Organocatalytic Asymmetric Conjugate Additions to Cyclopent-1-enecarbaldehyde: A Critical Assessment of Organocatalytic Approaches towards the Telaprevir Bicyclic Core
Bernardi, Luca, Fochi, Mariafrancesca, Carbone, Riccardo, Martinelli, Ada, Fox, Martin E., Cobley, Christopher J., Kandagatla, Bhaskar, Oruganti, Srinivas, Dahanukar, Vilas H., Carlone, Armando
Published in Chemistry : a European journal (21.12.2015)
Published in Chemistry : a European journal (21.12.2015)
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Journal Article
Investigation of a Kumada Cross Coupling Reaction for Large-Scale Production of (2S, 7R, E)‑2-Isopropyl-7-(4-methoxy-3-(3-methoxypropoxy)benzyl)‑N,N,8-trimethylnon-4-enamide
Gangula, Srinivas, Neelam, Uday Kumar, Baddam, Sudharkar Reddy, Dahanukar, Vilas H, Bandichhor, Rakeshwar
Published in Organic process research & development (20.03.2015)
Published in Organic process research & development (20.03.2015)
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Journal Article
Synthesis and Optimization of Canagliflozin by Employing Quality by Design (QbD) Principles
Metil, Dattatray S, Sonawane, Swapnil P, Pachore, Sharad S, Mohammad, Aaseef, Dahanukar, Vilas H, McCormack, Peter J, Reddy, Ch. Venkatramana, Bandichhor, Rakeshwar
Published in Organic process research & development (19.01.2018)
Published in Organic process research & development (19.01.2018)
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Journal Article
A morpholine-free process amenable convergent synthesis of apixaban: a potent factor Xa inhibitor
Nevuluri, Narasimha Rao, Rapolu, Rajesh Kumar, Iqbal, Javed, Kandagatla, Bhaskar, Sen, Saikat, Dahanukar, Vilas H., Oruganti, Srinivas
Published in Monatshefte für Chemie (01.08.2017)
Published in Monatshefte für Chemie (01.08.2017)
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Journal Article
Synthesis and Process Optimization of Boceprevir: A Protease Inhibitor Drug
Bhalerao, Dinesh S, Arkala, Anil Kumar Reddy, Madhavi, Y. V, Nagaraju, M, Gade, Srinivas Reddy, Kumar, U. K. Syam, Bandichhor, Rakeshwar, Dahanukar, Vilas H
Published in Organic process research & development (20.11.2015)
Published in Organic process research & development (20.11.2015)
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Journal Article
Practical, Asymmetric Route to Sitagliptin and Derivatives: Development and Origin of Diastereoselectivity
Gutierrez, Osvaldo, Metil, Dattatray, Dwivedi, Namrata, Gudimalla, Nagaraju, Chandrashekar, E. R. R, Dahanukar, Vilas H, Bhattacharya, Apurba, Bandichhor, Rakeshwar, Kozlowski, Marisa C
Published in Organic letters (03.04.2015)
Published in Organic letters (03.04.2015)
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Journal Article
Correction to “Synthesis and Optimization of Canagliflozin by Employing Quality by Design (QbD) Principles”
Metil, Dattatray S, Murugan, Andiappan, Sonawane, Swapnil P, Pachore, Sharad S, Mohammad, Aaseef, Dahanukar, Vilas H, McCormack, Peter J, Reddy, Ch. Venkatramana, Bandichhor, Rakeshwar
Published in Organic process research & development (16.03.2018)
Published in Organic process research & development (16.03.2018)
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Journal Article
One pot oxidative dehydration - oxidation of polyhydroxyhexanal oxime to polyhydroxy oxohexanenitrile: A versatile methodology for the facile access of azasugar alkaloids
Khobare, Sandip R., Gajare, Vikas, Reddy, E. Vishnuvardhan, Datrika, Rajender, Banda, Malavika, Siddaiah, Vidavalur, Pachore, Sharad S., Timanna, Upadhya, Dahanukar, Vilas H., Syam Kumar, U.K.
Published in Carbohydrate research (29.11.2016)
Published in Carbohydrate research (29.11.2016)
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Journal Article
Successful utilization of β-ketonitrile in Biginelli reaction: synthesis of 5-cyanodihydropyrimidine
Pachore, Sharad S, Ambhaikar, Narendra B, Siddaiah, Vidavalur, Khobare, Sandip R, Kumar, Sarvesh, Dahanukar, Vilas H, Kumar, U K Syam
Published in Journal of chemical sciences (Bangalore, India) (2018)
Published in Journal of chemical sciences (Bangalore, India) (2018)
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Journal Article
Enantiospecific Synthesis of 3-Fluoromethyl-, 3-Hydroxymethyl-, and 3-Chloromethyl-1,2,3,4-tetrahydroisoquinolines as Selective Inhibitors of Phenylethanolamine N-Methyltransferase versus the α2-Adrenoceptor
Grunewald, Gary L, Caldwell, Timothy M, Li, Qifang, Dahanukar, Vilas H, McNeil, Brynn, Criscione, Kevin R
Published in Journal of medicinal chemistry (21.10.1999)
Published in Journal of medicinal chemistry (21.10.1999)
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Journal Article
New and Practical Method for Synthesis of 1- and 1,3-Substituted Xanthines
Zavialov, Ilia A, Dahanukar, Vilas H, Nguyen, Hoa, Orr, Cecilia, Andrews, David R
Published in Organic letters (24.06.2004)
Published in Organic letters (24.06.2004)
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Journal Article
Effects of a 3-alkyl-, 4-hydroxy- and/or 8-aromatic-substituent on the phenylethanolamine N-methyltransferase inhibitor potency and α2-adrenoceptor affinity of 2,3,4,5-tetrahydro-1H-2-benzazepines
GRUNEWALD, Gary L, DAHANUKAR, Vilas H, CRISCIONE, Kevin R
Published in Bioorganic & medicinal chemistry (01.08.2001)
Published in Bioorganic & medicinal chemistry (01.08.2001)
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Journal Article
Development of an Efficient Process for the Preparation of Sch 39166: Aziridinium Chemistry on Scale
Gala, Dinesh, Dahanukar, Vilas H, Eckert, Jeffery M, Lucas, Brian S, Schumacher, Doris P, Zavialov, Ilia A, Buholzer, Patrik, Kubisch, Peter, Mergelsberg, Ingrid, Scherer, Dominik
Published in Organic process research & development (01.09.2004)
Published in Organic process research & development (01.09.2004)
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Journal Article
Reaction of aziridinium ions with organometallic reagents: optimization of the key step of ecopipam synthesis
Andrews, David R, Dahanukar, Vilas H, Eckert, Jeffrey M, Gala, Dinesh, Lucas, Brian S, Schumacher, Doris P, Zavialov, Ilia A
Published in Tetrahedron letters (26.08.2002)
Published in Tetrahedron letters (26.08.2002)
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Journal Article
New and Practical Method for Synthesis of 1- and 1,3-Substituted Xanthines
Zavialov, Ilia A, Dahanukar, Vilas H, Nguyen, Hoa, Orr, Cecilia, Zhang, Fucheng, Andrews, David R
Published in Organic letters (19.08.2004)
Published in Organic letters (19.08.2004)
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