Discovery and Optimization of Novel Antagonists to the Human Neurokinin‑3 Receptor for the Treatment of Sex-Hormone Disorders (Part I)
Hoveyda, Hamid R, Fraser, Graeme L, Roy, Marie-Odile, Dutheuil, Guillaume, Batt, Frédéric, El Bousmaqui, Mohamed, Korac, Julien, Lenoir, François, Lapin, Alexey, Noël, Sophie, Blanc, Sébastien
Published in Journal of medicinal chemistry (09.04.2015)
Published in Journal of medicinal chemistry (09.04.2015)
Get full text
Journal Article
Optimization of Novel Antagonists to the Neurokinin‑3 Receptor for the Treatment of Sex-Hormone Disorders (Part II)
Hoveyda, Hamid R, Fraser, Graeme L, Dutheuil, Guillaume, El Bousmaqui, Mohamed, Korac, Julien, Lenoir, François, Lapin, Alexey, Noël, Sophie
Published in ACS medicinal chemistry letters (09.07.2015)
Published in ACS medicinal chemistry letters (09.07.2015)
Get full text
Journal Article
EP102: Pharmacological Inhibition of METTL3 Elicits Tumor Growth Inhibition In Vivo and Demonstrates Synergy with Venetoclax in Various AML Models
Fraser, Graeme, Sorlet, Catherine, Parmentier, Nicolas, Hartiel, Anne-France, Hospied, Sandrine, Mompied, Clement, Absil, Genevieve, Oukoloff, Killian, Dutheuil, Guillaume
Published in Blood (02.11.2023)
Published in Blood (02.11.2023)
Get full text
Journal Article
Lithiated Carbamates: Chiral Carbenoids for Iterative Homologation of Boranes and Boronic Esters
Stymiest, Jake L., Dutheuil, Guillaume, Mahmood, Adeem, Aggarwal, Varinder K.
Published in Angewandte Chemie (01.10.2007)
Published in Angewandte Chemie (01.10.2007)
Get full text
Journal Article
Abstract 6282: EP102: Pharmacological inhibition of METTL3 arrests tumor progression and prolongs survival in CDX and PDX models of AML
Fraser, Graeme, Sorlet, Catherine, Parmentier, Nicolas, Brunel, Elodie, Hartiel, Anne-France, Oukoloff, Killian, Dutheuil, Guillaume
Published in Cancer research (Chicago, Ill.) (04.04.2023)
Published in Cancer research (Chicago, Ill.) (04.04.2023)
Get full text
Journal Article
Abstract 3233: EP102: Pharmacological Inhibition of METTL3 causes tumor growth inhibition and prolongs survival in preclinical models of NSCLC, ovarian and squamous cell carcinoma
Fraser, Graeme, Sorlet, Catherine, Parmentier, Nicolas, Brunel, Elodie, Coremans, Christian, Rorive, Sarah, Hartiel, Anne-France, Oukoloff, Killian, Dutheuil, Guillaume
Published in Cancer research (Chicago, Ill.) (22.03.2024)
Published in Cancer research (Chicago, Ill.) (22.03.2024)
Get full text
Journal Article
Synthesis of tetrasubstituted α-fluoroenones
Dutheuil, Guillaume, Couve-Bonnaire, Samuel, Pannecoucke, Xavier
Published in Tetrahedron (01.08.2009)
Published in Tetrahedron (01.08.2009)
Get full text
Journal Article
Stereocontrolled Synthesis of Carbon Chains Bearing Contiguous Methyl Groups by Iterative Boronic Ester Homologations: Application to the Total Synthesis of (+)-Faranal
Dutheuil, Guillaume, Webster, Matthew P, Worthington, Paul A, Aggarwal, Varinder K
Published in Angewandte Chemie (International ed.) (10.08.2009)
Published in Angewandte Chemie (International ed.) (10.08.2009)
Get full text
Journal Article
Straightforward asymmetric synthesis of Ala-Psi[CF=CH]-Pro, a proline-containing pseudodipeptide bearing a fluoroolefin as a peptide bond mimic
Dutheuil, Guillaume, Pierry, Camille, Villiers, Emilie, Couve-Bonnaire, Samuel, Pannecoucke, Xavier
Published in New journal of chemistry (01.01.2013)
Published in New journal of chemistry (01.01.2013)
Get full text
Journal Article