Do 2‑(Benzoyl)piperidines Represent a Novel Class of hDAT Reuptake Inhibitors?
Jones, Charles B., Eltit, Jose M., Dukat, Małgorzata
Published in ACS chemical neuroscience (15.02.2023)
Published in ACS chemical neuroscience (15.02.2023)
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Journal Article
Non-conserved residues dictate dopamine transporter selectivity for the potent synthetic cathinone and psychostimulant MDPV
Steele, Tyler W.E., Spires, Zachary, Jones, Charles B., Glennon, Richard A., Dukat, Małgorzata, Eltit, Jose M.
Published in Neuropharmacology (01.12.2021)
Published in Neuropharmacology (01.12.2021)
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Journal Article
Binding and functional structure-activity similarities of 4-substituted 2,5-dimethoxyphenyl isopropylamine analogues at 5-HT2A and 5-HT2B serotonin receptors
Hemanth, Prithvi, Nistala, Pallavi, Nguyen, Vy T., Eltit, Jose M., Glennon, Richard A., Dukat, Małgorzata
Published in Frontiers in pharmacology (24.01.2023)
Published in Frontiers in pharmacology (24.01.2023)
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Journal Article
Structure-Activity Relationships of Synthetic Cathinones
Glennon, Richard A., Dukat, Małgorzata
Published in Current topics in behavioral neurosciences (01.01.2017)
Published in Current topics in behavioral neurosciences (01.01.2017)
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Book Chapter
Journal Article
A new chemotype inhibitor for the human organic cation transporter 3 (hOCT3)
Pan, Xiaolei, Iyer, Kavita A., Liu, Hebing, Sweet, Douglas H., Dukat, Małgorzata
Published in Bioorganic & medicinal chemistry letters (15.09.2017)
Published in Bioorganic & medicinal chemistry letters (15.09.2017)
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Journal Article
Multi-modal antidepressant-like action of 6- and 7-chloro-2-aminodihydroquinazolines in the mouse tail suspension test
Iyer, Kavita A., Alix, Katie, Eltit, Jose M., Solis, Ernesto, Pan, Xiaolei, Argade, Malaika D., Khatri, Shailesh, De Felice, Louis J., Sweet, Douglas H., Schulte, Marvin K., Dukat, Małgorzata
Published in Psychopharmacology (01.07.2019)
Published in Psychopharmacology (01.07.2019)
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Journal Article
X-ray crystal structure of a 2-amino-3,4-dihydroquinazoline 5-HT3 serotonin receptor antagonist and related analogs
Abdelkhalek, Ahmed S., Musayev, Faik N., Iyer, Kavita A., Hemanth, Prithvi, Safo, Martin K., Dukat, Małgorzata
Published in Journal of molecular structure (15.02.2020)
Published in Journal of molecular structure (15.02.2020)
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Journal Article
Superagonist, Full Agonist, Partial Agonist, and Antagonist Actions of Arylguanidines at 5‑Hydroxytryptamine‑3 (5-HT3) Subunit A Receptors
Alix, Katie, Khatri, Shailesh, Mosier, Philip D, Casterlow, Samantha, Yan, Dong, Nyce, Heather L, White, Michael M, Schulte, Marvin K, Dukat, Małgorzata
Published in ACS chemical neuroscience (16.11.2016)
Published in ACS chemical neuroscience (16.11.2016)
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Journal Article
Revised Pharmacophore Model for 5‑HT2A Receptor Antagonists Derived from the Atypical Antipsychotic Agent Risperidone
Shah, Urjita H, Gaitonde, Supriya A, Moreno, José L, Glennon, Richard A, Dukat, Małgorzata, González-Maeso, Javier
Published in ACS chemical neuroscience (15.05.2019)
Published in ACS chemical neuroscience (15.05.2019)
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Journal Article
Toward selective drug development for the human 5-hydroxytryptamine 1E receptor: a comparison of 5-hydroxytryptamine 1E and 1F receptor structure-affinity relationships
Klein, Michael T, Dukat, Małgorzata, Glennon, Richard A, Teitler, Milt
Published in The Journal of pharmacology and experimental therapeutics (01.06.2011)
Published in The Journal of pharmacology and experimental therapeutics (01.06.2011)
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Journal Article
The medicinal chemistry of 5-HT6 receptor ligands with a focus on arylsulfonyltryptamine analogs
Glennon, Richard A, Siripurapu, Uma, Roth, Bryan L, Kolanos, Renata, Bondarev, Mikhail L, Sikazwe, Donald, Lee, Mase, Dukat, Małgorzata
Published in Current topics in medicinal chemistry (01.04.2010)
Published in Current topics in medicinal chemistry (01.04.2010)
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Journal Article
“Methylene Bridge” to 5‑HT3 Receptor Antagonists: Conformationally Constrained Phenylguanidines
Abdelkhalek, Ahmed S, Alley, Genevieve S, Alwassil, Osama I, Khatri, Shailesh, Mosier, Philip D, Nyce, Heather L, White, Michael M, Schulte, Marvin K, Dukat, Małgorzata
Published in ACS chemical neuroscience (20.03.2019)
Published in ACS chemical neuroscience (20.03.2019)
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Journal Article
α4β2 nACh Receptor pharmacophore models
Glennon, Richard A, Dukat, Małgorzata
Published in Bioorganic & medicinal chemistry letters (19.04.2004)
Published in Bioorganic & medicinal chemistry letters (19.04.2004)
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Journal Article