RP 73870, a gastrin/cholecystokinin-B receptor antagonist with potent anti-ulcer activity in the rat
Pendley, C E, Fitzpatrick, L R, Capolino, A J, Davis, M A, Esterline, N J, Jakubowska, A, Bertrand, P, Guyon, C, Dubroeucq, M C, Martin, G E
Published in The Journal of pharmacology and experimental therapeutics (01.06.1995)
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Published in The Journal of pharmacology and experimental therapeutics (01.06.1995)
Journal Article
PK 11195, an antagonist of peripheral benzodiazepine receptors, reduces ventricular arrhythmias during myocardial ischemia and reperfusion in the dog
Mestre, M, Bouetard, G, Uzan, A, Gueremy, C, Renault, C, Dubroeucq, M C, Le Fur, G
Published in European journal of pharmacology (07.06.1985)
Published in European journal of pharmacology (07.06.1985)
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Journal Article
Modulation of voltage-operated, but not receptor-operated, calcium channels in the rabbit aorta by PK 11195, an antagonist of peripheral-type benzodiazepine receptors
Mestre, M, Belin, C, Uzan, A, Renault, C, Dubroeucq, M C, Gueremy, C, Le Fur, G
Published in Journal of cardiovascular pharmacology (01.07.1986)
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Published in Journal of cardiovascular pharmacology (01.07.1986)
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In vivo labelling in several rat tissues of 'peripheral type' benzodiazepine binding sites
Benavides, J, Guilloux, F, Rufat, P, Uzan, A, Renault, C, Dubroeucq, M C, Gueremy, C, Le Fur, G
Published in European journal of pharmacology (16.03.1984)
Published in European journal of pharmacology (16.03.1984)
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Journal Article
Labelling of "peripheral-type" benzodiazepine binding sites in the rat brain by using [3H]PK 11195, an isoquinoline carboxamide derivative: kinetic studies and autoradiographic localization
Benavides, J, Quarteronet, D, Imbault, F, Malgouris, C, Uzan, A, Renault, C, Dubroeucq, M C, Gueremy, C, Le Fur, G
Published in Journal of neurochemistry (01.12.1983)
Published in Journal of neurochemistry (01.12.1983)
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Journal Article
Peripheral benzodiazepine binding sites: effect of PK 11195, 1-(2-chlorophenyl)-N-methyl-N-(1-methylpropyl)-3-isoquinolinecarboxamide. I. In vitro studies
Le Fur, G, Perrier, M L, Vaucher, N, Imbault, F, Flamier, A, Benavides, J, Uzan, A, Renault, C, Dubroeucq, M C, Guérémy, C
Published in Life sciences (1973) (18.04.1983)
Published in Life sciences (1973) (18.04.1983)
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Journal Article
Photoaffinity labeling of peripheral-type benzodiazepine-binding sites
DOBLE, A, FERRIS, O, BURGEVIN, M. C, MENAGER, J, UZAN, A, DUBRŒUCQ, M. C, RENAULT, C, GUEREMY, C, LE FUR, G
Published in Molecular pharmacology (01.01.1987)
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Published in Molecular pharmacology (01.01.1987)
Journal Article
Electrophysiological and pharmacological evidence that peripheral type benzodiazepine receptors are coupled to calcium channels in the heart
Mestre, M, Carriot, T, Belin, C, Uzan, A, Renault, C, Dubroeucq, M C, Guérémy, C, Doble, A, Le Fur, G
Published in Life sciences (1973) (01.01.1985)
Published in Life sciences (1973) (01.01.1985)
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Journal Article
Peripheral benzodiazepine binding sites: effect of PK 11195, 1-(2-chlorophenyl)-N-methyl-(1-methylpropyl)-3 isoquinolinecarboxamide. II. In vivo studies
Le Fur, G, Guilloux, F, Rufat, P, Benavides, J, Uzan, A, Renault, C, Dubroeucq, M C, Guérémy, C
Published in Life sciences (1973) (18.04.1983)
Published in Life sciences (1973) (18.04.1983)
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Journal Article
Electrophysiological and pharmacological characterization of peripheral benzodiazepine receptors in a guinea pig heart preparation
Mestre, M, Carriot, T, Belin, C, Uzan, A, Renault, C, Dubroeucq, M C, Guérémy, C, Le Fur, G
Published in Life sciences (1973) (27.08.1984)
Published in Life sciences (1973) (27.08.1984)
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Journal Article
The ureidoacetamides, a novel family of non-peptide CCK-B/gastrin antagonists
Böhme, G A, Bertrand, P, Guyon, C, Capet, M, Pendley, C, Stutzmann, J M, Doble, A, Dubroeucq, M C, Martin, G, Blanchard, J C
Published in Annals of the New York Academy of Sciences (01.03.1994)
Published in Annals of the New York Academy of Sciences (01.03.1994)
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Journal Article
Pharmacological evidence that PK 8165 behaves as a partial agonist of brain type benzodiazepine receptors
Mizoule, J, Rataud, J, Uzan, A, Mazadier, M, Daniel, M, Gauthier, A, Ollat, C, Gueremy, C, Renault, C, Dubroeucq, M C
Published in Archives internationales de pharmacodynamie et de thérapie (01.01.1984)
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Published in Archives internationales de pharmacodynamie et de thérapie (01.01.1984)
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Synthesis and pharmacological properties of 5H,10H-imidazo[1,2-a]indeno[1,2-e]pyrazine-4-one, a new competitive AMPA/KA receptor antagonist
Mignani, Serge, Aloup, Jean-Claude, Barreau, Michel, Blanchard, Jean Charles, Böhme, Georg Andrees, Boireau, Alain, Damour, Dominique, Debono, Marc-Williams, Dubroeucq, Marie-Christine, Genevois-Borella, Arielle, Imperato, Assunta, Jimonet, Patrick, Pratt, Jeremy, Randle, John C.R., Reibaud, Michel, Ribeill, Yves, Stutzmann, Jean-Marie
Published in Drug development research (01.11.1999)
Published in Drug development research (01.11.1999)
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Journal Article
Opposite effects of two ligands for peripheral type benzodiazepine binding sites, PK 11195 and RO5-4864, in a conflict situation in the rat
Mizoule, J, Gauthier, A, Uzan, A, Renault, C, Dubroeucq, M C, Guérémy, C, Le Fur, G
Published in Life sciences (1973) (18.03.1985)
Published in Life sciences (1973) (18.03.1985)
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Journal Article
"Peripheral type" benzodiazepine binding sites in rat adrenals: binding studies with [3H]PK 11195 and autoradiographic localization
Benavides, J, Malgouris, C, Imbault, F, Begassat, F, Uzan, A, Renault, C, Dubroeucq, M C, Gueremy, C, Le Fur, G
Published in Archives internationales de pharmacodynamie et de thérapie (01.11.1983)
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Published in Archives internationales de pharmacodynamie et de thérapie (01.11.1983)
Journal Article
Opposite effects of an agonist, RO5-4864, and an antagonist, PK 11195, of the peripheral type benzodiazepine binding sites on audiogenic seizures in DBA/2J mice
Bénavidès, J, Guilloux, F, Allam, D E, Uzan, A, Mizoule, J, Renault, C, Dubroeucq, M C, Guérémy, C, Le Fur, G
Published in Life sciences (1973) (25.06.1984)
Published in Life sciences (1973) (25.06.1984)
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Journal Article
Autoradiographic localization of peripheral benzodiazepine binding sites in the cat brain with [3H]PK 11195
Bénavidès, J, Savaki, H E, Malgouris, C, Laplace, C, Daniel, M, Begassat, F, Desban, M, Uzan, A, Dubroeucq, M C, Renault, C
Published in Brain research bulletin (01.07.1984)
Published in Brain research bulletin (01.07.1984)
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Journal Article
Evaluation of brain penetration of CCK-B antagonists
Dubroeucq, M C, Guyon, C, Manfré, F, Capet, M, Barreau, M, Bertrand, P, Jeantaud, B, Doble, A, Blanchard, J C
Published in Annals of the New York Academy of Sciences (01.03.1994)
Published in Annals of the New York Academy of Sciences (01.03.1994)
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Journal Article
PK 11195, an antagonist of peripheral type benzodiazepine receptors, modulates Bay K8644 sensitive but not beta- or H2-receptor sensitive voltage operated calcium channels in the guinea pig heart
Mestre, M, Carriot, T, Néliat, G, Uzan, A, Renault, C, Dubroeucq, M C, Guérémy, C, Doble, A, Le Fur, G
Published in Life sciences (1973) (28.07.1986)
Published in Life sciences (1973) (28.07.1986)
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