Total synthesis of amphotericin B. 3. The final stages
Nicolaou, Kyriacos C, Daines, R. A, Ogawa, Y, Chakraborty, T. K
Published in Journal of the American Chemical Society (01.07.1988)
Published in Journal of the American Chemical Society (01.07.1988)
Get full text
Journal Article
Total synthesis of amphoteronolide B and amphotericin B. 1. Strategy and stereocontrolled construction of key building blocks
Nicolaou, Kyriacos C, Daines, R. A, Uenishi, J, Li, W. S, Papahatjis, D. P, Chakraborty, T. K
Published in Journal of the American Chemical Society (01.07.1988)
Published in Journal of the American Chemical Society (01.07.1988)
Get full text
Journal Article
Chemistry of amphotericin B. Degradation studies and preparation of amphoteronolide B
Nicolaou, K. C, Chakraborty, T. K, Ogawa, Y, Daines, R. A, Simpkins, N. S, Furst, G. T
Published in Journal of the American Chemical Society (01.07.1988)
Published in Journal of the American Chemical Society (01.07.1988)
Get full text
Journal Article
In vitro and in vivo pharmacological characterization of SB 201993, an eicosanoid-like LTB4 receptor antagonist with anti-inflammatory activity
SARAU, H. M, FOLEY, J. J, KINGSBURY, W. D, CHAMBERS, P. A, PENDRAK, I, JAKAS, D. R, SATHE, G. M, VAN HORN, S, DAINES, R. A, GRISWOLD, D. E, SCHMIDT, D. B, MARTIN, L. D, WEBB, E. F, TZIMAS, M. N, BRETON, J. J, CHABOT-FLETCHER, M, UNDERWOOD, D. C, HAY, D. W. P
Published in Prostaglandins, leukotrienes and essential fatty acids (01.07.1999)
Published in Prostaglandins, leukotrienes and essential fatty acids (01.07.1999)
Get full text
Journal Article
Identification, substrate specificity, and inhibition of the Streptococcus pneumoniae beta-ketoacyl-acyl carrier protein synthase III (FabH)
Khandekar, S S, Gentry, D R, Van Aller, G S, Warren, P, Xiang, H, Silverman, C, Doyle, M L, Chambers, P A, Konstantinidis, A K, Brandt, M, Daines, R A, Lonsdale, J T
Published in The Journal of biological chemistry (10.08.2001)
Published in The Journal of biological chemistry (10.08.2001)
Get full text
Journal Article
First X-ray Cocrystal Structure of a Bacterial FabH Condensing Enzyme and a Small Molecule Inhibitor Achieved Using Rational Design and Homology Modeling
Daines, Robert A, Pendrak, Israil, Sham, Kelvin, Van Aller, Glenn S, Konstantinidis, Alex K, Lonsdale, John T, Janson, Cheryl A, Qiu, Xiayang, Brandt, Martin, Khandekar, Sanjay S, Silverman, Carol, Head, Martha S
Published in Journal of medicinal chemistry (02.01.2003)
Published in Journal of medicinal chemistry (02.01.2003)
Get full text
Journal Article
Total synthesis of amphotericin B
Nicolaou, K. C, Daines, R. A, Chakraborty, T. K, Ogawa, Y
Published in Journal of the American Chemical Society (01.04.1987)
Published in Journal of the American Chemical Society (01.04.1987)
Get full text
Journal Article
Stereocontrolled construction of key building blocks for the total synthesis of amphoteronolide B and amphotericin B
Nicolaou, Kyriacos C, Daines, R. A, Uenishi, J, Li, W. S, Papahatjis, D. P, Chakraborty, T. K
Published in Journal of the American Chemical Society (01.04.1987)
Published in Journal of the American Chemical Society (01.04.1987)
Get full text
Journal Article
Total synthesis of amphoteronolide B
Nicolaou, Kyriacos C, Daines, R. A, Chakraborty, T. K
Published in Journal of the American Chemical Society (01.04.1987)
Published in Journal of the American Chemical Society (01.04.1987)
Get full text
Journal Article
Pharmacology of SB-273779, a Nonpeptide Calcitonin Gene-Related Peptide 1 Receptor Antagonist
Aiyar, N, Daines, R A, Disa, J, Chambers, P A, Sauermelch, C F, Quiniou, M, Khandoudi, N, Gout, B, Douglas, S A, Willette, R N
Published in The Journal of pharmacology and experimental therapeutics (01.03.2001)
Get full text
Published in The Journal of pharmacology and experimental therapeutics (01.03.2001)
Journal Article
(E)-3-[6-[[(2,6-Dichlorophenyl)thio]methyl]-3-(2-phenylethoxy)-2-pyridinyl]-2- propenoic Acid: A High-Affinity Leukotriene B4 Receptor Antagonist with Oral Antiinflammatory Activity
Daines, Robert A, Chambers, Pamela A, Foley, James J, Griswold, Don E, Kingsbury, William D, Martin, Lenox D, Schmidt, Dulcie B, Sham, Kelvin K. C, Sarau, Henry M
Published in Journal of medicinal chemistry (13.09.1996)
Published in Journal of medicinal chemistry (13.09.1996)
Get full text
Journal Article
Quinine analogs as non-peptide calcitonin gene-related peptide (CGRP) receptor antagonists
Daines, Robert A., Sham, Kelvin K.C., Taggart, Jack J., Kingsbury, William D., Chan, James, Breen, Ann, Disa, Jyoti, Aiyar, Nambi
Published in Bioorganic & medicinal chemistry letters (21.10.1997)
Published in Bioorganic & medicinal chemistry letters (21.10.1997)
Get full text
Journal Article
Synthesis of structural analogs of leukotriene B4 and their receptor binding activity
Kingsbury, William D, Pendrak, Israil, Leber, Jack D, Boehm, Jeffery C, Mallet, Brenda, Sarau, Henry M, Foley, James J, Schmidt, Dulcie B, Daines, Robert A
Published in Journal of medicinal chemistry (01.10.1993)
Published in Journal of medicinal chemistry (01.10.1993)
Get full text
Journal Article
Trisubstituted pyridine leukotriene B4 receptor antagonists: synthesis and structure-activity relationships
Daines, Robert A, Chambers, Pamela A, Pendrak, Israil, Jakas, Dalia R, Sarau, Henry M, Foley, James J, Schmidt, Dulcie B, Kingsbury, William D
Published in Journal of medicinal chemistry (01.10.1993)
Published in Journal of medicinal chemistry (01.10.1993)
Get full text
Journal Article
(E)-3-[[[[6-(2-Carboxyethenyl)-5-[[8-(4-methoxyphenyl)octyl]oxy]-2-pyridinyl]methyl]thio]methyl]benzoic acid: a novel high-affinity leukotriene B4 receptor antagonist
Daines, Robert A, Chambers, Pamela A, Pendrak, Israil, Jakas, Dalia R, Sarau, Henry M, Foley, James J, Schmidt, Dulcie B, Griswold, Don E, Martin, Lenox D
Published in Journal of medicinal chemistry (01.09.1993)
Published in Journal of medicinal chemistry (01.09.1993)
Get full text
Journal Article
RETROSYNTHETIC AND SYNTHETIC CHEMISTRY ON AMPHOTERICIN-B - SYNTHESIS OF C(1)-C(20) AND C(21)-C(38) FRAGMENTS AND CONSTRUCTION OF THE 38-MEMBERED MACROCYCLE
NICOLAOU, KC, CHAKRABORTY, TK, DAINES, RA, SIMPKINS, NS
Published in Journal of the Chemical Society. Chemical communications (1986)
Published in Journal of the Chemical Society. Chemical communications (1986)
Get full text
Journal Article
SB 209247, a high affinity LTB4 receptor antagonist demonstrating potent antiinflammatory activity
Sarau, H M, Foley, J J, Schmidt, D B, Tzimas, M N, Martin, L D, Daines, R A, Chambers, P A, Kingsbury, W D, Griswold, D E
Published in Advances in prostaglandin, thromboxane, and leukotriene research (1995)
Get more information
Published in Advances in prostaglandin, thromboxane, and leukotriene research (1995)
Journal Article