INHIBITION OF FGF-1 RECEPTOR TYROSINE KINASE ACTIVITY BY PD 161570, A NEW PROTEIN-TYROSINE KINASE INHIBITOR
Batley, Brian L, Doherty, Annette M, Hamby, James M, Lu, Gina H, Keller, Paul, Dahring, Tawny K, Hwang, Ok, Crickard, Kent, Panek, Robert L
Published in Life sciences (1973) (1998)
Published in Life sciences (1973) (1998)
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In Vitro Pharmacological Characterization of PD 166285, a New Nanomolar Potent and Broadly Active Protein Tyrosine Kinase Inhibitor
Panek, R L, Lu, G H, Klutchko, S R, Batley, B L, Dahring, T K, Hamby, J M, Hallak, H, Doherty, A M, Keiser, J A
Published in The Journal of pharmacology and experimental therapeutics (01.12.1997)
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Published in The Journal of pharmacology and experimental therapeutics (01.12.1997)
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In Vitro Biological Characterization and Antiangiogenic Effects of PD 166866, a Selective Inhibitor of the FGF-1 Receptor Tyrosine Kinase
Panek, R L, Lu, G H, Dahring, T K, Batley, B L, Connolly, C, Hamby, J M, Brown, K J
Published in The Journal of pharmacology and experimental therapeutics (01.07.1998)
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Published in The Journal of pharmacology and experimental therapeutics (01.07.1998)
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Structure−Activity Relationships for 1-Phenylbenzimidazoles as Selective ATP Site Inhibitors of the Platelet-Derived Growth Factor Receptor
Palmer, Brian D, Smaill, Jeff B, Boyd, Maruta, Boschelli, Diane H, Doherty, Annette M, Hamby, James M, Khatana, Sonya S, Kramer, James B, Kraker, Alan J, Panek, Robert L, Lu, Gina H, Dahring, Tawny K, Winters, R. Thomas, Showalter, H. D. Hollis, Denny, William A
Published in Journal of medicinal chemistry (31.12.1998)
Published in Journal of medicinal chemistry (31.12.1998)
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Inhibition of Growth Factor-Mediated Tyrosine Phosphorylation in Vascular Smooth Muscle by PD 089828, a New Synthetic Protein Tyrosine Kinase Inhibitor
Dahring, T K, Lu, G H, Hamby, J M, Batley, B L, Kraker, A J, Panek, R L
Published in The Journal of pharmacology and experimental therapeutics (01.06.1997)
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Published in The Journal of pharmacology and experimental therapeutics (01.06.1997)
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2-Substituted Aminopyrido[2,3-d]pyrimidin-7(8H)-ones. Structure−Activity Relationships Against Selected Tyrosine Kinases and in Vitro and in Vivo Anticancer Activity
Klutchko, Sylvester R, Hamby, James M, Boschelli, Diane H, Wu, Zhipei, Kraker, Alan J, Amar, Aneesa M, Hartl, Brian G, Shen, Cynthia, Klohs, Wayne D, Steinkampf, Randall W, Driscoll, Denise L, Nelson, James M, Elliott, William L, Roberts, Billy J, Stoner, Chad L, Vincent, Patrick W, Dykes, Donald J, Panek, Robert L, Lu, Gina H, Major, Terry C, Dahring, Tawny K, Hallak, Hussein, Bradford, Laura A, Showalter, H. D. Hollis, Doherty, Annette M
Published in Journal of medicinal chemistry (13.08.1998)
Published in Journal of medicinal chemistry (13.08.1998)
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Synthesis and Tyrosine Kinase Inhibitory Activity of a Series of 2-Amino-8H-pyrido[2,3-d]pyrimidines: Identification of Potent, Selective Platelet-Derived Growth Factor Receptor Tyrosine Kinase Inhibitors
Boschelli, Diane H, Wu, Zhipei, Klutchko, Sylvester R, Showalter, H. D. Hollis, Hamby, James M, Lu, Gina H, Major, Terry C, Dahring, Tawny K, Batley, Brian, Panek, Robert L, Keiser, Joan, Hartl, Brian G, Kraker, Alan J, Klohs, Wayne D, Roberts, Bill J, Patmore, Sandra, Elliott, William L, Steinkampf, Randy, Bradford, Laura A, Hallak, Hussein, Doherty, Annette M
Published in Journal of medicinal chemistry (22.10.1998)
Published in Journal of medicinal chemistry (22.10.1998)
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Soluble 2-Substituted Aminopyrido[2,3-d]pyrimidin-7-yl Ureas. Structure−Activity Relationships against Selected Tyrosine Kinases and Exploration of in Vitro and in Vivo Anticancer Activity
Schroeder, Mel C, Hamby, James M, Connolly, Cleo J. C, Grohar, Patrick J, Winters, R. Thomas, Barvian, Mark R, Moore, Charles W, Boushelle, Stacey L, Crean, Sheila M, Kraker, Alan J, Driscoll, Denise L, Vincent, Patrick W, Elliott, William L, Lu, Gina H, Batley, Brian L, Dahring, Tawny K, Major, Terry C, Panek, Robert L, Doherty, Annette M, Showalter, H. D. Hollis
Published in Journal of medicinal chemistry (07.06.2001)
Published in Journal of medicinal chemistry (07.06.2001)
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