The role of histamine H1 and H4 receptors in allergic inflammation: the search for new antihistamines
Thurmond, Robin L, Gelfand, Erwin W, Dunford, Paul J
Published in Nature reviews. Drug discovery (01.01.2008)
Published in Nature reviews. Drug discovery (01.01.2008)
Get full text
Journal Article
The CSF-1-receptor inhibitor, JNJ-40346527 (PRV-6527), reduced inflammatory macrophage recruitment to the intestinal mucosa and suppressed murine T cell mediated colitis
Manthey, Carl L, Moore, Beverley A, Chen, Yanqing, Loza, Matthew J, Yao, Xiang, Liu, Hao, Belkowski, Stanley M, Raymond-Parks, Holly, Dunford, Paul J, Leon, Francisco, Towne, Jennifer E, Plevy, Scott E
Published in PloS one (11.11.2019)
Published in PloS one (11.11.2019)
Get full text
Journal Article
Histamine H4 receptor antagonists are superior to traditional antihistamines in the attenuation of experimental pruritus
Dunford, Paul J., MSc, Williams, Kacy N., BS, Desai, Pragnya J., MSc, Karlsson, Lars, MD, PhD, McQueen, Daniel, PhD, Thurmond, Robin L., PhD
Published in Journal of allergy and clinical immunology (2007)
Published in Journal of allergy and clinical immunology (2007)
Get full text
Journal Article
The histamine H₄ receptor antagonist, JNJ 39758979, is effective in reducing histamine-induced pruritus in a randomized clinical study in healthy subjects
Kollmeier, Alexa, Francke, Klaus, Chen, Bin, Dunford, Paul J, Greenspan, Andrew J, Xia, Yichuan, Xu, Xie L, Zhou, Bei, Thurmond, Robin L
Published in The Journal of pharmacology and experimental therapeutics (01.07.2014)
Published in The Journal of pharmacology and experimental therapeutics (01.07.2014)
Get full text
Journal Article
The histamine H4 receptor mediates inflammation and Th17 responses in preclinical models of arthritis
Cowden, Jeffery M, Yu, Fuqu, Banie, Homayon, Farahani, Mandana, Ling, Ping, Nguyen, Steven, Riley, Jason P, Zhang, Mai, Zhu, Jian, Dunford, Paul J, Thurmond, Robin L
Published in Annals of the rheumatic diseases (01.03.2014)
Published in Annals of the rheumatic diseases (01.03.2014)
Get full text
Journal Article
The histamine H 4 receptor mediates inflammation and Th17 responses in preclinical models of arthritis
Cowden, Jeffery M, Yu, Fuqu, Banie, Homayon, Farahani, Mandana, Ling, Ping, Nguyen, Steven, Riley, Jason P, Zhang, Mai, Zhu, Jian, Dunford, Paul J, Thurmond, Robin L
Published in Annals of the rheumatic diseases (01.03.2014)
Published in Annals of the rheumatic diseases (01.03.2014)
Get full text
Journal Article
The Histamine H4 Receptor Mediates Allergic Airway Inflammation by Regulating the Activation of CD4+ T Cells
Dunford, Paul J, O'Donnell, Niall, Riley, Jason P, Williams, Kacy N, Karlsson, Lars, Thurmond, Robin L
Published in The Journal of immunology (1950) (01.06.2006)
Published in The Journal of immunology (1950) (01.06.2006)
Get full text
Journal Article
A Potent and Selective Histamine H4 Receptor Antagonist with Anti-Inflammatory Properties
Thurmond, Robin L, Desai, Pragnya J, Dunford, Paul J, Fung-Leung, Wai-Ping, Hofstra, Claudia L, Jiang, Wen, Nguyen, Steven, Riley, Jason P, Sun, Siquan, Williams, Kacy N, Edwards, James P, Karlsson, Lars
Published in The Journal of pharmacology and experimental therapeutics (01.04.2004)
Published in The Journal of pharmacology and experimental therapeutics (01.04.2004)
Get full text
Journal Article
Toreforant, an orally active histamine H 4 -receptor antagonist, in patients with active rheumatoid arthritis despite methotrexate: mechanism of action results from a phase 2, multicenter, randomized, double-blind, placebo-controlled synovial biopsy study
Boyle, David L, DePrimo, Samuel E, Calderon, Cesar, Chen, Dion, Dunford, Paul J, Barchuk, William, Firestein, Gary S, Thurmond, Robin L
Published in Inflammation research (01.04.2019)
Published in Inflammation research (01.04.2019)
Get full text
Journal Article
Toreforant, an orally active histamine H4-receptor antagonist, in patients with active rheumatoid arthritis despite methotrexate: mechanism of action results from a phase 2, multicenter, randomized, double-blind, placebo-controlled synovial biopsy study
Boyle, David L., DePrimo, Samuel E., Calderon, Cesar, Chen, Dion, Dunford, Paul J., Barchuk, William, Firestein, Gary S., Thurmond, Robin L.
Published in Inflammation research (01.04.2019)
Published in Inflammation research (01.04.2019)
Get full text
Journal Article
Leukotriene A(4) hydrolase inhibition attenuates allergic airway inflammation and hyperresponsiveness
Rao, Navin L, Riley, Jason P, Banie, Homayon, Xue, Xiaohua, Sun, Binggang, Crawford, Shelby, Lundeen, Katherine A, Yu, Fuqu, Karlsson, Lars, Fourie, Anne M, Dunford, Paul J
Published in American journal of respiratory and critical care medicine (01.05.2010)
Published in American journal of respiratory and critical care medicine (01.05.2010)
Get full text
Journal Article
Leukotriene A4 Hydrolase Inhibition Attenuates Allergic Airway Inflammation and Hyperresponsiveness
RAO, Navin L, RILEY, Jason P, DUNFORD, Paul J, BANIE, Homayon, XIAOHUA XUE, BINGGANG SUN, CRAWFORD, Shelby, LUNDEEN, Katherine A, FUQU YU, KARLSSON, Lars, FOURIE, Anne M
Published in American journal of respiratory and critical care medicine (01.05.2010)
Published in American journal of respiratory and critical care medicine (01.05.2010)
Get full text
Journal Article
Anti-Inflammatory Activity of a Potent, Selective Leukotriene A4 Hydrolase Inhibitor in Comparison with the 5-Lipoxygenase Inhibitor Zileuton
Rao, Navin L, Dunford, Paul J, Xue, Xiaohua, Jiang, Xiaohui, Lundeen, Katherine A, Coles, Fawn, Riley, Jason P, Williams, Kacy N, Grice, Cheryl A, Edwards, James P, Karlsson, Lars, Fourie, Anne M
Published in The Journal of pharmacology and experimental therapeutics (01.06.2007)
Published in The Journal of pharmacology and experimental therapeutics (01.06.2007)
Get full text
Journal Article
Antagonism of the histamine H4 receptor reduces LPS-induced TNF production in vivo
Cowden, Jeffery M., Yu, Fuqu, Challapalli, Mamatha, Huang, Jing-Feng, Kim, Sunhwa, Fung-Leung, Wai-Ping, Ma, Jing Ying, Riley, Jason P., Zhang, Mai, Dunford, Paul J., Thurmond, Robin L.
Published in Inflammation research (01.06.2013)
Published in Inflammation research (01.06.2013)
Get full text
Journal Article