oligosaccharide-based HIV-1 2G12 mimotope vaccine induces carbohydrate-specific antibodies that fail to neutralize HIV-1 virions
Joyce, Joseph G, Krauss, Isaac J, Song, Hong C, Opalka, David W, Grimm, Karen M, Nahas, Deborah D, Esser, Mark T, Hrin, Renee, Feng, Meizhen, Dudkin, Vadim Y, Chastain, Michael, Shiver, John W, Danishefsky, Samuel J
Published in Proceedings of the National Academy of Sciences - PNAS (14.10.2008)
Published in Proceedings of the National Academy of Sciences - PNAS (14.10.2008)
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Journal Article
Fully Synthetic Carbohydrate HIV Antigens Designed on the Logic of the 2G12 Antibody
Krauss, Isaac J, Joyce, Joseph G, Finnefrock, Adam C, Song, Hong C, Dudkin, Vadim Y, Geng, Xudong, Warren, J. David, Chastain, Michael, Shiver, John W, Danishefsky, Samuel J
Published in Journal of the American Chemical Society (12.09.2007)
Published in Journal of the American Chemical Society (12.09.2007)
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Journal Article
In Pursuit of Carbohydrate-Based HIV Vaccines, Part 2: The Total Synthesis of High-Mannose-Type gp120 Fragments-Evaluation of Strategies Directed to Maximal Convergence
Geng, Xudong, Dudkin, Vadim Y., Mandal, Mihirbaran, Danishefsky, Samuel J.
Published in Angewandte Chemie (International ed.) (03.05.2004)
Published in Angewandte Chemie (International ed.) (03.05.2004)
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Journal Article
Chemical Synthesis of Normal and Transformed PSA Glycopeptides
Dudkin, Vadim Y, Miller, Justin S, Danishefsky, Samuel J
Published in Journal of the American Chemical Society (28.01.2004)
Published in Journal of the American Chemical Society (28.01.2004)
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Journal Article
Toward a Prostate Specific Antigen-Based Prostate Cancer Diagnostic Assay: Preparation of Keyhole Limpet Hemocyanin -Conjugated Normal and Transformed Prostate Specific Antigen Fragments
Dudkin, Vadim Y, Miller, Justin S, Dudkina, Anna S, Antczak, Christophe, Scheinberg, David A, Danishefsky, Samuel J
Published in Journal of the American Chemical Society (15.10.2008)
Published in Journal of the American Chemical Society (15.10.2008)
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Journal Article
Toward Fully Synthetic N-Linked Glycoproteins
Miller, Justin S., Dudkin, Vadim Y., Lyon, Gholson J., Muir, Tom W., Danishefsky, Samuel J.
Published in Angewandte Chemie (International ed.) (27.01.2003)
Published in Angewandte Chemie (International ed.) (27.01.2003)
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Journal Article
Optimization of a pyrazoloquinolinone class of Chk1 kinase inhibitors
Brnardic, Edward J., Garbaccio, Robert M., Fraley, Mark E., Tasber, Edward S., Steen, Justin T., Arrington, Kenneth L., Dudkin, Vadim Y., Hartman, George D., Stirdivant, Steven M., Drakas, Bob A., Rickert, Keith, Walsh, Eileen S., Hamilton, Kelly, Buser, Carolyn A., Hardwick, James, Tao, Weikang, Beck, Stephen C., Mao, Xianzhi, Lobell, Robert B., Sepp-Lorenzino, Laura, Yan, Youwei, Ikuta, Mari, Munshi, Sanjeev K., Kuo, Lawrence C., Kreatsoulas, Constantine
Published in Bioorganic & medicinal chemistry letters (01.11.2007)
Published in Bioorganic & medicinal chemistry letters (01.11.2007)
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Journal Article
Evaluation of a Centyrin-Based Near-Infrared Probe for Fluorescence-Guided Surgery of Epidermal Growth Factor Receptor Positive Tumors
Mahalingam, Sakkarapalayam M, Dudkin, Vadim Y, Goldberg, Shalom, Klein, Donna, Yi, Fang, Singhal, Sunil, O’Neil, Karyn T, Low, Philip S
Published in Bioconjugate chemistry (15.11.2017)
Published in Bioconjugate chemistry (15.11.2017)
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Journal Article
Pyridyl aminothiazoles as potent inhibitors of Chk1 with slow dissociation rates
Dudkin, Vadim Y., Rickert, Keith, Kreatsoulas, Constantine, Wang, Cheng, Arrington, Kenneth L., Fraley, Mark E., Hartman, George D., Yan, Yowei, Ikuta, Mari, Stirdivant, Steven M., Drakas, Robert A., Walsh, Eileen S., Hamilton, Kelly, Buser, Carolyn A., Lobell, Robert B., Sepp-Lorenzino, Laura
Published in Bioorganic & medicinal chemistry letters (01.04.2012)
Published in Bioorganic & medicinal chemistry letters (01.04.2012)
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Journal Article
Toward Fully Synthetic Carbohydrate-Based HIV Antigen Design: On the Critical Role of Bivalency
Dudkin, Vadim Y, Orlova, Marianna, Geng, Xudong, Mandal, Mihirbaran, Olson, William C, Danishefsky, Samuel J
Published in Journal of the American Chemical Society (11.08.2004)
Published in Journal of the American Chemical Society (11.08.2004)
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Journal Article
마크로사이클릭 화합물 및 이의 사용 방법
SONG FENGBIN, SALTER RHYS, DUDKIN VADIM Y, ZHANG WEI, GOLDBERG SHALOM, KEITH JOHN
Year of Publication 13.07.2023
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Year of Publication 13.07.2023
Patent
Pyridyl aminothiazoles as potent Chk1 inhibitors: Optimization of cellular activity
Dudkin, Vadim Y., Wang, Cheng, Arrington, Kenneth L., Fraley, Mark E., Hartman, George D., Stirdivant, Steven M., Drakas, Robert A., Rickert, Keith, Walsh, Eileen S., Hamilton, Kelly, Buser, Carolyn A., Hardwick, James, Tao, Weikang, Beck, Stephen C., Mao, Xianzhi, Lobell, Robert B., Sepp-Lorenzino, Laura
Published in Bioorganic & medicinal chemistry letters (01.04.2012)
Published in Bioorganic & medicinal chemistry letters (01.04.2012)
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Journal Article
Small Molecule Mimetics of an HIV-1 gp41 Fusion Intermediate as Vaccine Leads
Caulfield, Michael J., Dudkin, Vadim Y., Ottinger, Elizabeth A., Getty, Krista L., Zuck, Paul D., Kaufhold, Robin M., Hepler, Robert W., McGaughey, Georgia B., Citron, Michael, Hrin, Renee C., Wang, Ying-Jie, Miller, Michael D., Joyce, Joseph G.
Published in The Journal of biological chemistry (24.12.2010)
Published in The Journal of biological chemistry (24.12.2010)
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Journal Article
A concise route to the core pentasaccharide of N-linked glycoproteins
Dudkin, Vadim Y., Miller, Justin S., Danishefsky, Samuel J.
Published in Tetrahedron letters (24.02.2003)
Published in Tetrahedron letters (24.02.2003)
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Journal Article
A highly convergent synthesis of an N-linked glycopeptide presenting the H-type 2 human blood group determinant
Wang, Zhi-Guang, Warren, J. David, Dudkin, Vadim Y., Zhang, Xufang, Iserloh, Ulrich, Visser, Michael, Eckhardt, Matthias, Seeberger, Peter H., Danishefsky, Samuel J.
Published in Tetrahedron (15.05.2006)
Published in Tetrahedron (15.05.2006)
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Journal Article
Pyridyi aminothiazoles as potent inhibitors of Chk1 with slow dissociation rates
DUDKIN, Vadim Y, RICKERT, Keith, DRAKAS, Robert A, WALSH, Eileen S, HAMILTON, Kelly, BUSER, Carolyn A, LOBELL, Robert B, SEPP-LORENZINO, Laura, KREATSOULAS, Constantine, CHENG WANG, ARRINGTON, Kenneth L, FRALEY, Mark E, HARTMAN, George D, YOWEI YAN, IKUTA, Mari, STIRDIVANT, Steven M
Published in Bioorganic & medicinal chemistry letters (2012)
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Published in Bioorganic & medicinal chemistry letters (2012)
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