MLi-2, a Potent, Selective, and Centrally Active Compound for Exploring the Therapeutic Potential and Safety of LRRK2 Kinase Inhibition
Fell, Matthew J, Mirescu, Christian, Basu, Kallol, Cheewatrakoolpong, Boonlert, DeMong, Duane E, Ellis, J Michael, Hyde, Lynn A, Lin, Yinghui, Markgraf, Carrie G, Mei, Hong, Miller, Michael, Poulet, Frederique M, Scott, Jack D, Smith, Michelle D, Yin, Zhizhang, Zhou, Xiaoping, Parker, Eric M, Kennedy, Matthew E, Morrow, John A
Published in The Journal of pharmacology and experimental therapeutics (01.12.2015)
Published in The Journal of pharmacology and experimental therapeutics (01.12.2015)
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Journal Article
Asymmetric Synthesis of (2S,3R)-Capreomycidine and the Total Synthesis of Capreomycin IB
DeMong, Duane E, Williams, Robert M
Published in Journal of the American Chemical Society (16.07.2003)
Published in Journal of the American Chemical Society (16.07.2003)
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Journal Article
Discovery of a 3‑(4-Pyrimidinyl) Indazole (MLi-2), an Orally Available and Selective Leucine-Rich Repeat Kinase 2 (LRRK2) Inhibitor that Reduces Brain Kinase Activity
Scott, Jack D, DeMong, Duane E, Greshock, Thomas J, Basu, Kallol, Dai, Xing, Harris, Joel, Hruza, Alan, Li, Sarah W, Lin, Sue-Ing, Liu, Hong, Macala, Megan K, Hu, Zhiyong, Mei, Hong, Zhang, Honglu, Walsh, Paul, Poirier, Marc, Shi, Zhi-Cai, Xiao, Li, Agnihotri, Gautam, Baptista, Marco A. S, Columbus, John, Fell, Matthew J, Hyde, Lynn A, Kuvelkar, Reshma, Lin, Yinghui, Mirescu, Christian, Morrow, John A, Yin, Zhizhang, Zhang, Xiaoping, Zhou, Xiaoping, Chang, Ronald K, Embrey, Mark W, Sanders, John M, Tiscia, Heather E, Drolet, Robert E, Kern, Jonathan T, Sur, Sylvie M, Renger, John J, Bilodeau, Mark T, Kennedy, Matthew E, Parker, Eric M, Stamford, Andrew W, Nargund, Ravi, McCauley, John A, Miller, Michael W
Published in Journal of medicinal chemistry (13.04.2017)
Published in Journal of medicinal chemistry (13.04.2017)
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Journal Article
Discovery and Optimization of Potent, Selective, and Brain-Penetrant 1-Heteroaryl-1 H -Indazole LRRK2 Kinase Inhibitors for the Treatment of Parkinson's Disease
Candito, David A, Simov, Vladimir, Gulati, Anmol, Kattar, Solomon, Chau, Ryan W, Lapointe, Blair T, Methot, Joey L, DeMong, Duane E, Graham, Thomas H, Kurukulasuriya, Ravi, Keylor, Mitchell H, Tong, Ling, Morriello, Gregori J, Acton, John J, Pio, Barbara, Liu, Weiguo, Scott, Jack D, Ardolino, Michael J, Martinot, Theodore A, Maddess, Matthew L, Yan, Xin, Gunaydin, Hakan, Palte, Rachel L, McMinn, Spencer E, Nogle, Lisa, Yu, Hongshi, Minnihan, Ellen C, Lesburg, Charles A, Liu, Ping, Su, Jing, Hegde, Laxminarayan G, Moy, Lily Y, Woodhouse, Janice D, Faltus, Robert, Xiong, Tina, Ciaccio, Paul, Piesvaux, Jennifer A, Otte, Karin M, Kennedy, Matthew E, Bennett, David Jonathan, DiMauro, Erin F, Fell, Matthew J, Neelamkavil, Santhosh, Wood, Harold B, Fuller, Peter H, Ellis, J Michael
Published in Journal of medicinal chemistry (22.12.2022)
Published in Journal of medicinal chemistry (22.12.2022)
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Journal Article
A Novel Method for the Preparation of 4‑Arylimidazolones
DeMong, Duane E, Ng, Irene, Miller, Michael W, Stamford, Andrew W
Published in Organic letters (07.06.2013)
Published in Organic letters (07.06.2013)
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Journal Article
Synthesis, Structure−Activity Relationship and in Vivo Antiinflammatory Efficacy of Substituted Dipiperidines as CCR2 Antagonists
Xia, Mingde, Hou, Cuifen, DeMong, Duane E, Pollack, Scott R, Pan, Meng, Brackley, James A, Jain, Nareshkumar, Gerchak, Chrissy, Singer, Monica, Malaviya, Ravi, Matheis, Michele, Olini, Gil, Cavender, Druie, Wachter, Michael
Published in Journal of medicinal chemistry (15.11.2007)
Published in Journal of medicinal chemistry (15.11.2007)
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Journal Article
STING 효능제로서의 벤조티오펜 및 관련 화합물
CASH BRANDON D, CUMMING JARED N, JEWELL JAMES P, LARSEN MATTHEW A, DEMONG DUANE E, ALTMAN MICHAEL D, LIM JONGWON, HENDERSON TIMOTHY J, LU MIN, CHILDERS MATTHEW LLOYD, OTTE RYAN D, HAIDLE ANDREW MARC, TROTTER BENJAMIN WESLEY
Year of Publication 11.12.2020
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Year of Publication 11.12.2020
Patent
Asymmetric Synthesis of (+)-Hypusine
Jain, Rajendra P, Albrecht, Brian K, DeMong, Duane E, Williams, Robert M
Published in Organic letters (27.12.2001)
Published in Organic letters (27.12.2001)
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Journal Article
ANTIDIABETIC BICYCLIC COMPOUNDS
CHOBANIAN HARRY R, HAGMANN WILLIAM K, MARCANTONIO KAREN M, XIAO DONG, CRESPO ALEJANDRO, DEMONG DUANE E, MILLER MICHAEL, PIO BARBARA, BROCKUNIER LINDA L, CHEN HELEN, PLUMMER CHRISTOPHER W, GUO YAN, CLEMENTS MATTHEW J
Year of Publication 21.10.2015
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Year of Publication 21.10.2015
Patent
Discovery and Optimization of Potent, Selective, and Brain-Penetrant 1‑Heteroaryl‑1H‑Indazole LRRK2 Kinase Inhibitors for the Treatment of Parkinson’s Disease
Candito, David A., Simov, Vladimir, Gulati, Anmol, Kattar, Solomon, Chau, Ryan W., Lapointe, Blair T., Methot, Joey L., DeMong, Duane E., Graham, Thomas H., Kurukulasuriya, Ravi, Keylor, Mitchell H., Tong, Ling, Morriello, Gregori J., Acton, John J., Pio, Barbara, Liu, Weiguo, Scott, Jack D., Ardolino, Michael J., Martinot, Theodore A., Maddess, Matthew L., Yan, Xin, Gunaydin, Hakan, Palte, Rachel L., McMinn, Spencer E., Nogle, Lisa, Yu, Hongshi, Minnihan, Ellen C., Lesburg, Charles A., Liu, Ping, Su, Jing, Hegde, Laxminarayan G., Moy, Lily Y., Woodhouse, Janice D., Faltus, Robert, Xiong, Tina, Ciaccio, Paul, Piesvaux, Jennifer A., Otte, Karin M., Kennedy, Matthew E., Bennett, David Jonathan, DiMauro, Erin F., Fell, Matthew J., Neelamkavil, Santhosh, Wood, Harold B., Fuller, Peter H., Ellis, J. Michael
Published in Journal of medicinal chemistry (22.12.2022)
Published in Journal of medicinal chemistry (22.12.2022)
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Journal Article
ChemInform Abstract: A Novel Method for the Preparation of 4-Arylimidazolones
DeMong, Duane E., Ng, Irene, Miller, Michael W., Stamford, Andrew W.
Published in ChemInform (01.10.2013)
Published in ChemInform (01.10.2013)
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Journal Article
A Novel Carbohydrate-Glycosphingolipid Interaction between a β-(1–3)-Glucan Immunomodulator, PGG-glucan, and Lactosylceramide of Human Leukocytes
Zimmerman, Janet W., Lindermuth, Johanna, Fish, Pamela A., Palace, Gerard P., Stevenson, Tom T., DeMong, Duane E.
Published in The Journal of biological chemistry (21.08.1998)
Published in The Journal of biological chemistry (21.08.1998)
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Journal Article
ADENOSINE A2A AND A2B RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITIONS AND USE THEREOF
MORENO, Jesus, ALI, Amjad, PLUMMER, Christopher W, DEMONG, Duane E, CUMMING, Jared N, SATHER, Aaron C, HENNESSY, Elisabeth T, JOHNSON, Rebecca Elizabeth, LARSEN, Matthew A, KAPLAN, William P, LI, Derun, MANSOOR, Umar Faruk, DENG, Qiaolin
Year of Publication 06.06.2024
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Year of Publication 06.06.2024
Patent
ADENOSINE RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITIONS AND THEIR USE THEREOF
BRILL, Zachary G, ALI, Amjad, PLUMMER, Christopher W, DEMONG, Duane E, LIM, Yeon-Hee, SU, Jing, CHRISTIAN, Alec Hiroshi, CUMMING, Jared N, RICO DUQUE, Jenny Lorena, HENNESSY, Elisabeth T, LI, Derun
Year of Publication 24.08.2023
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Year of Publication 24.08.2023
Patent
Aza-benzothiophene compounds as STING agonists
Lu, Min, Trotter, Benjamin Wesley, Cash, Brandon D, Cumming, Jared N, DeMong, Duane E, Truong, Quang T, Altman, Michael D, Jewell, James P, Taoka, Brandon M, Haidle, Andrew M, Larsen, Matthew A, Otte, Ryan D
Year of Publication 18.07.2023
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Year of Publication 18.07.2023
Patent
Benzothiophenes and related compounds as sting agonists
TROTTER, Benjamin Wesley, LU, Min, DEMONG, Duane E, CHILDERS, Matthew Lloyd, CUMMING, Jared N, JEWELL, James P, OTTE, Ryan D, LARSEN, Matthew A, HAIDLE, Andrew Marc, LIM, Jongwon, CASH, Brandon D, HENDERSON, Timothy, ALTMAN, Michael D
Year of Publication 11.08.2022
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Year of Publication 11.08.2022
Patent
AZA-BENZOTHIOPHENE COMPOUNDS AS STING AGONISTS
CUMMING, Jared, N, TROTTER, Benjamin Wesley, CASH, Brandon, D, LU, Min, LARSEN, Matthew, A, TAOKA, Brandon, M, DEMONG, Duane, E, HAIDLE, Andrew, M, OTTE, Ryan, D, JEWELL, James, P, TRUONG, Quang, T, ALTMAN, Michael, D
Year of Publication 29.12.2021
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Year of Publication 29.12.2021
Patent