The first potent inhibitor of squalene synthase: a profound contribution of an ether oxygen to inhibitor-enzyme interaction
Biller, Scott A, Sofia, Michael J, DeLange, Barbara, Forster, Cornelia, Gordon, Eric M, Harrity, Thomas, Rich, Lois C, Ciosek, Carl P
Published in Journal of the American Chemical Society (01.10.1991)
Published in Journal of the American Chemical Society (01.10.1991)
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Phosphorus-containing inhibitors of HMG-CoA reductase. I. 4-[(2-Arylethyl)hydroxyphosphinyl]-3-hydroxybutanoic acids: a new class of cell selective inhibitors of cholesterol biosynthesis
Karanewsky, Donald S, Badia, Michael C, Ciosek, Carl P, Robl, Jeffrey A, Sofia, Michael J, Simpkins, Ligaya M, DeLange, Barbara, Harrity, Thomas W, Biller, Scott A, Gordon, Eric M
Published in Journal of medicinal chemistry (01.11.1990)
Published in Journal of medicinal chemistry (01.11.1990)
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Journal Article
Phosphorus-containing inhibitors of HMG-CoA reductase. 1. 4-[(2-arylethyl)hydroxyphosphinyl]-3-hydroxy-butanoic acids: a new class of cell-selective inhibitors of cholesterol biosynthesis
Karanewsky, D S, Badia, M C, Ciosek, Jr, C P, Robl, J A, Sofia, M J, Simpkins, L M, DeLange, B, Harrity, T W, Biller, S A, Gordon, E M
Published in Journal of medicinal chemistry (01.11.1990)
Published in Journal of medicinal chemistry (01.11.1990)
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Journal Article