Novel Class of Benzoic Acid Ester Derivatives as Potent PDE4 Inhibitors for Inhaled Administration in the Treatment of Respiratory Diseases
Armani, Elisabetta, Amari, Gabriele, Rizzi, Andrea, Fanti, Renato De, Ghidini, Eleonora, Capaldi, Carmelida, Carzaniga, Laura, Caruso, Paola, Guala, Matilde, Peretto, Ilaria, La Porta, Elena, Bolzoni, Pier T, Facchinetti, Fabrizio, Carnini, Chiara, Moretto, Nadia, Patacchini, Riccardo, Bassani, Franco, Cenacchi, Valentina, Volta, Roberta, Amadei, Francesco, Capacchi, Silvia, Delcanale, Maurizio, Puccini, Paola, Catinella, Silvia, Civelli, Maurizio, Villetti, Gino
Published in Journal of medicinal chemistry (13.02.2014)
Published in Journal of medicinal chemistry (13.02.2014)
Get full text
Journal Article
Discovery of M-3 Antagonist-PDE4 Inhibitor Dual Pharmacology Molecules for the Treatment of Chronic Obstructive Pulmonary Disease
Armani, Elisabetta, Rizzi, Andrea, Capaldi, Carmelida, De Fanti, Renato, Delcanale, Maurizio, Villetti, Gino, Marchini, Gessica, Pisano, Anna Rita, Pitozzi, Vanessa, Pittelli, Maria Gloria, Trevisani, Marcello, Salvadori, Michela, Cenacchi, Valentina, Puccini, Paola, Amadei, Francesco, Pappani, Alice, Civelli, Maurizio, Patacchini, Riccardo, Baker-Glenn, Charles A. G., Van de Poel, Herve, Blackaby, Wesley P., Nash, Kevin, Amari, Gabriele
Published in Journal of medicinal chemistry (08.07.2021)
Published in Journal of medicinal chemistry (08.07.2021)
Get full text
Journal Article
CHF6001 I: a novel highly potent and selective phosphodiesterase 4 inhibitor with robust anti-inflammatory activity and suitable for topical pulmonary administration
Moretto, Nadia, Caruso, Paola, Bosco, Raffaella, Marchini, Gessica, Pastore, Fiorella, Armani, Elisabetta, Amari, Gabriele, Rizzi, Andrea, Ghidini, Eleonora, De Fanti, Renato, Capaldi, Carmelida, Carzaniga, Laura, Hirsch, Emilio, Buccellati, Carola, Sala, Angelo, Carnini, Chiara, Patacchini, Riccardo, Delcanale, Maurizio, Civelli, Maurizio, Villetti, Gino, Facchinetti, Fabrizio
Published in The Journal of pharmacology and experimental therapeutics (01.03.2015)
Published in The Journal of pharmacology and experimental therapeutics (01.03.2015)
Get full text
Journal Article
Discovery of M3 Antagonist-PDE4 Inhibitor Dual Pharmacology Molecules for the Treatment of Chronic Obstructive Pulmonary Disease
Armani, Elisabetta, Rizzi, Andrea, Capaldi, Carmelida, De Fanti, Renato, Delcanale, Maurizio, Villetti, Gino, Marchini, Gessica, Pisano, Anna Rita, Pitozzi, Vanessa, Pittelli, Maria Gloria, Trevisani, Marcello, Salvadori, Michela, Cenacchi, Valentina, Puccini, Paola, Amadei, Francesco, Pappani, Alice, Civelli, Maurizio, Patacchini, Riccardo, Baker-Glenn, Charles A.G, Van de Poël, Hervé, Blackaby, Wesley P, Nash, Kevin, Amari, Gabriele
Published in Journal of medicinal chemistry (08.07.2021)
Published in Journal of medicinal chemistry (08.07.2021)
Get full text
Journal Article
Discovery and Optimization of Thiazolidinyl and Pyrrolidinyl Derivatives as Inhaled PDE4 Inhibitors for Respiratory Diseases
Carzaniga, Laura, Amari, Gabriele, Rizzi, Andrea, Capaldi, Carmelida, De Fanti, Renato, Ghidini, Eleonora, Villetti, Gino, Carnini, Chiara, Moretto, Nadia, Facchinetti, Fabrizio, Caruso, Paola, Marchini, Gessica, Battipaglia, Loredana, Patacchini, Riccardo, Cenacchi, Valentina, Volta, Roberta, Amadei, Francesco, Pappani, Alice, Capacchi, Silvia, Bagnacani, Valentina, Delcanale, Maurizio, Puccini, Paola, Catinella, Silvia, Civelli, Maurizio, Armani, Elisabetta
Published in Journal of medicinal chemistry (28.12.2017)
Published in Journal of medicinal chemistry (28.12.2017)
Get full text
Journal Article
Synthesis and anticonvulsant activity of a class of 2-amino 3-hydroxypropanamide and 2-aminoacetamide derivatives
Ghidini, Eleonora, Delcanale, Maurizio, De Fanti, Renato, Rizzi, Andrea, Mazzuferi, Manuela, Rodi, Donata, Simonato, Michele, Lipreri, Milco, Bassani, Franco, Battipaglia, Loredana, Bergamaschi, Marco, Villetti, Gino
Published in Bioorganic & medicinal chemistry (15.05.2006)
Published in Bioorganic & medicinal chemistry (15.05.2006)
Get full text
Journal Article
Derivatives of 1-phenyl-2-pyridinyl alkyl alcohols as phosphodiesterase inhibitors
Carzaniga Laura, Armani Elisabetta, Capaldi Carmelida, Esposito Oriana, Amari Gabriele, De Fanti Renato, Villetti Gino
Year of Publication 03.04.2018
Get full text
Year of Publication 03.04.2018
Patent
Alfa-aminosyreamider, fremstilling og terapeutisk anvendelse derav
VENTURA PAOLO, DELCANALE MAURIZIO, PIETRA CLAUDIO, FANTI RENATO DE, ARMANI ELISABETTA, CHIESI PAOLO, VILETTI GINO
Year of Publication 07.06.2010
Get full text
Year of Publication 07.06.2010
Patent
Alfa-aminosyreamider, fremstilling og terapeutisk anvendelse derav
VENTURA PAOLO, DELCANALE MAURIZIO, PIETRA CLAUDIO, FANTI RENATO DE, ARMANI ELISABETTA, CHIESI PAOLO, VILETTI GINO
Year of Publication 23.02.2009
Get full text
Year of Publication 23.02.2009
Patent
composto, processo para o preparo de um composto, combinação de um composto, composição farmacêutica, uso de um composto, dispositivo e kit
CARMELIDA CAPALDI, ELISABETTA ARMANI, GINO VILLETTI, LAURA CARZANIGA, GABRIELE AMARI, RENATO DE FANTI, ORIANA ESPOSITO
Year of Publication 30.08.2016
Get full text
Year of Publication 30.08.2016
Patent
BENZHYDRYL DERIVATIVES FOR THE TREATMENT OF RESPIRATORY DISEASES
RICCABONI, Mauro, ARMANI, Elisabetta, BAKER-GLENN, Charles, AMARI, Gabriele, DE FANTI, Renato, CAPALDI, Carmelida, VAN DE PÖEL, Hervé
Year of Publication 06.09.2017
Get full text
Year of Publication 06.09.2017
Patent
DERIVATIVES OF 1-PHENYL-2-PYRIDINYL ALKYL ALCOHOLS AS PHOSPHODIESTERASE INHIBITORS
ESPOSITO ORIANA, DE FANTI RENATO, AMARI GABRIELE, CAPALDI CARMELIDA, VILLETTI GINO, CARZANIGA LAURA, ARMANI ELISABETTA
Year of Publication 14.01.2016
Get full text
Year of Publication 14.01.2016
Patent
BENZHYDRYL DERIVATIVES FOR THE TREATMENT OF RESPIRATORY DISEASES
ARMANI, ELISABETTA, DE FANTI, RENATO, RICCABONI, MAURO, BAKER-GLENN, CHARLES, AMARI, GABRIELE, CAPALDI, CARMELIDA, VAN DE PÖEL, HERVÉ
Year of Publication 12.10.2016
Get full text
Year of Publication 12.10.2016
Patent
Benzhydryl derivatives
VAN DE POËL HERVÉ, DE FANTI RENATO, AMARI GABRIELE, CAPALDI CARMELIDA, RICCABONI MAURO, BAKER-GLENN CHARLES, ARMANI ELISABETTA
Year of Publication 29.09.2015
Get full text
Year of Publication 29.09.2015
Patent
BENZHYDRYL DERIVATIVES
VAN DE POËL HERVÉ, DE FANTI RENATO, AMARI GABRIELE, CAPALDI CARMELIDA, RICCABONI MAURO, BAKER-GLENN CHARLES, ARMANI ELISABETTA
Year of Publication 11.06.2015
Get full text
Year of Publication 11.06.2015
Patent