α-Synuclein O-GlcNAcylation alters aggregation and toxicity, revealing certain residues as potential inhibitors of Parkinson’s disease
Levine, Paul M., Galesic, Ana, Balana, Aaron T., Mahul-Mellier, Anne-Laure, Navarro, Mariana X., De Leon, Cesar A., Lashuel, Hilal A., Pratt, Matthew R.
Published in Proceedings of the National Academy of Sciences - PNAS (29.01.2019)
Published in Proceedings of the National Academy of Sciences - PNAS (29.01.2019)
Get full text
Journal Article
The Sulfur-Linked Analogue of O‑GlcNAc (S-GlcNAc) Is an Enzymatically Stable and Reasonable Structural Surrogate for O‑GlcNAc at the Peptide and Protein Levels
De Leon, Cesar A, Levine, Paul M, Craven, Timothy W, Pratt, Matthew R
Published in Biochemistry (Easton) (11.07.2017)
Published in Biochemistry (Easton) (11.07.2017)
Get full text
Journal Article
Simple and Efficient Preparation of O- and S‑GlcNAcylated Amino Acids through InBr3‑Catalyzed Synthesis of β‑N‑Acetylglycosides from Commercially Available Reagents
De Leon, Cesar A, Lang, Geoffrey, Saavedra, Marcos I, Pratt, Matthew R
Published in Organic letters (17.08.2018)
Published in Organic letters (17.08.2018)
Get full text
Journal Article
Regulated induced proximity targeting chimeras—RIPTACs—A heterobifunctional small molecule strategy for cancer selective therapies
Raina, Kanak, Forbes, Chris D., Stronk, Rebecca, Rappi, Jonathan P., Eastman, Kyle J., Zaware, Nilesh, Yu, Xinheng, Li, Hao, Bhardwaj, Amit, Gerritz, Samuel W., Forgione, Mia, Hundt, Abigail, King, Madeline P., Posner, Zoe M., Correia, Allison D., McGovern, Andrew, Puleo, David E., Chenard, Rebekka, Mousseau, James J., Vergara, J. Ignacio, Garvin, Ethan, Macaluso, Jennifer, Martin, Michael, Bassoli, Kyle, Jones, Kelli, Garcia, Marco, Howard, Katia, Yaggi, Madeleine, Smith, Levi M., Chen, Jinshan M., Mayfield, Andrew B., De Leon, Cesar A., Hines, John, Kayser-Bricker, Katherine J., Crews, Craig M.
Published in Cell chemical biology (15.08.2024)
Published in Cell chemical biology (15.08.2024)
Get full text
Journal Article
Simple and Efficient Preparation of O- and S-GlcNAcylated Amino Acids through InBr 3 -Catalyzed Synthesis of β- N-Acetylglycosides from Commercially Available Reagents
De Leon, Cesar A, Lang, Geoffrey, Saavedra, Marcos I, Pratt, Matthew R
Published in Organic letters (17.08.2018)
Published in Organic letters (17.08.2018)
Get full text
Journal Article
Simple and Efficient Preparation of O- and S-GIcNAcylated Amino Acids through InBr3-Catalyzed Synthesis of beta-N-Acetylglycosides from Commercially Available Reagents
De Leon, Cesar A., Lang, Geoffrey, Saavedra, Marcos I., Pratt, Matthew R.
Published in Organic letters (17.08.2018)
Published in Organic letters (17.08.2018)
Get full text
Journal Article
Regulated Induced Proximity Targeting Chimeras (RIPTACs): a Novel Heterobifunctional Small Molecule Therapeutic Strategy for Killing Cancer Cells Selectively
Raina, Kanak, Forbes, Chris D, Stronk, Rebecca, Rappi, Jr, Jonathan P, Eastman, Kyle J, Gerritz, Samuel W, Yu, Xinheng, Li, Hao, Bhardwaj, Amit, Forgione, Mia, Hundt, Abigail, King, Madeline P, Posner, Zoe M, Denny, Allison, McGovern, Andrew, Puleo, David E, Garvin, Ethan, Chenard, Rebekka, Zaware, Nilesh, Mousseau, James J, Macaluso, Jennifer, Martin, Michael, Bassoli, Kyle, Jones, Kelli, Garcia, Marco, Howard, Katia, Smith, Levi M, Chen, Jinshan M, De Leon, Cesar A, Hines, John, Kayser-Bricker, Katherine J, Crews, Craig M
Published in bioRxiv (02.01.2023)
Published in bioRxiv (02.01.2023)
Get full text
Journal Article
Paper