ACP Reductases FabI and FabK
Seefeld, Mark A, Miller, William H, Newlander, Kenneth A, Burgess, Walter J, DeWolf, Walter E, Elkins, Patricia A, Head, Martha S, Jakas, Dalia R, Janson, Cheryl A, Keller, Paul M, Manley, Peter J, Moore, Terrance D, Payne, David J, Pearson, Stewart, Polizzi, Brian J, Qiu, Xiayang, Rittenhouse, Stephen F, Uzinskas, Irene N, Wallis, Nicola G, Huffman, William F
Published in Journal of medicinal chemistry (24.04.2003)
Published in Journal of medicinal chemistry (24.04.2003)
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Potent and Selective Nonpeptide Inhibitors of Caspases 3 and 7 Inhibit Apoptosis and Maintain Cell Functionality
Lee, Dennis, Long, Scott A., Adams, Jerry L., Chan, George, Vaidya, Kalindi S., Francis, Terry A., Kikly, Kristine, Winkler, James D., Sung, Chiu-Mei, Debouck, Christine, Richardson, Susan, Levy, Mark A., DeWolf, Walter E., Keller, Paul M., Tomaszek, Thaddeus, Head, Martha S., Ryan, M.Dominic, Haltiwanger, R.Curtis, Liang, Po-Huang, Janson, Cheryl A., McDevitt, Patrick J., Johanson, Kyung, Concha, Nestor O., Chan, Winnie, Abdel-Meguid, Sherin S., Badger, Alison M., Lark, Michael W., Nadeau, Daniel P., Suva, Larry J., Gowen, Maxine, Nuttall, Mark E.
Published in The Journal of biological chemistry (26.05.2000)
Published in The Journal of biological chemistry (26.05.2000)
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Characterization of Streptococcus pneumoniae enoyl-(acyl-carrier protein) reductase (FabK)
Marrakchi, Hedia, Dewolf, Jr, Walter E, Quinn, Chad, West, Joshua, Polizzi, Brian J, So, Chi Y, Holmes, David J, Reed, Shannon L, Heath, Richard J, Payne, David J, Rock, Charles O, Wallis, Nicola G
Published in Biochemical journal (15.03.2003)
Published in Biochemical journal (15.03.2003)
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Discovery of Aminopyridine-Based Inhibitors of Bacterial Enoyl-ACP Reductase (FabI)
Miller, William H, Seefeld, Mark A, Newlander, Kenneth A, Uzinskas, Irene N, Burgess, Walter J, Heerding, Dirk A, Yuan, Catherine C. K, Head, Martha S, Payne, David J, Rittenhouse, Stephen F, Moore, Terrance D, Pearson, Stewart C, Berry, Valerie, DeWolf, Walter E, Keller, Paul M, Polizzi, Brian J, Qiu, Xiayang, Janson, Cheryl A, Huffman, William F
Published in Journal of medicinal chemistry (18.07.2002)
Published in Journal of medicinal chemistry (18.07.2002)
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Inhibition of caspase-3-like activity prevents apoptosis while retaining functionality of human chondrocytes in vitro
Nuttall, Mark E., Nadeau, Daniel P., Fisher, Paul W., Wang, Feilan, Keller, Paul M., Dewolf Jr, Walter E., Goldring, Mary B., Badger, Alison M., Lee, Dennis, Levy, Mark A., Gowen, Maxine, Lark, Michael W.
Published in Journal of orthopaedic research (01.05.2000)
Published in Journal of orthopaedic research (01.05.2000)
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Apoptosis in polycystic kidney disease: involvement of caspases
Ali, Shujath M, Wong, Victoria Y, Kikly, Kristine, Fredrickson, Todd A, Keller, Paul M, DeWolf, Walter E., Jr, Lee, Dennis, Brooks, David P
Published in American journal of physiology. Regulatory, integrative and comparative physiology (01.03.2000)
Published in American journal of physiology. Regulatory, integrative and comparative physiology (01.03.2000)
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Endothelin-Converting Enzyme: Substrate Specificity and Inhibition by Novel Analogs of Phosphoramidon
Keller, Paul M., Lee, Chao-Pin, Fenwick, Ashley E., Atkinson, Steven T., Elliott, John D., DeWolf, Jr, Walter E.
Published in Biochemical and biophysical research communications (14.06.1996)
Published in Biochemical and biophysical research communications (14.06.1996)
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TL1, a Novel Tumor Necrosis Factor-like Cytokine, Induces Apoptosis in Endothelial Cells
Yue, Tian-Li, Ni, Jian, Romanic, Anne M., Gu, Juan-Li, Keller, Paul, Wang, Chuanlin, Kumar, Sanjay, Yu, Guo-liang, Hart, Timothy K., Wang, Xinkang, Xia, Zhengui, DeWolf, Walter E., Feuerstein, Giora Z.
Published in The Journal of biological chemistry (01.01.1999)
Published in The Journal of biological chemistry (01.01.1999)
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FAB I inhibitors
Miller, William H, Newlander, Kenneth A, Seefeld, Mark A, Uzinskas, Irene N, Dewolf, Jr, Walter E, Jakas, Dalia R
Year of Publication 08.05.2012
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Year of Publication 08.05.2012
Patent
Fab I inhibitors
Miller, William H, Newlander, Kenneth A, Seefeld, Mark A, Uzinskas, Irene N, Dewolf, Jr, Walter E, Jakas, Dalia R
Year of Publication 07.09.2010
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Year of Publication 07.09.2010
Patent