Characteristic Physical Properties and Structural Fragments of Marketed Oral Drugs
Vieth, Michal, Siegel, Miles G, Higgs, Richard E, Watson, Ian A, Robertson, Daniel H, Savin, Kenneth A, Durst, Gregory L, Hipskind, Philip A
Published in Journal of medicinal chemistry (01.01.2004)
Published in Journal of medicinal chemistry (01.01.2004)
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Journal Article
Identification of potent and selective retinoic acid receptor gamma (RARγ) antagonists for the treatment of osteoarthritis pain using structure based drug design
Hughes, Norman E., Bleisch, Thomas J., Jones, Scott A., Richardson, Timothy I., Doti, Robert A., Wang, Yong, Stout, Stephanie L., Durst, Gregory L., Chambers, Mark G., Oskins, Jennifer L., Lin, Chaohua, Adams, Lisa A., Page, Todd J., Barr, Robert J., Zink, Richard W., Osborne, Harold, Montrose-Rafizadeh, Chahrzad, Norman, Bryan H.
Published in Bioorganic & medicinal chemistry letters (15.07.2016)
Published in Bioorganic & medicinal chemistry letters (15.07.2016)
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Journal Article
Structural features underlying raloxifene’s biophysical interaction with bone matrix
Bivi, Nicoletta, Hu, Haitao, Chavali, Balagopalakrishna, Chalmers, Michael J., Reutter, Christopher T., Durst, Gregory L., Riley, Anna, Sato, Masahiko, Allen, Matthew R., Burr, David B., Dodge, Jeffrey A.
Published in Bioorganic & medicinal chemistry (15.02.2016)
Published in Bioorganic & medicinal chemistry (15.02.2016)
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Journal Article
Corrigendum to “Structural features underlying raloxifene’s biophysical interaction with bone matrix” [Bioorg. Med. Chem. 24 (2016) 759–767]
Bivi, Nicoletta, Hu, Haitao, Chavali, Balagopalakrishna, Chalmers, Michael J., Reutter, Christopher T., Durst, Gregory L., Riley, Anna, Sato, Masahiko, Allen, Matthew R., Burr, David B., Dodge, Jeffrey A.
Published in Bioorganic & medicinal chemistry (15.09.2016)
Published in Bioorganic & medicinal chemistry (15.09.2016)
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Journal Article
Benzopyrans Are Selective Estrogen Receptor β Agonists with Novel Activity in Models of Benign Prostatic Hyperplasia
Norman, Bryan H, Dodge, Jeffrey A, Richardson, Timothy I, Borromeo, Peter S, Lugar, Charles W, Jones, Scott A, Chen, Keyue, Wang, Yong, Durst, Gregory L, Barr, Robert J, Montrose-Rafizadeh, Chahrzad, Osborne, Harold E, Amos, Robert M, Guo, Sherry, Boodhoo, Amechand, Krishnan, Venkatesh
Published in Journal of medicinal chemistry (19.10.2006)
Published in Journal of medicinal chemistry (19.10.2006)
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Journal Article
Design and synthesis of a novel series of [1-(4-hydroxy-benzyl)-1H-indol-5-yloxy]-acetic acid compounds as potent, selective, thyroid hormone receptor β agonists
Burkholder, Timothy P., Cunningham, Brian E., Clayton, Joshua R., Lander, Peter A., Brown, Matthew L., Doti, Robert A., Durst, Gregory L., Montrose-Rafizadeh, Chahrzad, King, Constance, Osborne, Harold E., Amos, Robert M., Zink, Richard W., Stramm, Lawrence E., Burris, Thomas P., Cardona, Guemalli, Konkol, Debra L., Reidy, Charles, Christe, Michael E., Genin, Michael J.
Published in Bioorganic & medicinal chemistry letters (01.04.2015)
Published in Bioorganic & medicinal chemistry letters (01.04.2015)
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Journal Article
Benzopyrans as selective estrogen receptor β agonists (SERBAs). Part 3: Synthesis of cyclopentanone and cyclohexanone intermediates for C-ring modification
Richardson, Timothy I., Dodge, Jeffrey A., Durst, Gregory L., Pfeifer, Lance A., Shah, Jikesh, Wang, Yong, Durbin, Jim D., Krishnan, Venkatesh, Norman, Bryan H.
Published in Bioorganic & medicinal chemistry letters (01.09.2007)
Published in Bioorganic & medicinal chemistry letters (01.09.2007)
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Journal Article
Benzopyrans as selective estrogen receptor β agonists (SERBAs). Part 4: Functionalization of the benzopyran A-ring
Norman, Bryan H., Richardson, Timothy I., Dodge, Jeffrey A., Pfeifer, Lance A., Durst, Gregory L., Wang, Yong, Durbin, Jim D., Krishnan, Venkatesh, Dinn, Sean R., Liu, Shengquan, Reilly, John E., Ryter, Kendal T.
Published in Bioorganic & medicinal chemistry letters (15.09.2007)
Published in Bioorganic & medicinal chemistry letters (15.09.2007)
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Journal Article
Interaction of Cyclohexanediones with Acetyl Coenzyme-A Carboxylase and an Artificial Target-Site Antibody Mimic: A Comparative Molecular Field Analysis
Webb, Steve R, Durst, Gregory L, Pernich, Dan, Hall, J. Christopher
Published in Journal of agricultural and food chemistry (01.06.2000)
Published in Journal of agricultural and food chemistry (01.06.2000)
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Journal Article
Three-Dimensional Quantitative Structure-Permeability Relationship Analysis for a Series of Inhibitors of Rhinovirus Replication
Ekins, Sean, Durst, Gregory L, Stratford, Robert E, Thorner, David A, Lewis, Richard, Loncharich, Richard J, Wikel, James H
Published in Journal of Chemical Information and Computer Sciences (01.11.2001)
Published in Journal of Chemical Information and Computer Sciences (01.11.2001)
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Journal Article
A Target Enablement Package for the Inhibition of SHIP1 as a Therapeutic Strategy for the Treatment of Alzheimer’s Disease
Richardson, Timothy I, Jesudason, Cynthia D, Lobb, Karen L, Durst, Gregory L, Clayton, Brent, Massey, Steven M, Beck, Daniel E, Zhang, Zhong‐Yin, Dong, Jiajun, Lin, Jianping, Miao, Jinmin, Putt, Karson S, Mesecar, Andrew D, Hamdani, Adam K, Lendy, Emma K, Souza, Sarah, Jacobson, Marlene, Salvo, Jerry Di, Chu, Shaoyou, Mason, Emily R, Oblak, Adrian L, Soni, Disha, Quinney, Sara K, Silva, Larissa L, Kandasamy, Murugesh, Masters, Andrea R, Rizzo, Stacey J Sukoff, Doolen, Suzanne, Huang, Kun, Zhang, Jie, Lamb, Bruce T, Palkowitz, Alan D
Published in Alzheimer's & dementia (01.12.2022)
Published in Alzheimer's & dementia (01.12.2022)
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Journal Article
Identification of potent and selective retinoic acid receptor gamma (RARγ) antagonists for the treatment of osteoarthritis pain using structure based drug design
Hughes, Norman E., Bleisch, Thomas J., Jones, Scott A., Richardson, Timothy I., Doti, Robert A., Wang, Yong, Stout, Stephanie L., Durst, Gregory L., Chambers, Mark G., Oskins, Jennifer L., Lin, Chaohua, Adams, Lisa A., Page, Todd J., Barr, Robert J., Zink, Richard W., Osborne, Harold, Montrose-Rafizadeh, Chahrzad, Norman, Bryan H.
Published in Bioorganic & medicinal chemistry letters (01.07.2016)
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Published in Bioorganic & medicinal chemistry letters (01.07.2016)
Journal Article
Acyl Sulfonamide Anti-Proliferatives: Benzene Substituent Structure−Activity Relationships for a Novel Class of Antitumor Agents
Lobb, Karen L, Hipskind, Philip A, Aikins, James A, Alvarez, Enrique, Cheung, Yiu-Yin, Considine, Eileen L, De Dios, Alfonso, Durst, Gregory L, Ferritto, Rafael, Grossman, Cora Sue, Giera, Deborah D, Hollister, Beth A, Huang, Zhongping, Iversen, Philip W, Law, Kevin L, Li, Tiechao, Lin, Ho-Shen, Lopez, Beatriz, Lopez, Jose E, Cabrejas, Luisa M. Martin, McCann, Denis J, Molero, Victoriano, Reilly, John E, Richett, Michael E, Shih, Chuan, Teicher, Beverly, Wikel, James H, White, Wesley T, Mader, Mary M
Published in Journal of medicinal chemistry (21.10.2004)
Published in Journal of medicinal chemistry (21.10.2004)
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Journal Article
Molecular mechanics (MM2) calculations and cone angles of phosphine ligands
Chin, Mian, Durst, Gregory L., Head, Simone R., Bock, Paul L., Mosbo, John A.
Published in Journal of organometallic chemistry (17.05.1994)
Published in Journal of organometallic chemistry (17.05.1994)
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Journal Article
Substituted benzopyrans as selective estrogen receptor-beta agonists
DURST GREGORY L, RICHARDSON TIMOTHY I, NORMAN BRYAN H, PFEIFER LANCE A
Year of Publication 10.05.2007
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Year of Publication 10.05.2007
Patent
Substituted benzopyrans as selective estrogen receptor-beta agonists
DURST GREGORY L, RICHARDSON TIMOTHY I, NORMAN BRYAN H, PFEIFER LANCE A
Year of Publication 07.09.2006
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Year of Publication 07.09.2006
Patent