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Comparative metabolite profiling and identification of GalNAc-conjugated siRNA, siRNA01, in plasma prepared with various anticoagulants, serum, and in vivo plasma using LC-UV-HRMS
Zhang, Hong, Chen, Tianhong, Wang, Junjie, Shi, Liqi, Qin, Gengyao, Cao, Weiqun, Tao, Yi, Shen, Liang
Published in Drug metabolism and pharmacokinetics (01.06.2025)
Published in Drug metabolism and pharmacokinetics (01.06.2025)
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Chida, Katsuyuki, Ishikawa, Tetsuo, Hanai, Akiko, Hananoe, Ayaka, Kashiwagi, Yusuke, Hatakeyama, Hiroto, Kawakami, Eiryo
Published in Drug metabolism and pharmacokinetics (01.06.2025)
Published in Drug metabolism and pharmacokinetics (01.06.2025)
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Characterization of human immortalized cell-based blood-brain barrier spheroid models as a tool for brain vascular inflammation studies
Morio, Hanae, Ebisawa, Ayuka, Kunitomo, Furano, Minasato, Asuka, Furihata, Tomomi
Published in Drug metabolism and pharmacokinetics (01.06.2025)
Published in Drug metabolism and pharmacokinetics (01.06.2025)
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Analytical validation of a genotyping technique for a single-nucleotide polymorphism to predict of the onset SJS/TEN in Japanese
Tsukagoshi, Eri, Nakamura, Ryosuke, Tanaka, Yoichi, Maekawa, Keiko, Hiratsuka, Masahiro, Asada, Hideo, Saito, Yoshiro, Kikura-Hanajiri, Ruri
Published in Drug metabolism and pharmacokinetics (01.06.2025)
Published in Drug metabolism and pharmacokinetics (01.06.2025)
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Assessment of in vitro methods for UGT1A1 inhibition in recombinant isozyme
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Published in Drug metabolism and pharmacokinetics (01.06.2025)
Published in Drug metabolism and pharmacokinetics (01.06.2025)
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Human aldo-keto reductase (AKR) 1C1 and 1C2 act as coactivators of pregnane X receptor, a master regulator of drug-metabolizing and gluconeogenesis enzymes
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Published in Drug metabolism and pharmacokinetics (01.06.2025)
Published in Drug metabolism and pharmacokinetics (01.06.2025)
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Primary culture of rat kidney tissue slice for evaluation of drug-induced kidney injury using gas-permeable plates
Kadoguchi, Moeno, Esashika, Katsuhiro, Matsushita, Kohei, Yang, Jingjing, Takahashi, Jun, Tamai, Ikumi, Arakawa, Hiroshi
Published in Drug metabolism and pharmacokinetics (01.06.2025)
Published in Drug metabolism and pharmacokinetics (01.06.2025)
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Monkey CYP2C8-mediated formation of rearranged metabolites of the selective Nav1.7 inhibitor DS-1971a
Michiba, Kazuyoshi, Asano, Daigo, Shiozawa, Hideyuki, Masuda, Kayoko, Arai, Atsushi, Takakusa, Hideo, Nakai, Daisuke
Published in Drug metabolism and pharmacokinetics (01.06.2025)
Published in Drug metabolism and pharmacokinetics (01.06.2025)
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Solanidine metabolites as dietary CYP2D6 biomarkers of tamoxifen metabolism
Medwid, Samantha, Schwarz, Ute I., Keller, Denise, Ross, Cameron, Kim, Richard B.
Published in Drug metabolism and pharmacokinetics (01.06.2025)
Published in Drug metabolism and pharmacokinetics (01.06.2025)
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Comphrehensive metabolite profiling of SHO0302 in human plasma, urine and feces using LC-HRMS and an advanced data processing workflow: Comparison with radiochromatographic analysis
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Published in Drug metabolism and pharmacokinetics (01.06.2025)
Published in Drug metabolism and pharmacokinetics (01.06.2025)
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Functional characteristics of equilibrative nucleoside transporter 2 (ENT2/SLC29A2) for the transport of urate as a newly identified substrate
Matake, Isamu, Yasujima, Tomoya, Matsuo, Hirotaka, Toyoda, Yu, Kawamura, Yusuke, Takada, Tappei, Inoue, Katsuhisa, Yamashiro, Takahiro, Yuasa, Hiroaki
Published in Drug metabolism and pharmacokinetics (01.06.2025)
Published in Drug metabolism and pharmacokinetics (01.06.2025)
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Model-based exploration of parent-metabolite kinetics of MT-202: Nonclinical characterization and feasibility of clinical metabolite exposure prediction
Sun, Austin, Smukste, Inese, Dowling, James E., McTeague, T. Andrew, Yan, Liping, Zhou, Xiaoying, Bursavich, Matthew G., Lippa, Blaise, Tang, Cuyue
Published in Drug metabolism and pharmacokinetics (01.06.2025)
Published in Drug metabolism and pharmacokinetics (01.06.2025)
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