Reversible biotinylated oligosaccharides: a new approach for a better management of anticoagulant therapy
SAVI, P., HERAULT, J. P., DUCHAUSSOY, P., MILLET, L., SCHAEFFER, P., PETITOU, M., BONO, F., HERBERT, J. M.
Published in Journal of thrombosis and haemostasis (01.10.2008)
Published in Journal of thrombosis and haemostasis (01.10.2008)
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Reversible biotinylated oligosaccharides: a new approach for a better management of anticoagulant therapy
SAVI, P., HERAULT, J.P., DUCHAUSSOY, P., MILLET, L., SCHAEFFER, P., PETITOU, M., BONO, F., HERBERT, J.M.
Published in Journal of thrombosis and haemostasis (01.10.2008)
Published in Journal of thrombosis and haemostasis (01.10.2008)
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The structure of synthetic oligosaccharides in relation to factor IXa inhibition
Hérault, J P, Gaich, C, Bono, F, Driguez, P A, Duchaussoy, P, Petitou, M, Herbert, J M
Published in Thrombosis and haemostasis (01.09.2002)
Published in Thrombosis and haemostasis (01.09.2002)
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Experimental Proof for the Structure of a Thrombin-Inhibiting Heparin Molecule
Petitou, Maurice, Imberty, Anne, Duchaussoy, Philippe, Driguez, Pierre-Alexandre, Ceccato, Marie-Line, Gourvenec, Françoise, Sizun, Philippe, Hérault, Jean-Pascal, Pérez, Serge, Herbert, Jean-Marc
Published in Chemistry : a European journal (16.02.2001)
Published in Chemistry : a European journal (16.02.2001)
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Comparative effects of two synthetic oligosaccharides on platelet activation induced by plasma from HIT patients
Savi, P., Pflieger, A‐M., Hérault, J‐P., Michaux, C., Duchaussoy, P., Petitou, M., Herbert, J‐M.
Published in Journal of thrombosis and haemostasis (01.09.2003)
Published in Journal of thrombosis and haemostasis (01.09.2003)
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Synthesis of conformationally locked L-iduronic acid derivatives: Direct evidence for a critical role of the skew-boat S-2(0) conformer in the activation of antithrombin by heparin
Das, SK, Mallet, JM, Esnault, J, Driguez, PA, Duchaussoy, P, Sizun, P, Herault, JP, Herbert, JM, Petitou, M, Sinay, P
Published in Chemistry : a European journal (19.11.2001)
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Published in Chemistry : a European journal (19.11.2001)
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Synthesis of conformationally locked carbohydrates: A skew-boat conformation of L-iduronic acid governs the antithrombotic activity of heparin
Das, SK, Mallet, JM, Esnault, J, Driguez, PA, Duchaussoy, P, Sizun, P, Herault, JP, Herbert, JM, Petitou, M, Sinay, P
Published in Angewandte Chemie International Edition (01.01.2001)
Published in Angewandte Chemie International Edition (01.01.2001)
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The synthetic pentasaccharide fondaparinux: first in the class of antithrombotic agents that selectively inhibit coagulation factor Xa
Petitou, Maurice, Duchaussoy, Philippe, Herbert, Jean-Marc, Duc, Gérald, El Hajji, Mohamed, Branellec, Jean-François, Donat, François, Necciari, José, Cariou, Roger, Bouthier, Jean, Garrigou, Eric
Published in Seminars in thrombosis and hemostasis (01.08.2002)
Published in Seminars in thrombosis and hemostasis (01.08.2002)
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SR123781A, a synthetic heparin mimetic
Herbert, J M, Hérault, J P, Bernat, A, Savi, P, Schaeffer, P, Driguez, P A, Duchaussoy, P, Petitou, M
Published in Thrombosis and haemostasis (01.05.2001)
Published in Thrombosis and haemostasis (01.05.2001)
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First Synthetic Carbohydrates with the Full Anticoagulant Properties of Heparin
Petitou, Maurice, Duchaussoy, Philippe, Driguez, Pierre-A., Jaurand, Guy, Hérault, Jean-P., Lormeau, Jean-C., van Boeckel, Constant A. A., Herbert, Jean-M.
Published in Angewandte Chemie (International ed.) (16.11.1998)
Published in Angewandte Chemie (International ed.) (16.11.1998)
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A synthetic heparan sulfate pentasaccharide, exclusively containing L-iduronic acid, displays higher affinity for FGF-2 than its D-glucuronic acid-containing isomers
KOVENSKY, J, DUCHAUSSOY, P, BONO, F, SALMIVIRTA, M, SIZUN, P, HERBERT, J.-M, PETITOU, M, SINAY, P
Published in Bioorganic & medicinal chemistry (01.08.1999)
Published in Bioorganic & medicinal chemistry (01.08.1999)
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Synthesis and Pharmacological Properties of a Close Analogue of an Antithrombotic Pentasaccharide (SR 90107A/ORG 31540)
Petitou, Maurice, Duchaussoy, Philippe, Jaurand, Guy, Gourvenec, Françoise, Lederman, Isidore, Strassel, Jean-Marc, Bârzu, Tereza, Crépon, Bertrand, Hérault, Jean-Pascal, Lormeau, Jean-Claude, Bernat, André, Herbert, Jean-Marc
Published in Journal of medicinal chemistry (23.05.1997)
Published in Journal of medicinal chemistry (23.05.1997)
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Design and synthesis of heparin mimetics able to inhibit thrombin. Part 1 - Identification of a hexasaccharide sequence able to inhibit thrombin and suitable for 'polymerisation'
Duchaussoy, P, Jaurand, G, Driguez, PA, Lederman, Gourvenec, F, Strassel, JM, Sizun, P, Petitou, M, Herbert, JM
Published in Carbohydrate research (30.04.1999)
Published in Carbohydrate research (30.04.1999)
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l-Iduronic acid derivatives as glycosyl donors
Tabeur, Christine, Machetto, Françoise, Mallet, Jean-Maurice, Duchaussoy, Philippe, Petitou, Maurice, Sinaÿ, Pierre
Published in Carbohydrate research (23.02.1996)
Published in Carbohydrate research (23.02.1996)
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Synthetic oligosaccharides having various functional domains: Potent and potentially safe heparin mimetics
Petitou, Maurice, Driguez, Pierre-Alexandre, Duchaussoy, Philippe, Hérault, Jean-Pascal, Lormeau, Jean-Claude, Herbert, Jean-Marc
Published in Bioorganic & medicinal chemistry letters (19.04.1999)
Published in Bioorganic & medicinal chemistry letters (19.04.1999)
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