Nitric oxide donors and selective carbonic anhydrase inhibitors: a dual pharmacological approach for the treatment of glaucoma, cancer and osteoporosis
Carradori, Simone, Mollica, Adriano, De Monte, Celeste, Ganese, Arianna, Supuran, Claudiu T
Published in Molecules (31.03.2015)
Published in Molecules (31.03.2015)
Get full text
Journal Article
Book Review
Design, synthesis and evaluation of N-substituted saccharin derivatives as selective inhibitors of tumor-associated carbonic anhydrase XII
D’Ascenzio, Melissa, Carradori, Simone, De Monte, Celeste, Secci, Daniela, Ceruso, Mariangela, Supuran, Claudiu T.
Published in Bioorganic & medicinal chemistry (15.03.2014)
Published in Bioorganic & medicinal chemistry (15.03.2014)
Get full text
Journal Article
A novel library of saccharin and acesulfame derivatives as potent and selective inhibitors of carbonic anhydrase IX and XII isoforms
Carradori, Simone, Secci, Daniela, De Monte, Celeste, Mollica, Adriano, Ceruso, Mariangela, Akdemir, Atilla, Sobolev, Anatoly P., Codispoti, Rossella, De Cosmi, Federica, Guglielmi, Paolo, Supuran, Claudiu T.
Published in Bioorganic & medicinal chemistry (01.03.2016)
Published in Bioorganic & medicinal chemistry (01.03.2016)
Get full text
Journal Article
Dual Cyclooxygenase and Carbonic Anhydrase Inhibition by Nonsteroidal Anti-Inflammatory Drugs for the Treatment of Cancer
De Monte, Celeste, Carradori, Simone, Gentili, Andrea, Mollica, Adriano, Trisciuoglio, Daniela, Supuran, Claudiu T
Published in Current medicinal chemistry (01.01.2015)
Published in Current medicinal chemistry (01.01.2015)
Get more information
Journal Article
Design, synthesis and biological activity of selective hCAs inhibitors based on 2-(benzylsulfinyl)benzoic acid scaffold
Rotondi, Giulia, Guglielmi, Paolo, Carradori, Simone, Secci, Daniela, De Monte, Celeste, De Filippis, Barbara, Maccallini, Cristina, Amoroso, Rosa, Cirilli, Roberto, Akdemir, Atilla, Angeli, Andrea, Supuran, Claudiu T.
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2019)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2019)
Get full text
Journal Article
Identification of the stereochemical requirements in the 4-aryl-2-cycloalkylidenhydrazinylthiazole scaffold for the design of selective human monoamine oxidase B inhibitors
D’Ascenzio, Melissa, Carradori, Simone, Secci, Daniela, Mannina, Luisa, Sobolev, Anatoly P., De Monte, Celeste, Cirilli, Roberto, Yáñez, Matilde, Alcaro, Stefano, Ortuso, Francesco
Published in Bioorganic & medicinal chemistry (15.05.2014)
Published in Bioorganic & medicinal chemistry (15.05.2014)
Get full text
Journal Article
Synthesis and biological evaluation of anti-Toxoplasma gondii activity of a novel scaffold of thiazolidinone derivatives
Carradori, Simone, Secci, Daniela, Bizzarri, Bruna, Chimenti, Paola, De Monte, Celeste, Guglielmi, Paolo, Campestre, Cristina, Rivanera, Daniela, Bordón, Claudia, Jones-Brando, Lorraine
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2017)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2017)
Get full text
Journal Article
Geographical characterization by MAE-HPLC and NIR methodologies and carbonic anhydrase inhibition of Saffron components
Nescatelli, Riccardo, Carradori, Simone, Marini, Federico, Caponigro, Vicky, Bucci, Remo, De Monte, Celeste, Mollica, Adriano, Mannina, Luisa, Ceruso, Mariangela, Supuran, Claudiu T., Secci, Daniela
Published in Food chemistry (15.04.2017)
Published in Food chemistry (15.04.2017)
Get full text
Journal Article
Anti-Candida activity and cytotoxicity of a large library of new N-substituted-1,3-thiazolidin-4-one derivatives
De Monte, Celeste, Carradori, Simone, Bizzarri, Bruna, Bolasco, Adriana, Caprara, Federica, Mollica, Adriano, Rivanera, Daniela, Mari, Emanuela, Zicari, Alessandra, Akdemir, Atilla, Secci, Daniela
Published in European journal of medicinal chemistry (01.01.2016)
Published in European journal of medicinal chemistry (01.01.2016)
Get full text
Journal Article
Novel 1,3-thiazolidin-4-one derivatives as promising anti-Candida agents endowed with anti-oxidant and chelating properties
Secci, Daniela, Carradori, Simone, Bizzarri, Bruna, Chimenti, Paola, De Monte, Celeste, Mollica, Adriano, Rivanera, Daniela, Zicari, Alessandra, Mari, Emanuela, Zengin, Gokhan, Aktumsek, Abdurrahman
Published in European journal of medicinal chemistry (19.07.2016)
Published in European journal of medicinal chemistry (19.07.2016)
Get full text
Journal Article
Design, synthesis and biochemical evaluation of novel multi-target inhibitors as potential anti-Parkinson agents
Carradori, Simone, Ortuso, Francesco, Petzer, Anél, Bagetta, Donatella, De Monte, Celeste, Secci, Daniela, De Vita, Daniela, Guglielmi, Paolo, Zengin, Gokhan, Aktumsek, Abdurrahman, Alcaro, Stefano, Petzer, Jacobus P.
Published in European journal of medicinal chemistry (01.01.2018)
Published in European journal of medicinal chemistry (01.01.2018)
Get full text
Journal Article
Computational investigation of the selectivity of salen and tetrahydrosalen compounds towards the tumor-associated hCA XII isozyme
Akdemir, Atilla, De Monte, Celeste, Carradori, Simone, Supuran, Claudiu T.
Published in Journal of enzyme inhibition and medicinal chemistry (01.02.2015)
Published in Journal of enzyme inhibition and medicinal chemistry (01.02.2015)
Get full text
Journal Article
Synthesis, biological evaluation and quantitative structure-active relationships of 1,3-thiazolidin-4-one derivatives. A promising chemical scaffold endowed with high antifungal potency and low cytotoxicity
Carradori, Simone, Bizzarri, Bruna, D'Ascenzio, Melissa, De Monte, Celeste, Grande, Rossella, Rivanera, Daniela, Zicari, Alessanda, Mari, Emanuela, Sabatino, Manuela, Patsilinakos, Alexandros, Ragno, Rino, Secci, Daniela
Published in European journal of medicinal chemistry (10.11.2017)
Published in European journal of medicinal chemistry (10.11.2017)
Get full text
Journal Article
Cyclic tertiary sulfamates: Selective inhibition of the tumor-associated carbonic anhydrases IX and XII by N- and O-substituted acesulfame derivatives
De Monte, Celeste, Carradori, Simone, Secci, Daniela, D'Ascenzio, Melissa, Vullo, Daniela, Ceruso, Mariangela, Supuran, Claudiu T.
Published in European journal of medicinal chemistry (12.09.2014)
Published in European journal of medicinal chemistry (12.09.2014)
Get full text
Journal Article
Modern extraction techniques and their impact on the pharmacological profile of Serenoa repens extracts for the treatment of lower urinary tract symptoms
De Monte, Celeste, Carradori, Simone, Granese, Arianna, Di Pierro, Giovanni Battista, Leonardo, Costantino, De Nunzio, Cosimo
Published in BMC urology (11.08.2014)
Published in BMC urology (11.08.2014)
Get full text
Journal Article
Design, synthesis and biological characterization of thiazolidin-4-one derivatives as promising inhibitors of Toxoplasma gondii
D'Ascenzio, Melissa, Bizzarri, Bruna, De Monte, Celeste, Carradori, Simone, Bolasco, Adriana, Secci, Daniela, Rivanera, Daniela, Faulhaber, Nathan, Bordón, Claudia, Jones-Brando, Lorraine
Published in European journal of medicinal chemistry (30.10.2014)
Published in European journal of medicinal chemistry (30.10.2014)
Get full text
Journal Article
Evaluation of a large library of (thiazol-2-yl)hydrazones and analogues as histone acetyltransferase inhibitors: Enzyme and cellular studies
Carradori, Simone, Rotili, Dante, De Monte, Celeste, Lenoci, Alessia, D'Ascenzio, Melissa, Rodriguez, Veronica, Filetici, Patrizia, Miceli, Marco, Nebbioso, Angela, Altucci, Lucia, Secci, Daniela, Mai, Antonello
Published in European journal of medicinal chemistry (10.06.2014)
Published in European journal of medicinal chemistry (10.06.2014)
Get full text
Journal Article
Bioactive compounds of Crocus sativus L. and their semi-synthetic derivatives as promising anti-Helicobacter pylori, anti-malarial and anti-leishmanial agents
De Monte, Celeste, Bizzarri, Bruna, Gidaro, Maria Concetta, Carradori, Simone, Mollica, Adriano, Luisi, Grazia, Granese, Arianna, Alcaro, Stefano, Costa, Giosuè, Basilico, Nicoletta, Parapini, Silvia, Scaltrito, Maria Maddalena, Masia, Carla, Sisto, Francesca
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2015)
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2015)
Get full text
Journal Article
New amide derivatives of Probenecid as selective inhibitors of carbonic anhydrase IX and XII: Biological evaluation and molecular modelling studies
Carradori, Simone, Mollica, Adriano, Ceruso, Mariangela, D’Ascenzio, Melissa, De Monte, Celeste, Chimenti, Paola, Sabia, Rocchina, Akdemir, Atilla, Supuran, Claudiu T.
Published in Bioorganic & medicinal chemistry (01.07.2015)
Published in Bioorganic & medicinal chemistry (01.07.2015)
Get full text
Journal Article
Salen and tetrahydrosalen derivatives act as effective inhibitors of the tumor-associated carbonic anhydrase XII—A new scaffold for designing isoform-selective inhibitors
Carradori, Simone, De Monte, Celeste, D’Ascenzio, Melissa, Secci, Daniela, Celik, Gulsah, Ceruso, Mariangela, Vullo, Daniela, Scozzafava, Andrea, Supuran, Claudiu T.
Published in Bioorganic & medicinal chemistry letters (15.12.2013)
Published in Bioorganic & medicinal chemistry letters (15.12.2013)
Get full text
Journal Article