Development of a natural product optimization strategy for inhibitors against MraY, a promising antibacterial target
Yamamoto, Kazuki, Sato, Toyotaka, Hao, Aili, Asao, Kenta, Kaguchi, Rintaro, Kusaka, Shintaro, Ruddarraju, Radhakrishnam Raju, Kazamori, Daichi, Seo, Kiki, Takahashi, Satoshi, Horiuchi, Motohiro, Yokota, Shin-ichi, Lee, Seok-Yong, Ichikawa, Satoshi
Published in Nature communications (14.06.2024)
Published in Nature communications (14.06.2024)
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Journal Article
Discovery of WQ-3810: Design, synthesis, and evaluation of 7-(3-alkylaminoazetidin-1-yl)fluoro-quinolones as orally active antibacterial agents
Itoh, Kenji, Kuramoto, Yasuhiro, Amano, Hirotaka, Kazamori, Daichi, Yazaki, Akira
Published in European journal of medicinal chemistry (20.10.2015)
Published in European journal of medicinal chemistry (20.10.2015)
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Journal Article
Evaluation of the Effects of S-Allyl-L-cysteine, S-Methyl-L-cysteine, trans-S-1-Propenyl-L-cysteine, and Their N-Acetylated and S-Oxidized Metabolites on Human CYP Activities
Amano, Hirotaka, Kazamori, Daichi, Itoh, Kenji
Published in Biological & pharmaceutical bulletin (2016)
Published in Biological & pharmaceutical bulletin (2016)
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Journal Article
Discovery of a Novel Fluoroquinolone Antibiotic Candidate WFQ-228 with Potent Antimicrobial Activity and the Potential to Overcome Major Drug Resistance
Hirano, Tatsuya, Kinoshita, Tomohiko, Kazamori, Daichi, Inoue, Satoshi, Nishimura, Kouji, Sakurai, Asuka, Ohishi, Kensuke, Kuramoto, Yasuhiro, Amano, Hirotaka, Yazaki, Akira
Published in Chemical & pharmaceutical bulletin (01.03.2018)
Published in Chemical & pharmaceutical bulletin (01.03.2018)
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Journal Article
In vitro activity of WQ-3810, a novel fluoroquinolone, against multidrug-resistant and fluoroquinolone-resistant pathogens
Kazamori, Daichi, Aoi, Hiroshi, Sugimoto, Kaori, Ueshima, Taichi, Amano, Hirotaka, Itoh, Kenji, Kuramoto, Yasuhiro, Yazaki, Akira
Published in International journal of antimicrobial agents (01.11.2014)
Published in International journal of antimicrobial agents (01.11.2014)
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Journal Article
Evaluation of the Effects of S-Allyl-L-cysteine, S-Methyl-L-cysteine, trans-S-1-Propenyl-L-cysteine, and Their N-Acetylated and S-Oxidized Metabolites on Human CYP Activities
Hirotaka Amano, Daichi Kazamori, Kenji Itoh
Published in Biological and Pharmaceutical Bulletin (01.10.2016)
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Published in Biological and Pharmaceutical Bulletin (01.10.2016)
Journal Article
Discovery of a Novel Fluoroquinolone Antibiotic Candidate WFQ-228 with Potent Antimicrobial Activity and the Potential to Overcome Major Drug Resistance
Tatsuya Hirano, Tomohiko Kinoshita, Daichi Kazamori, Satoshi Inoue, Kouji Nishimura, Asuka Sakurai, Kensuke Ohishi, Yasuhiro Kuramoto, Hirotaka Amano, Akira Yazaki
Published in Chemical and Pharmaceutical Bulletin (01.03.2018)
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Published in Chemical and Pharmaceutical Bulletin (01.03.2018)
Journal Article
The mechanism causing the difference in kinetic properties between rat CYP2D4 and human CYP2D6 in the oxidation of dextromethorphan and bufuralol
Narimatsu, Shizuo, Kazamori, Daichi, Masuda, Kazufumi, Katsu, Takashi, Funae, Yoshihiko, Naito, Shinsaku, Nakura, Hironori, Yamano, Shigeru, Hanioka, Nobumitsu
Published in Biochemical pharmacology (01.03.2009)
Published in Biochemical pharmacology (01.03.2009)
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Journal Article
Metabolism, excretion, and pharmacokinetics of S-allyl-L-cysteine in rats and dogs
Amano, Hirotaka, Kazamori, Daichi, Itoh, Kenji, Kodera, Yukihiro
Published in Drug metabolism and disposition (01.05.2015)
Published in Drug metabolism and disposition (01.05.2015)
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Journal Article
The roles of amino acid residues at positions 216 and 219 in the structural stability and metabolic functions of rat cytochrome P450 2D1 and 2D2
Narimatsu, Shizuo, Kiryu, Kimio, Yonemoto, Rei, Yoshino, Manabu, Kobatake, Mitsuko, Kazamori, Daichi, Hagino, Saori, Masuda, Kazufumi, Katsu, Takashi, Asanuma, Masato, Kumamoto, Takuya, Ishikawa, Tsutomu, Funae, Yoshihiko, Yamano, Shigeru, Hanioka, Nobumitsu, Naito, Shinsaku
Published in Chemico-biological interactions (10.03.2008)
Published in Chemico-biological interactions (10.03.2008)
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Journal Article
Novel pyridonecarboxylic acid derivative or salt thereof
Sasaki, Ayuka, Nishimura, Kouji, Kinoshita, Tomohiko, Hirano, Tatsuya, Sakurai, Asuka, Inoue, Satoshi, Arai, Mai, Kazamori, Daichi, Kuramoto, Yasuhiro
Year of Publication 07.01.2021
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Year of Publication 07.01.2021
Patent
NOVEL PYRIDONECARBOXYLIC ACID DERIVATIVE OR SALT THEREOF
KURAMOTO, Yasuhiro, KINOSHITA, Tomohiko, SAKURAI, Asuka, SASAKI, Ayuka, ARAI, Mai, KAZAMORI, Daichi, NISHIMURA, Kouji, INOUE, Satoshi, HIRANO, Tatsuya
Year of Publication 19.02.2020
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Year of Publication 19.02.2020
Patent
Pyridonecarboxylic acid derivative or salt thereof
Sasaki, Ayuka, Nishimura, Kouji, Kinoshita, Tomohiko, Hirano, Tatsuya, Sakurai, Asuka, Inoue, Satoshi, Arai, Mai, Kazamori, Daichi, Kuramoto, Yasuhiro
Year of Publication 14.01.2020
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Year of Publication 14.01.2020
Patent
NOVEL PYRIDONECARBOXYLIC ACID DERIVATIVE OR SALT THEREOF
KURAMOTO, Yasuhiro, KINOSHITA, Tomohiko, SAKURAI, Asuka, SASAKI, Ayuka, ARAI, Mai, KAZAMORI, Daichi, NISHIMURA, Kouji, INOUE, Satoshi, HIRANO, Tatsuya
Year of Publication 12.09.2019
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Year of Publication 12.09.2019
Patent
NOVEL PYRIDONECARBOXYLIC ACID DERIVATIVE OR SALT THEREOF
KURAMOTO, Yasuhiro, KINOSHITA, Tomohiko, SAKURAI, Asuka, SASAKI, Ayuka, ARAI, Mai, KAZAMORI, Daichi, NISHIMURA, Kouji, INOUE, Satoshi, HIRANO, Tatsuya
Year of Publication 24.04.2019
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Year of Publication 24.04.2019
Patent
Novel pyridonecarboxylic acid derivative or salt thereof
Sasaki, Ayuka, Nishimura, Kouji, Kinoshita, Tomohiko, Hirano, Tatsuya, Sakurai, Asuka, Inoue, Satoshi, Arai, Mai, Kazamori, Daichi, Kuramoto, Yasuhiro
Year of Publication 03.01.2019
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Year of Publication 03.01.2019
Patent