Characterization of rofecoxib as a cyclooxygenase-2 isoform inhibitor and demonstration of analgesia in the dental pain model
Ehrich, E W, Dallob, A, De Lepeleire, I, Van Hecken, A, Riendeau, D, Yuan, W, Porras, A, Wittreich, J, Seibold, J R, De Schepper, P, Mehlisch, D R, Gertz, B J
Published in Clinical pharmacology and therapeutics (01.03.1999)
Published in Clinical pharmacology and therapeutics (01.03.1999)
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Comparative inhibitory activity of rofecoxib, meloxicam, diclofenac, ibuprofen, and naproxen on COX-2 versus COX-1 in healthy volunteers
Van Hecken, A, Schwartz, J I, Depré, M, De Lepeleire, I, Dallob, A, Tanaka, W, Wynants, K, Buntinx, A, Arnout, J, Wong, P H, Ebel, D L, Gertz, B J, De Schepper, P J
Published in Journal of clinical pharmacology (01.10.2000)
Published in Journal of clinical pharmacology (01.10.2000)
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A human whole blood assay for clinical evaluation of biochemical efficacy of cyclooxygenase inhibitors
Brideau, C, Kargman, S, Liu, S, Dallob, A L, Ehrich, E W, Rodger, I W, Chan, C C
Published in Inflammation research (01.02.1996)
Published in Inflammation research (01.02.1996)
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The effects of finasteride on scalp skin and serum androgen levels in men with androgenetic alopecia
Drake, Lynn, Hordinsky, Maria, Fiedler, Virginia, Swinehart, James, Unger, Walter P., Cotterill, Paul C., Thiboutot, Diane M., Lowe, Nicholas, Jacobson, Coleman, Whiting, David, Stieglitz, Sam, Kraus, Stephen J., Griffin, Edmond I., Weiss, Darryl, Carrington, Patrick, Gencheff, Christopher, Cole, Gary W., Pariser, David M., Epstein, Edwin S., Tanaka, Wesley, Dallob, Aimée, Vandormael, Kristel, Geissler, Lori, Waldsteicher, Joanne
Published in Journal of the American Academy of Dermatology (01.10.1999)
Published in Journal of the American Academy of Dermatology (01.10.1999)
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The effect of finasteride, a 5 alpha-reductase inhibitor, on scalp skin testosterone and dihydrotestosterone concentrations in patients with male pattern baldness
Dallob, A L, Sadick, N S, Unger, W, Lipert, S, Geissler, L A, Gregoire, S L, Nguyen, H H, Moore, E C, Tanaka, W K
Published in The journal of clinical endocrinology and metabolism (01.09.1994)
Published in The journal of clinical endocrinology and metabolism (01.09.1994)
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Pharmacokinetics, COX-2 specificity, and tolerability of supratherapeutic doses of rofecoxib in humans
DEPRE, M, EHRICH, E, VAN HECKEN, A, DE LEPELEIRE, I, DALLOB, A, WONG, P, PORRAS, A, GERTZ, B. J, DE SCHEPPER, P. J
Published in European journal of clinical pharmacology (01.05.2000)
Published in European journal of clinical pharmacology (01.05.2000)
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Ex vivo assays demonstrate potency and selectivity of the COX-2 inhibitor DFP after single dose administration
Dallob, A, De Lepeleire, I, Van Hecken, A, Porras, A, Depré, M, Mukhopadhyay, S, Flynn, M, Wildonger, L, Gottesdiener, K, Tanaka, W, De Schepper, P
Published in Inflammation research (01.12.1999)
Published in Inflammation research (01.12.1999)
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Measurement of Plasma Angiotensin II: Purification by Cation-Exchange Chromatography
Ledwith, B.J., Cahill, M.K., Losse, L.S., Satiritz, S.M., Eydelloth, R.S., Dallob, A.L., Tanaka, W.K., Galloway, S.M., Nichols, W.W.
Published in Analytical biochemistry (01.09.1993)
Published in Analytical biochemistry (01.09.1993)
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Synthesis and structure-activity relationships of a novel class of 5-lipoxygenase inhibitors. 2-(Phenylmethyl)-4-hydroxy-3,5-dialkylbenzofurans: the development of L-656,224
Lau, Cheuk K, Belanger, Patrice C, Scheigetz, John, Dufresne, Claude, Williams, Haydn W. R, Maycock, Alan L, Guindon, Yvan, Bach, Thomas, Dallob, Aimee L
Published in Journal of medicinal chemistry (01.06.1989)
Published in Journal of medicinal chemistry (01.06.1989)
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Phase I pharmacokinetic (PK), and pharmacodynamic (PD) trial of the novel oral Notch inhibitor MK-0752 in patients (pts) with advanced breast cancer (BC) and other solid tumors
Krop, I. E., Kosh, M., Fearen, I., Savoie, J., Dallob, A., Matthews, C., Stone, J., Winer, E., Freedman, S. J., Lorusso, P.
Published in Journal of clinical oncology (20.06.2006)
Published in Journal of clinical oncology (20.06.2006)
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A phase I clinical trial of the notch inhibitor MK-0752 in patients with T-cell acute lymphoblastic leukemia/lymphoma (T-ALL) and other leukemias
Deangelo, D. J., Stone, R. M., Silverman, L. B., Stock, W., Attar, E. C., Fearen, I., Dallob, A., Matthews, C., Stone, J., Freedman, S. J., Aster, J.
Published in Journal of clinical oncology (20.06.2006)
Published in Journal of clinical oncology (20.06.2006)
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L-651,392: a novel, potent and selective 5-lipoxygenase inhibitor
Guindon, Y, Girard, Y, Maycock, A, Ford-Hutchinson, A W, Atkinson, J G, Bélanger, P C, Dallob, A, DeSousa, D, Dougherty, H, Egan, R
Published in Advances in prostaglandin, thromboxane, and leukotriene research (1987)
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Published in Advances in prostaglandin, thromboxane, and leukotriene research (1987)
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Rofecoxib, a COX-2 inhibitor, does not inhibit human gastric mucosal prostaglandin production
Wight, N J, Gottesdiener, K, Garlick, N M, Atherton, C T, Novak, S, Gertz, B J, Calder, N A, Cote, J, Wong, P, Dallob, A, Hawkey, C J
Published in Gastroenterology (New York, N.Y. 1943) (01.03.2001)
Published in Gastroenterology (New York, N.Y. 1943) (01.03.2001)
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L-652,343: a novel dual 5-lipoxygenase/cyclooxygenase inhibitor
Tischler, A, Bailey, P, Dallob, A, Witzel, B, Durette, P, Rupprecht, K, Allison, D, Dougherty, H, Humes, J, Ham, E
Published in Advances in prostaglandin, thromboxane, and leukotriene research (1986)
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Published in Advances in prostaglandin, thromboxane, and leukotriene research (1986)
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MK-386, an inhibitor of 5α-reductase type 1, reduces dihydrotestosterone concentrations in serum and sebum without affecting dihydrotestosterone concentrations in semen
SCHWARTZ, J. I, TANAKA, W. K, WANG, D. Z, EBEL, D. L, GEISSLER, L. A, DALLOB, A, HAFKIN, B, GERTZ, B. J
Published in The journal of clinical endocrinology and metabolism (1997)
Published in The journal of clinical endocrinology and metabolism (1997)
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MK-386, an inhibitor of 5alpha-reductase type 1, reduces dihydrotestosterone concentrations in serum and sebum without affecting dihydrotestosterone concentrations in semen
Schwartz, J I, Tanaka, W K, Wang, D Z, Ebel, D L, Geissler, L A, Dallob, A, Hafkin, B, Gertz, B J
Published in The journal of clinical endocrinology and metabolism (01.05.1997)
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Published in The journal of clinical endocrinology and metabolism (01.05.1997)
Journal Article
The effects of finasteride on scalp skin and serum androgen levels in men with androgenetic alopecia
DRAKE, L, HORDINSKY, M, STIEGLITZ, S, KRAUS, S. J, GRIFFIN, E. I, WEISS, D, CARRINGTON, P, GENCHEFF, C, COLE, G. W, PARISER, P. D. M, EPSTEIN, E. S, TANAKA, W, FIEDLER, V, DALLOB, A, VANDORMAEL, K, GEISSLER, L, WALDSTREICHER, J, SWINEHART, J, UNGER, W. P, COTTERILL, P. C, THIBOUTOT, D. M, LOWE, N, JACOBSON, C, WHITING, D
Published in Journal of the American Academy of Dermatology (01.10.1999)
Published in Journal of the American Academy of Dermatology (01.10.1999)
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Journal Article
Pharmacokinetics and pharmacodynamics of multiple oral doses of MK-0591, a 5-lipoxygenase-activating protein inhibitor
Depré, M, Friedman, B, Van Hecken, A, de Lepeleire, I, Tanaka, W, Dallob, A, Shingo, S, Porras, A, Lin, C, de Schepper, P J
Published in Clinical pharmacology and therapeutics (01.07.1994)
Published in Clinical pharmacology and therapeutics (01.07.1994)
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Pharmacology of the dual inhibitor of cyclooxygenase and 5-lipoxygenase 3-hydroxy-5-trifluoromethyl-N-(2-(2-thienyl)-2-phenyl-ethenyl)-benzo (b)thiophene-2-carboxamide
Bailey, P J, Dallob, A L, Allison, D L, Anderson, R L, Bach, T, Durette, P L, Hand, K M, Hopple, S L, Luell, S, Meurer, R
Published in Arzneimittel-Forschung (01.03.1988)
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Published in Arzneimittel-Forschung (01.03.1988)
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