Synthetic Approaches to New Drugs Approved during 2018
Flick, Andrew C, Leverett, Carolyn A, Ding, Hong X, McInturff, Emma, Fink, Sarah J, Helal, Christopher J, DeForest, Jacob C, Morse, Peter D, Mahapatra, Subham, O’Donnell, Christopher J
Published in Journal of medicinal chemistry (08.10.2020)
Published in Journal of medicinal chemistry (08.10.2020)
Get full text
Journal Article
Discovery of compounds that reactivate p53 mutants in vitro and in vivo
Durairaj, Geetha, Demir, Özlem, Lim, Bryant, Baronio, Roberta, Tifrea, Delia, Hall, Linda V., DeForest, Jacob C., Lauinger, Linda, Jebril Fallatah, Maryam M., Yu, Clinton, Bae, Hosung, Lin, Da-Wei, Kim, Jin Kwang, Salehi, Faezeh, Jang, Cholsoon, Qiao, Feng, Lathrop, Richard H., Huang, Lan, Edwards, Robert, Rychnovsky, Scott, Amaro, Rommie E., Kaiser, Peter
Published in Cell chemical biology (15.09.2022)
Published in Cell chemical biology (15.09.2022)
Get full text
Journal Article
Synthetic Approaches to the New Drugs Approved During 2022
France, Scott P., Lindsey, Erick A., McInturff, Emma L., Berritt, Simon, Carney, Daniel W., DeForest, Jacob C., Fink, Sarah J., Flick, Andrew C., Gibson, Tony S., Gray, Kaitlyn, Johnson, Amber M., Leverett, Carolyn A., Liu, Yiyang, Mahapatra, Subham, Watson, Rebecca B.
Published in Journal of medicinal chemistry (28.03.2024)
Published in Journal of medicinal chemistry (28.03.2024)
Get full text
Journal Article
Synthetic Approaches to the New Drugs Approved During 2020
Flick, Andrew C., Leverett, Carolyn A., Ding, Hong X., McInturff, Emma L., Fink, Sarah J., Mahapatra, Subham, Carney, Daniel W., Lindsey, Erick A., DeForest, Jacob C., France, Scott P., Berritt, Simon, Bigi-Botterill, Simone V., Gibson, Tony S., Watson, Rebecca B., Liu, Yiyang, O’Donnell, Christopher J.
Published in Journal of medicinal chemistry (28.07.2022)
Published in Journal of medicinal chemistry (28.07.2022)
Get full text
Journal Article
Second-Generation Synthesis of (+)-Fastigiatine Inspired by Conformational Studies
DeForest, Jacob C, Samame, Renzo A, Suryn, Gregory, Burtea, Alexander, Rychnovsky, Scott D
Published in Journal of organic chemistry (17.08.2018)
Published in Journal of organic chemistry (17.08.2018)
Get full text
Journal Article
Synthetic Approaches to the New Drugs Approved During 2021
McInturff, Emma L., France, Scott P., Leverett, Carolyn A., Flick, Andrew C., Lindsey, Erick A., Berritt, Simon, Carney, Daniel W., DeForest, Jacob C., Ding, Hong X., Fink, Sarah J., Gibson, Tony S., Gray, Kaitlyn, Hubbell, Aran K., Johnson, Amber M., Liu, Yiyang, Mahapatra, Subham, McAlpine, Indrawan J., Watson, Rebecca B., O’Donnell, Christopher J.
Published in Journal of medicinal chemistry (10.08.2023)
Published in Journal of medicinal chemistry (10.08.2023)
Get full text
Journal Article
Development of a Nitrene-Type Rearrangement for the Commercial Route of the JAK1 Inhibitor Abrocitinib
Connor, Christina G, DeForest, Jacob C, Dietrich, Phil, Do, Nga M, Doyle, Kevin M, Eisenbeis, Shane, Greenberg, Elizabeth, Griffin, Sarah H, Jones, Brian P, Jones, Kris N, Karmilowicz, Michael, Kumar, Rajesh, Lewis, Chad A, McInturff, Emma L, McWilliams, J. Christopher, Mehta, Ruchi, Nguyen, Bao D, Rane, Anil M, Samas, Brian, Sitter, Barbara J, Ward, Howard W, Webster, Mark E
Published in Organic process research & development (19.03.2021)
Published in Organic process research & development (19.03.2021)
Get full text
Journal Article
4′,4‴,7,7″-Tetra‑O‑methylcupressuflavone Inhibits Seed Germination of Lactuca sativa
DeForest, Jacob C, Du, Lin, Joyner, P. Matthew
Published in Journal of natural products (Washington, D.C.) (25.04.2014)
Published in Journal of natural products (Washington, D.C.) (25.04.2014)
Get full text
Journal Article