Design and Synthesis of Janus Kinase 2 (JAK2) and Histone Deacetlyase (HDAC) Bispecific Inhibitors Based on Pacritinib and Evidence of Dual Pathway Inhibition in Hematological Cell Lines
Yang, Eugene Guorong, Mustafa, Nurulhuda, Tan, Eng Chong, Poulsen, Anders, Ramanujulu, Pondy Murugappan, Chng, Wee Joo, Yen, Jeffrey J. Y, Dymock, Brian W
Published in Journal of medicinal chemistry (22.09.2016)
Published in Journal of medicinal chemistry (22.09.2016)
Get full text
Journal Article
Hydrogen sulfide promotes adipogenesis in 3T3L1 cells
Tsai, Chin-Yi, Peh, Meng Teng, Feng, Wei, Dymock, Brian William, Moore, Philip Keith
Published in PloS one (30.03.2015)
Published in PloS one (30.03.2015)
Get full text
Journal Article
Design and Synthesis of Ligand Efficient Dual Inhibitors of Janus Kinase (JAK) and Histone Deacetylase (HDAC) Based on Ruxolitinib and Vorinostat
Yao, Lianbin, Mustafa, Nurulhuda, Tan, Eng Chong, Poulsen, Anders, Singh, Prachi, Duong-Thi, Minh-Dao, Lee, Jeannie X. T, Ramanujulu, Pondy Murugappan, Chng, Wee Joo, Yen, Jeffrey J. Y, Ohlson, Sten, Dymock, Brian W
Published in Journal of medicinal chemistry (26.10.2017)
Published in Journal of medicinal chemistry (26.10.2017)
Get full text
Journal Article
Merging of ruxolitinib and vorinostat leads to highly potent inhibitors of JAK2 and histone deacetylase 6 (HDAC6)
Yao, Lianbin, Ramanujulu, Pondy Murugappan, Poulsen, Anders, Ohlson, Sten, Dymock, Brian W.
Published in Bioorganic & medicinal chemistry letters (15.08.2018)
Published in Bioorganic & medicinal chemistry letters (15.08.2018)
Get full text
Journal Article
Dual blockade of the lipid kinase PIP4Ks and mitotic pathways leads to cancer-selective lethality
Kitagawa, Mayumi, Liao, Pei-Ju, Lee, Kyung Hee, Wong, Jasmine, Shang, See Cheng, Minami, Noriaki, Sampetrean, Oltea, Saya, Hideyuki, Lingyun, Dai, Prabhu, Nayana, Diam, Go Ka, Sobota, Radoslaw, Larsson, Andreas, Nordlund, Pär, McCormick, Frank, Ghosh, Sujoy, Epstein, David M., Dymock, Brian W., Lee, Sang Hyun
Published in Nature communications (19.12.2017)
Published in Nature communications (19.12.2017)
Get full text
Journal Article
Discovery of New H2S Releasing Phosphordithioates and 2,3-Dihydro-2-phenyl-2-sulfanylenebenzo[d][1,3,2]oxazaphospholes with Improved Antiproliferative Activity
Feng, Wei, Teo, Xin-Yi, Novera, Wisna, Ramanujulu, Pondy Murugappan, Liang, Dong, Huang, Dejian, Moore, Philip K, Deng, Lih-Wen, Dymock, Brian W
Published in Journal of medicinal chemistry (27.08.2015)
Published in Journal of medicinal chemistry (27.08.2015)
Get full text
Journal Article
Design and synthesis of potent dual inhibitors of JAK2 and HDAC based on fusing the pharmacophores of XL019 and vorinostat
Chu-Farseeva, Yu-yi, Mustafa, Nurulhuda, Poulsen, Anders, Tan, Eng Chong, Yen, Jeffrey J.Y., Chng, Wee Joo, Dymock, Brian W.
Published in European journal of medicinal chemistry (05.10.2018)
Published in European journal of medicinal chemistry (05.10.2018)
Get full text
Journal Article
Predicting Tacrolimus Concentrations in the Skin of Adult Kidney Transplant Recipients: A Feasibility Study
Sartain, Felicity, Viecelli, Andrea K, Veitch, Margaret, Franklin, Michael E, Dymock, Brian W, Wells, James W, Campbell, Scott B
Published in Transplant international (2024)
Published in Transplant international (2024)
Get full text
Journal Article
Discovery of a potent histone deacetylase (HDAC) 3/6 selective dual inhibitor
Soumyanarayanan, Uttara, Ramanujulu, Pondy Murugappan, Mustafa, Nurulhuda, Haider, Shozeb, Fang Nee, Adina Huey, Tong, Jie Xin, Tan, Kevin S.W., Chng, Wee Joo, Dymock, Brian W.
Published in European journal of medicinal chemistry (15.12.2019)
Published in European journal of medicinal chemistry (15.12.2019)
Get full text
Journal Article
Discovery of the cancer cell selective dual acting anti-cancer agent (Z)-2-(1H-indol-3-yl)-3-(isoquinolin-5-yl)acrylonitrile (A131)
See, Cheng Shang, Kitagawa, Mayumi, Liao, Pei-Ju, Lee, Kyung Hee, Wong, Jasmine, Lee, Sang Hyun, Dymock, Brian W.
Published in European journal of medicinal chemistry (05.08.2018)
Published in European journal of medicinal chemistry (05.08.2018)
Get full text
Journal Article
Towards Selective Mycobacterial ClpP1P2 Inhibitors with Reduced Activity against the Human Proteasome
Moreira, Wilfried, Santhanakrishnan, Sridhar, Ngan, Grace J Y, Low, Choon Bing, Sangthongpitag, Kanda, Poulsen, Anders, Dymock, Brian W, Dick, Thomas
Published in Antimicrobial agents and chemotherapy (01.05.2017)
Published in Antimicrobial agents and chemotherapy (01.05.2017)
Get full text
Journal Article
Discovery of the Macrocycle 11-(2-Pyrrolidin-1-yl-ethoxy)-14,19-dioxa-5,7,26-triaza-tetracyclo[19.3.1.1(2,6).1(8,12)]heptacosa-1(25),2(26),3,5,8,10,12(27),16,21,23-decaene (SB1518), a Potent Janus Kinase 2/Fms-Like Tyrosine Kinase-3 (JAK2/FLT3) Inhibitor for the Treatment of Myelofibrosis and Lymphoma
William, Anthony D, Lee, Angeline C.-H, Blanchard, Stéphanie, Poulsen, Anders, Teo, Ee Ling, Nagaraj, Harish, Tan, Evelyn, Chen, Dizhong, Williams, Meredith, Sun, Eric T, Goh, Kee Chuan, Ong, Wai Chung, Goh, Siok Kun, Hart, Stefan, Jayaraman, Ramesh, Pasha, Mohammed Khalid, Ethirajulu, Kantharaj, Wood, Jeanette M, Dymock, Brian W
Published in Journal of medicinal chemistry (14.07.2011)
Published in Journal of medicinal chemistry (14.07.2011)
Get full text
Journal Article
Hydrogen sulfide is an endogenous regulator of aging in Caenorhabditis elegans
Qabazard, Bedoor, Li, Ling, Gruber, Jan, Peh, Meng Teng, Ng, Li Fang, Kumar, Srinivasan Dinesh, Rose, Peter, Tan, Choon-Hong, Dymock, Brian W, Wei, Feng, Swain, Suresh C, Halliwell, Barry, Stürzenbaum, Stephen R, Moore, Philip K
Published in Antioxidants & redox signaling (01.06.2014)
Published in Antioxidants & redox signaling (01.06.2014)
Get more information
Journal Article
Bortezomib Warhead-Switch Confers Dual Activity against Mycobacterial Caseinolytic Protease and Proteasome and Selectivity against Human Proteasome
Moreira, Wilfried, Santhanakrishnan, Sridhar, Dymock, Brian W, Dick, Thomas
Published in Frontiers in microbiology (27.04.2017)
Published in Frontiers in microbiology (27.04.2017)
Get full text
Journal Article