Structural insight into selectivity and resistance profiles of ROS1 tyrosine kinase inhibitors
Davare, Monika A., Vellore, Nadeem A., Wagner, Jacob P., Eide, Christopher A., Goodman, James R., Drilon, Alexander, Deininger, Michael W., O’Hare, Thomas, Druker, Brian J.
Published in Proceedings of the National Academy of Sciences - PNAS (29.09.2015)
Published in Proceedings of the National Academy of Sciences - PNAS (29.09.2015)
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Journal Article
A Novel Crizotinib-Resistant Solvent-Front Mutation Responsive to Cabozantinib Therapy in a Patient with ROS1-Rearranged Lung Cancer
Drilon, Alexander, Somwar, Romel, Wagner, Jacob P, Vellore, Nadeem A, Eide, Christopher A, Zabriskie, Matthew S, Arcila, Maria E, Hechtman, Jaclyn F, Wang, Lu, Smith, Roger S, Kris, Mark G, Riely, Gregory J, Druker, Brian J, O'Hare, Thomas, Ladanyi, Marc, Davare, Monika A
Published in Clinical cancer research (15.05.2016)
Published in Clinical cancer research (15.05.2016)
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Journal Article
Foretinib is a potent inhibitor of oncogenic ROS1 fusion proteins
Davare, Monika A., Saborowski, Anna, Eide, Christopher A., Tognon, Cristina, Smith, Rebecca L., Elferich, Johannes, Agarwal, Anupriya, Tyner, Jeffrey W., Shinde, Ujwal P., Lowe, Scott W., Druker, Brian J.
Published in Proceedings of the National Academy of Sciences - PNAS (26.11.2013)
Published in Proceedings of the National Academy of Sciences - PNAS (26.11.2013)
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Journal Article
Inhibition of interleukin-1 receptor-associated kinase-1 is a therapeutic strategy for acute myeloid leukemia subtypes
Hosseini, Mona M, Kurtz, Stephen E, Abdelhamed, Sherif, Mahmood, Shawn, Davare, Monika A, Kaempf, Andy, Elferich, Johannes, McDermott, Jason E, Liu, Tao, Payne, Samuel H, Shinde, Ujwal, Rodland, Karin D, Mori, Motomi, Druker, Brian J, Singer, Jack W, Agarwal, Anupriya
Published in Leukemia (01.11.2018)
Published in Leukemia (01.11.2018)
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Journal Article
Long-term potentiation-dependent spine enlargement requires synaptic Ca2+-permeable AMPA receptors recruited by CaM-kinase I
Fortin, Dale A, Davare, Monika A, Srivastava, Taasin, Brady, James D, Nygaard, Sean, Derkach, Victor A, Soderling, Thomas R
Published in The Journal of neuroscience (01.09.2010)
Published in The Journal of neuroscience (01.09.2010)
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Journal Article
Discovery and Characterization of Recurrent, Targetable ALK Fusions in Leiomyosarcoma
Davis, Lara E, Nusser, Kevin D, Przybyl, Joanna, Pittsenbarger, Janét, Hofmann, Nicolle E, Varma, Sushama, Vennam, Sujay, Debiec-Rychter, Maria, van de Rijn, Matt, Davare, Monika A
Published in Molecular cancer research (01.03.2019)
Published in Molecular cancer research (01.03.2019)
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Journal Article
Discovery of oncogenic ROS1 missense mutations with sensitivity to tyrosine kinase inhibitors
Iyer, Sudarshan R, Nusser, Kevin, Jones, Kristen, Shinde, Pushkar, Keddy, Clare, Beach, Catherine Z, Aguero, Erin, Force, Jeremy, Shinde, Ujwal, Davare, Monika A
Published in EMBO molecular medicine (11.10.2023)
Published in EMBO molecular medicine (11.10.2023)
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Journal Article
Mouse model of intrahepatic cholangiocarcinoma validates FIG–ROS as a potent fusion oncogene and therapeutic target
Saborowski, Anna, Saborowski, Michael, Davare, Monika A., Druker, Brian J., Klimstra, David S., Lowe, Scott W.
Published in Proceedings of the National Academy of Sciences - PNAS (26.11.2013)
Published in Proceedings of the National Academy of Sciences - PNAS (26.11.2013)
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Journal Article
NTRK kinase domain mutations in cancer variably impact sensitivity to type I and type II inhibitors
Somwar, Romel, Hofmann, Nicolle E, Smith, Bryan, Odintsov, Igor, Vojnic, Morana, Linkov, Irina, Tam, Ashley, Khodos, Inna, Mattar, Marissa S, de Stanchina, Elisa, Flynn, Daniel, Ladanyi, Marc, Drilon, Alexander, Shinde, Ujwal, Davare, Monika A
Published in Communications biology (16.12.2020)
Published in Communications biology (16.12.2020)
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Journal Article
RET inhibition in novel patient-derived models of RET-fusion positive lung adenocarcinoma reveals a role for MYC upregulation
Hayashi, Takuo, Odintsov, Igor, Smith, Roger S, Ishizawa, Kota, Liu, Allan J W, Delasos, Lukas, Kurzatkowski, Christopher, Tai, Huichun, Gladstone, Eric, Vojnic, Morana, Kohsaka, Shinji, Suzawa, Ken, Liu, Zebing, Kunte, Siddharth, Mattar, Marissa S, Khodos, Inna, Davare, Monika A, Drilon, Alexander, Cheng, Emily, Stanchina, Elisa de, Ladanyi, Marc, Somwar, Romel
Published in Disease models & mechanisms (01.02.2021)
Published in Disease models & mechanisms (01.02.2021)
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Journal Article
TKI type switching overcomes ROS1 L2086F in ROS1 fusion-positive cancers
Thawani, Rajat, Repetto, Matteo, Keddy, Clare, Nicholson, Katelyn, Jones, Kristen, Nusser, Kevin, Beach, Catherine Z, Harada, Guilherme, Drilon, Alexander, Davare, Monika A
Published in NPJ precision oncology (08.08.2024)
Published in NPJ precision oncology (08.08.2024)
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Journal Article
Author Correction: TKI type switching overcomes ROS1 L2086F in ROS1 fusion-positive cancers
Thawani, Rajat, Repetto, Matteo, Keddy, Clare, Nicholson, Katelyn, Jones, Kristen, Nusser, Kevin, Beach, Catherine Z, Harada, Guilherme, Drilon, Alexander, Davare, Monika A
Published in NPJ precision oncology (28.08.2024)
Published in NPJ precision oncology (28.08.2024)
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Journal Article
Discovery and Validation of a Compound to Target Ewing's Sarcoma
Esfandiari Nazzaro, Ellie, Sabei, Fahad Y, Vogel, Walter K, Nazari, Mohamad, Nicholson, Katelyn S, Gafken, Philip R, Taratula, Olena, Taratula, Oleh, Davare, Monika A, Leid, Mark
Published in Pharmaceutics (24.09.2021)
Published in Pharmaceutics (24.09.2021)
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Journal Article
Critical Role of cAMP-Dependent Protein Kinase Anchoring to the L-Type Calcium Channel Cav1.2 via A-Kinase Anchor Protein 150 in Neurons
Hall, Duane D, Davare, Monika A, Shi, Mei, Allen, Margaret L, Weisenhaus, Michael, McKnight, G. Stanley, Hell, Johannes W
Published in Biochemistry (Easton) (13.02.2007)
Published in Biochemistry (Easton) (13.02.2007)
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Journal Article
Therapeutically Targetable ALK Mutations in Leukemia
Maxson, Julia E, Davare, Monika A, Luty, Samuel B, Eide, Christopher A, Chang, Bill H, Loriaux, Marc M, Tognon, Cristina E, Bottomly, Daniel, Wilmot, Beth, McWeeney, Shannon K, Druker, Brian J, Tyner, Jeffrey W
Published in Cancer research (Chicago, Ill.) (01.06.2015)
Published in Cancer research (Chicago, Ill.) (01.06.2015)
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Journal Article
Functional impact and targetability of PI3KCA , GNAS , and PTEN mutations in a spindle cell rhabdomyosarcoma with MYOD1 L122R mutation
Choo, Florence, Odintsov, Igor, Nusser, Kevin, Nicholson, Katelyn S, Davis, Lara, Corless, Christopher L, Stork, Linda, Somwar, Romel, Ladanyi, Marc, Davis, Jessica L, Davare, Monika A
Published in Cold Spring Harbor molecular case studies (01.01.2022)
Published in Cold Spring Harbor molecular case studies (01.01.2022)
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Journal Article
ROS1-dependent cancers - biology, diagnostics and therapeutics
Drilon, Alexander, Jenkins, Chelsea, Iyer, Sudarshan, Schoenfeld, Adam, Keddy, Clare, Davare, Monika A
Published in Nature reviews. Clinical oncology (01.01.2021)
Published in Nature reviews. Clinical oncology (01.01.2021)
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Journal Article
ERK activation and cell growth require CaM kinases in MCF-7 breast cancer cells
Schmitt, John M, Abell, Ellen, Wagner, Andrea, Davare, Monika A
Published in Molecular and cellular biochemistry (01.02.2010)
Published in Molecular and cellular biochemistry (01.02.2010)
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