Screening for AMPA receptor auxiliary subunit specific modulators
Azumaya, Caleigh M, Days, Emily L, Vinson, Paige N, Stauffer, Shaun, Sulikowski, Gary, Weaver, C David, Nakagawa, Terunaga
Published in PloS one (30.03.2017)
Published in PloS one (30.03.2017)
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Journal Article
Discovery and Characterization of VU0542270, the First Selective Inhibitor of Vascular Kir6.1/SUR2B K ATP Channels
Li, Kangjun, McClenahan, Samantha J, Han, Changho, Bungard, Joseph D, Rathnayake, Upendra, Boutaud, Olivier, Bauer, Joshua A, Days, Emily L, Lindsley, Craig W, Shelton, Elaine L, Denton, Jerod S
Published in Molecular pharmacology (01.03.2024)
Published in Molecular pharmacology (01.03.2024)
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Journal Article
Discovery and Characterization of VU0542270, the First Selective Inhibitor of Vascular Kir6.1/SUR2B KATP Channels
Li, Kangjun, McClenahan, Samantha J, Han, Changho, Bungard, Joseph D, Rathnayake, Upendra, Boutaud, Olivier, Bauer, Joshua A, Days, Emily L, Lindsley, Craig W, Shelton, Elaine L, Denton, Jerod S
Published in Molecular pharmacology (01.03.2024)
Published in Molecular pharmacology (01.03.2024)
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Journal Article
Synthesis and SAR of a novel Kir6.2/SUR1 channel opener scaffold identified by HTS
Dodd, Cayden J., Chronister, Keagan S., Rathnayake, Upendra, Parr, Lauren C., Li, Kangjun, Chang, Sichen, Mi, Dehui, Days, Emily L., Bauer, Joshua A., Cho, Hyekyung P., Boutaud, Olivier, Denton, Jerod S., Lindsley, Craig W., Han, Changho
Published in Bioorganic & medicinal chemistry letters (01.05.2023)
Published in Bioorganic & medicinal chemistry letters (01.05.2023)
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Journal Article
Discovery, Characterization, and Effects on Renal Fluid and Electrolyte Excretion of the Kir4.1 Potassium Channel Pore Blocker, VU0134992
Kharade, Sujay V, Kurata, Haruto, Bender, Aaron M, Blobaum, Anna L, Figueroa, Eric E, Duran, Amanda, Kramer, Meghan, Days, Emily, Vinson, Paige, Flores, Daniel, Satlin, Lisa M, Meiler, Jens, Weaver, C David, Lindsley, Craig W, Hopkins, Corey R, Denton, Jerod S
Published in Molecular pharmacology (01.08.2018)
Published in Molecular pharmacology (01.08.2018)
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Journal Article
VU6036720: The First Potent and Selective In Vitro Inhibitor of Heteromeric Kir4.1/5.1 Inward Rectifier Potassium Channels
McClenahan, Samantha J, Kent, Caitlin N, Kharade, Sujay V, Isaeva, Elena, Williams, Jade C, Han, Changho, Terker, Andrew, Gresham, 3rd, Robert, Lazarenko, Roman M, Days, Emily L, Romaine, Ian M, Bauer, Joshua A, Boutaud, Olivier, Sulikowski, Gary A, Harris, Raymond, Weaver, C David, Staruschenko, Alexander, Lindsley, Craig W, Denton, Jerod S
Published in Molecular pharmacology (01.05.2022)
Published in Molecular pharmacology (01.05.2022)
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Journal Article
Discovery of novel allosteric modulators of metabotropic glutamate receptor subtype 5 reveals chemical and functional diversity and in vivo activity in rat behavioral models of anxiolytic and antipsychotic activity
Rodriguez, Alice L, Grier, Mark D, Jones, Carrie K, Herman, Elizabeth J, Kane, Alexander S, Smith, Randy L, Williams, Richard, Zhou, Ya, Marlo, Joy E, Days, Emily L, Blatt, Tasha N, Jadhav, Satyawan, Menon, Usha N, Vinson, Paige N, Rook, Jerri M, Stauffer, Shaun R, Niswender, Colleen M, Lindsley, Craig W, Weaver, C David, Conn, P Jeffrey
Published in Molecular pharmacology (01.12.2010)
Published in Molecular pharmacology (01.12.2010)
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Journal Article
Discovery, Characterization, and Antiparkinsonian Effect of Novel Positive Allosteric Modulators of Metabotropic Glutamate Receptor 4
Niswender, Colleen M, Johnson, Kari A, Weaver, C David, Jones, Carrie K, Xiang, Zixiu, Luo, Qingwei, Rodriguez, Alice L, Marlo, Joy E, de Paulis, Tomas, Thompson, Analisa D, Days, Emily L, Nalywajko, Tasha, Austin, Cheryl A, Williams, Michael Baxter, Ayala, Jennifer E, Williams, Richard, Lindsley, Craig W, Conn, P Jeffrey
Published in Molecular pharmacology (01.11.2008)
Published in Molecular pharmacology (01.11.2008)
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Journal Article
Small-molecule screen identifies inhibitors of the neuronal K-Cl cotransporter KCC2
Delpire, Eric, Days, Emily, Lewis, L. Michelle, Mi, Dehui, Kim, Kwangho, Lindsley, Craig W, Weaver, C. David
Published in Proceedings of the National Academy of Sciences - PNAS (31.03.2009)
Published in Proceedings of the National Academy of Sciences - PNAS (31.03.2009)
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Journal Article
ML297 (VU0456810), the First Potent and Selective Activator of the GIRK Potassium Channel, Displays Antiepileptic Properties in Mice
Kaufmann, Kristian, Romaine, Ian, Days, Emily, Pascual, Conrado, Malik, Adam, Yang, Liya, Zou, Bende, Du, Yu, Sliwoski, Greg, Morrison, Ryan D, Denton, Jerod, Niswender, Colleen M, Daniels, J. Scott, Sulikowski, Gary A, Xie, Xinmin (Simon), Lindsley, Craig W, Weaver, C. David
Published in ACS chemical neuroscience (18.09.2013)
Published in ACS chemical neuroscience (18.09.2013)
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Discovery of (S)‑2-Cyclopentyl‑N‑((1-isopropylpyrrolidin2-yl)-9-methyl-1-oxo-2,9-dihydro‑1H‑pyrrido[3,4‑b]indole-4-carboxamide (VU0453379): A Novel, CNS Penetrant Glucagon-Like Peptide 1 Receptor (GLP-1R) Positive Allosteric Modulator (PAM)
Morris, Lindsey C, Nance, Kellie D, Gentry, Patrick R, Days, Emily L, Weaver, C. David, Niswender, Colleen M, Thompson, Analisa D, Jones, Carrie K, Locuson, Chuck W, Morrison, Ryan D, Daniels, J. Scott, Niswender, Kevin D, Lindsley, Craig W
Published in Journal of medicinal chemistry (11.12.2014)
Published in Journal of medicinal chemistry (11.12.2014)
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Discovery of a Novel Series of Orally Bioavailable and CNS Penetrant Glucagon-like Peptide-1 Receptor (GLP-1R) Noncompetitive Antagonists Based on a 1,3-Disubstituted-7-aryl-5,5-bis(trifluoromethyl)-5,8-dihydropyrimido[4,5-d]pyrimidine-2,4(1H,3H)-dione Core
Nance, Kellie D, Days, Emily L, Weaver, C David, Coldren, Anastasia, Farmer, Tiffany D, Cho, Hyekyung P, Niswender, Colleen M, Blobaum, Anna L, Niswender, Kevin D, Lindsley, Craig W
Published in Journal of medicinal chemistry (23.02.2017)
Published in Journal of medicinal chemistry (23.02.2017)
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Journal Article
Selective Small Molecule Activators of TREK‑2 Channels Stimulate Dorsal Root Ganglion c‑Fiber Nociceptor Two-Pore-Domain Potassium Channel Currents and Limit Calcium Influx
Dadi, Prasanna K, Vierra, Nicholas C, Days, Emily, Dickerson, Matthew T, Vinson, Paige N, Weaver, C. David, Jacobson, David A
Published in ACS chemical neuroscience (15.03.2017)
Published in ACS chemical neuroscience (15.03.2017)
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Journal Article
Discovery and characterization of a potent and selective inhibitor of Aedes aegypti inward rectifier potassium channels
Raphemot, Rene, Rouhier, Matthew F, Swale, Daniel R, Days, Emily, Weaver, C David, Lovell, Kimberly M, Konkel, Leah C, Engers, Darren W, Bollinger, Sean R, Bollinger, Sean F, Hopkins, Corey, Piermarini, Peter M, Denton, Jerod S
Published in PloS one (06.11.2014)
Published in PloS one (06.11.2014)
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Journal Article
Identification of Positive Allosteric Modulators VU0155094 (ML397) and VU0422288 (ML396) Reveals New Insights into the Biology of Metabotropic Glutamate Receptor 7
Jalan-Sakrikar, Nidhi, Field, Julie R, Klar, Rebecca, Mattmann, Margrith E, Gregory, Karen J, Zamorano, Rocio, Engers, Darren W, Bollinger, Sean R, Weaver, C. David, Days, Emily L, Lewis, L. Michelle, Utley, Thomas J, Hurtado, Miguel, Rigault, Delphine, Acher, Francine, Walker, Adam G, Melancon, Bruce J, Wood, Michael R, Lindsley, Craig W, Conn, P. Jeffrey, Xiang, Zixiu, Hopkins, Corey R, Niswender, Colleen M
Published in ACS chemical neuroscience (17.12.2014)
Published in ACS chemical neuroscience (17.12.2014)
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Journal Article
A Duplexed High-Throughput Screen to Identify Allosteric Modulators of the Glucagon-Like Peptide 1 and Glucagon Receptors
Morris, Lindsey C, Days, Emily L, Turney, Maxine, Mi, Dehui, Lindsley, Craig W, Weaver, C David, Niswender, Kevin D
Published in Journal of biomolecular screening (01.07.2014)
Published in Journal of biomolecular screening (01.07.2014)
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Journal Article
Discovery of N-Aryl Piperazines as Selective mGluR5 Potentiators with Improved In Vivo Utility
Zhou, Ya, Manka, Jason T, Rodriguez, Alice L, Weaver, C. David, Days, Emily L, Vinson, Paige N, Jadhav, Satyawan, Hermann, Elizabeth J, Jones, Carrie K, Conn, P. Jeffrey, Lindsley, Craig W, Stauffer, Shaun R
Published in ACS medicinal chemistry letters (11.11.2010)
Published in ACS medicinal chemistry letters (11.11.2010)
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Journal Article
Discovery and Characterization of Novel Allosteric Potentiators of M1 Muscarinic Receptors Reveals Multiple Modes of Activity
Marlo, Joy E, Niswender, Colleen M, Days, Emily L, Bridges, Thomas M, Xiang, Yun, Rodriguez, Alice L, Shirey, Jana K, Brady, Ashley E, Nalywajko, Tasha, Luo, Qingwei, Austin, Cheryl A, Williams, Michael Baxter, Kim, Kwangho, Williams, Richard, Orton, Darren, Brown, H Alex, Lindsley, Craig W, Weaver, C David, Conn, P Jeffrey
Published in Molecular pharmacology (01.03.2009)
Published in Molecular pharmacology (01.03.2009)
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Journal Article
225-LB: Targeting ß-Cell Endoplasmic Reticulum (ER) TALK-1 Channels to Restore Ca2+ Homeostasis and Reduce ER Stress in Diabetes
NAKHE, ARYA Y., DADI, PRASANNA, WESTOVER, DAVID, DAYS, EMILY, DENTON, JEROD, JACOBSON, DAVID
Published in Diabetes (New York, N.Y.) (01.06.2021)
Published in Diabetes (New York, N.Y.) (01.06.2021)
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