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Published in Science (American Association for the Advancement of Science) (21.08.2020)
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Targeting Xist with compounds that disrupt RNA structure and X inactivation
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Nanoscale synthesis and affinity ranking
Gesmundo, Nathan J., Sauvagnat, Bérengère, Curran, Patrick J., Richards, Matthew P., Andrews, Christine L., Dandliker, Peter J., Cernak, Tim
Published in Nature (London) (01.05.2018)
Published in Nature (London) (01.05.2018)
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Exploring new targets and chemical space with affinity selection-mass spectrometry
Prudent, Renaud, Annis, D. Allen, Dandliker, Peter J., Ortholand, Jean-Yves, Roche, Didier
Published in Nature reviews. Chemistry (01.01.2021)
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Discovery of Selective RNA-Binding Small Molecules by Affinity-Selection Mass Spectrometry
Rizvi, Noreen F, Howe, John A, Nahvi, Ali, Klein, Daniel J, Fischmann, Thierry O, Kim, Hai-Young, McCoy, Mark A, Walker, Scott S, Hruza, Alan, Richards, Matthew P, Chamberlin, Chad, Saradjian, Peter, Butko, Margaret T, Mercado, Gabriel, Burchard, Julja, Strickland, Corey, Dandliker, Peter J, Smith, Graham F, Nickbarg, Elliott B
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Published in ACS chemical biology (16.03.2018)
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Macrocyclic α helical peptide therapeutic modality: A perspective of learnings and challenges
Sawyer, Tomi K., Partridge, Anthony W., Kaan, Hung Yi Kristal, Juang, Yu-Chi, Lim, Shuhui, Johannes, Charles, Yuen, Tsz Ying, Verma, Chandra, Kannan, Srinivasaraghavan, Aronica, Pietro, Tan, Yaw Sing, Sherborne, Brad, Ha, Sookhee, Hochman, Jerome, Chen, Shiying, Surdi, Laura, Peier, Andrea, Sauvagnat, Berengere, Dandliker, Peter J., Brown, Christopher J., Ng, Simon, Ferrer, Fernando, Lane, David P.
Published in Bioorganic & medicinal chemistry (01.06.2018)
Published in Bioorganic & medicinal chemistry (01.06.2018)
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Evaluation of JAK3 Biology in Autoimmune Disease Using a Highly Selective, Irreversible JAK3 Inhibitor
Elwood, Fiona, Witter, David J, Piesvaux, Jennifer, Kraybill, Brian, Bays, Nathan, Alpert, Carla, Goldenblatt, Peter, Qu, Yujie, Ivanovska, Irena, Lee, Hyun-Hee, Chiu, Chi-Sung, Tang, Hao, Scott, Mark E, Deshmukh, Sujal V, Zielstorff, Mark, Byford, Alan, Chakravarthy, Kalyan, Dorosh, Lauren, Rivkin, Alexey, Klappenbach, Joel, Pan, Bo-Sheng, Kariv, Ilona, Dinsmore, Christopher, Slipetz, Deborah, Dandliker, Peter J
Published in The Journal of pharmacology and experimental therapeutics (01.05.2017)
Published in The Journal of pharmacology and experimental therapeutics (01.05.2017)
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Targeting RNA with Small Molecules: Identification of Selective, RNA-Binding Small Molecules Occupying Drug-Like Chemical Space
Rizvi, Noreen F., Santa Maria, John P., Nahvi, Ali, Klappenbach, Joel, Klein, Daniel J., Curran, Patrick J., Richards, Matthew P., Chamberlin, Chad, Saradjian, Peter, Burchard, Julja, Aguilar, Rodrigo, Lee, Jeannie T., Dandliker, Peter J., Smith, Graham F., Kutchukian, Peter, Nickbarg, Elliott B.
Published in SLAS discovery (01.04.2020)
Published in SLAS discovery (01.04.2020)
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Definitive Metabolite Identification Coupled with Automated Ligand Identification System (ALIS) Technology: A Novel Approach to Uncover Structure–Activity Relationships and Guide Drug Design in a Factor IXa Inhibitor Program
Zhang, Ting, Liu, Yong, Yang, Xianshu, Martin, Gary E, Yao, Huifang, Shang, Jackie, Bugianesi, Randal M, Ellsworth, Kenneth P, Sonatore, Lisa M, Nizner, Peter, Sherer, Edward C, Hill, Susan E, Knemeyer, Ian W, Geissler, Wayne M, Dandliker, Peter J, Helmy, Roy, Wood, Harold B
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Published in Journal of medicinal chemistry (10.03.2016)
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Integration of Affinity Selection-Mass Spectrometry and Functional Cell-Based Assays to Rapidly Triage Druggable Target Space within the NF-κB Pathway
Kutilek, Victoria D, Andrews, Christine L, Richards, Matthew P, Xu, Zangwei, Sun, Tianxiao, Chen, Yiping, Hashke, Andrew, Smotrov, Nadya, Fernandez, Rafael, Nickbarg, Elliott B, Chamberlin, Chad, Sauvagnat, Berengere, Curran, Patrick J, Boinay, Ryan, Saradjian, Peter, Allen, Samantha J, Byrne, Noel, Elsen, Nathaniel L, Ford, Rachael E, Hall, Dawn L, Kornienko, Maria, Rickert, Keith W, Sharma, Sujata, Shipman, Jennifer M, Lumb, Kevin J, Coleman, Kevin, Dandliker, Peter J, Kariv, Ilona, Beutel, Bruce
Published in Journal of biomolecular screening (01.07.2016)
Published in Journal of biomolecular screening (01.07.2016)
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Oxidative Thymine Dimer Repair in the DNA Helix
Dandliker, Peter J., Holmlin, R. Erik, Barton, Jacqueline K.
Published in Science (American Association for the Advancement of Science) (07.03.1997)
Published in Science (American Association for the Advancement of Science) (07.03.1997)
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SOS-NMR: A Saturation Transfer NMR-Based Method for Determining the Structures of Protein−Ligand Complexes
Hajduk, Philip J, Mack, Jamey C, Olejniczak, Edward T, Park, Chang, Dandliker, Peter J, Beutel, Bruce A
Published in Journal of the American Chemical Society (03.03.2004)
Published in Journal of the American Chemical Society (03.03.2004)
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Pharmacokinetic Enhancement of the Hepatitis C Virus Protease Inhibitors VX-950 and SCH 503034 by Co-Dosing with Ritonavir
Kempf, Dale J, Klein, Cheri, Chen, Hui-Ju, Klein, Larry L, Yeung, Clinton, Randolph, John T, Lau, Yau Y, Chovan, Linda E, Guan, Zhiwen, Hernandez, Lisa, Turner, Teresa M, Dandliker, Peter J, Marsh, Kennan C
Published in Antiviral chemistry & chemotherapy (01.06.2007)
Published in Antiviral chemistry & chemotherapy (01.06.2007)
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Thienopyridine urea inhibitors of KDR kinase
Heyman, H. Robin, Frey, Robin R., Bousquet, Peter F., Cunha, George A., Moskey, Maria D., Ahmed, Asma A., Soni, Niru B., Marcotte, Patrick A., Pease, Lori J., Glaser, Keith B., Yates, Melinda, Bouska, Jennifer J., Albert, Daniel H., Black-Schaefer, Candace L., Dandliker, Peter J., Stewart, Kent D., Rafferty, Paul, Davidsen, Steven K., Michaelides, Michael R., Curtin, Michael L.
Published in Bioorganic & medicinal chemistry letters (01.03.2007)
Published in Bioorganic & medicinal chemistry letters (01.03.2007)
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Rapid hit to lead evaluation of pyrazolo[3,4- d]pyrimidin-4-one as selective and orally bioavailable mGluR1 antagonists
Wang, Xueqing, Kolasa, Teodozyi, El Kouhen, Odile F., Chovan, Linda E., Black-Shaefer, Candace L., Wagenaar, Frank L., Garton, Jennifer A., Moreland, Robert B., Honore, Prisca, Lau, Yau Yi, Dandliker, Peter J., Brioni, Jorge D., Stewart, Andrew O.
Published in Bioorganic & medicinal chemistry letters (01.08.2007)
Published in Bioorganic & medicinal chemistry letters (01.08.2007)
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Synthesis of Metallointercalator−DNA Conjugates on a Solid Support
Holmlin, R. Erik, Dandliker, Peter J, Barton, Jacqueline K
Published in Bioconjugate chemistry (01.11.1999)
Published in Bioconjugate chemistry (01.11.1999)
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Novel Antibacterial Class
DANDLIKER, Peter J, PRATT, Steve D, CHOVAN, Linda E, HICKMAN, Robert K, DALY, Melissa M, KAKAVAS, Stephan, PING ZHONG, ZHENSHENG CAO, DAVID, Caroline A, XIAOLING XUEI, LERNER, Claude G, SONI, Niru B, NILIUS, Angela M, MAI BUI, SHEN, Linus L, YINGNA CAI, MERTA, Philip J, SAIKI, Anne Y. C, BEUTEL, Bruce A, BLACK-SCHAEFER, Candace, XIAOAN RUAN, TOWNE, Danli L, CLARK, Richard F, ENGLUND, Erika E, WAGNER, Rolf, WEITZBERG, Moshe
Published in Antimicrobial Agents and Chemotherapy (01.12.2003)
Published in Antimicrobial Agents and Chemotherapy (01.12.2003)
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