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Primary human intestinal cell model for estimating drug absorption, efflux and metabolism
Cheong, Jonathan, Jorski, Jamie, Chhin, Christopher, Ayehunie, Seyoum, Stevens, Zachary, Olda, Jon, Salphati, Laurent
Published in Drug metabolism and pharmacokinetics (01.06.2025)
Published in Drug metabolism and pharmacokinetics (01.06.2025)
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Identification of physiological factors suppressing colonic drug absorption using quantum imaging technology
Yasugi, Yugo, Hirosaki, Maho, Hotta, Kazuki, Kato, Yumi, Ueda, Yasuyuki, Iwatake, Mayumi, Yukawa, Hiroshi, Tamai, Ikumi, Shirasaka, Yoshiyuki
Published in Drug metabolism and pharmacokinetics (01.06.2025)
Published in Drug metabolism and pharmacokinetics (01.06.2025)
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Metabolism of pirocarpine in chimeric mice with humanized liver
Uehara, Shotaro, Higuchi, Yuichiro, Yoneda, Nao, Yamazaki, Hiroshi, Suemizu, Hiroshi
Published in Drug metabolism and pharmacokinetics (01.06.2025)
Published in Drug metabolism and pharmacokinetics (01.06.2025)
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CYP Induction assays using 10-Donor pooled human hepatocytes
Li, Feng, Nahrin, Adeeba, Parikh, Sweta, Bourgea, Joanne, Cooper, Kirsten, Desmond, Bryan, Clark, Robert, Li, Albert P.
Published in Drug metabolism and pharmacokinetics (01.06.2025)
Published in Drug metabolism and pharmacokinetics (01.06.2025)
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A simple approach for facile determination of metabolic softspots of macrocyclic peptides based on metabolite genealogy information revealed in the metabolite profiles
Zhang, Haiying, Lyu, Zhigang, Cannon, Joe R.
Published in Drug metabolism and pharmacokinetics (01.06.2025)
Published in Drug metabolism and pharmacokinetics (01.06.2025)
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Mechanistic studies supporting the evaluation of pharmacokinetic-drug interactions with drugs approved by the U.S. food and drug administration in 2023: A systematic review of new drug applications
Yu, Jingjing, Argon, Sophie, Wang, Yan, Ragueneau-Majlessi, Isabelle
Published in Drug metabolism and pharmacokinetics (01.06.2025)
Published in Drug metabolism and pharmacokinetics (01.06.2025)
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Evaluation of aldehyde-odorant metabolisms and AOX and ALDH expression profiles in human nasal mucosa and mucus
Takaoka, Naoki, Sanoh, Seigo, Kurosaki, Mami, Terao, Mineko, Garattini, Enrico, Sakatani, Hideki, Murakami, Daichi, Kono, Masamitsu, Hotomi, Muneki, Ohta, Shigeru
Published in Drug metabolism and pharmacokinetics (01.06.2025)
Published in Drug metabolism and pharmacokinetics (01.06.2025)
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Development of dissolution evaluation system for drug absorption (V): Additional intestinal absorption module of in vitro 3D gastric emptying mmodel for orally disintegrating tablet
Tagawa, Kozo, Kiriyama, Akiko, Lin, San Yuet, Fukunaga, Sota
Published in Drug metabolism and pharmacokinetics (01.06.2025)
Published in Drug metabolism and pharmacokinetics (01.06.2025)
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A combined quantitative and qualitative DMPK assay using pooled samples for increased throughput in macrocylic peptide drug development
Hackbusch, Sven, Morin, Sebastien, Cancilla, Mark, O'Callaghan, Lisa, Sun, Congliang, Habulihaz, Bahanu, Spellman, Daniel
Published in Drug metabolism and pharmacokinetics (01.06.2025)
Published in Drug metabolism and pharmacokinetics (01.06.2025)
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Comparative pharmacokinetics of andrographolide after repeated oral administration of andrographis paniculata formulation capsules in Beagles
Boonyarattanasoonthorn, Tussapon, Junsai, Thammaporn, Kongratanapasert, Teetat, Supannapan, Kittitach, Khemawoot, Phisit
Published in Drug metabolism and pharmacokinetics (01.06.2025)
Published in Drug metabolism and pharmacokinetics (01.06.2025)
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Investigation of pharmacokinetic properties and brain penetration of genipin: A potential pharmacophore for Parkinson's disease treatment
Cho, Hyunjin, Lee, Jeongmin, Hwang, Sangsoo, Park, Seojin, Lim, Jeonghyun, Lee, Juwon, Jang, Hyesu, Lee, Seokwoo, Moon, Minho, Shin, Young G.
Published in Drug metabolism and pharmacokinetics (01.06.2025)
Published in Drug metabolism and pharmacokinetics (01.06.2025)
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Identification of pazopanib as an OATP1B1 substrate by competitive counterflow screeen
Huang, Kevin, Drabison, Thomas, Boeckman, Mike, Sparreboom, Alex, Hu, Shuiying
Published in Drug metabolism and pharmacokinetics (01.06.2025)
Published in Drug metabolism and pharmacokinetics (01.06.2025)
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Development of a PAC-LC-MS/MS method for simultaneous quantification of mipomersen, its metabolites, and analogues in tissue samples
Sun, Yuchen, Nitta, Shin-ichiro, Aikawa, Hiroaki, Saito, Tomoko, Tsutomu, Yonemasu, Goda, Ryoya, Kakehi, Masaaki, Hayashi, Yoshiharu, Ito, Satoshi, Kawahara, Tsuyoshi, Masui, Naoto, Inoue, Kazuko, Shimbo, Kazutaka, Yamaguchi, Takeru, Jinno, Fumihiro, Murakoshi, Kaori, Takahara, Kentaro, Murata, Chie, Uchiyama, Hitoshi, Kawabata, Mitsuhiko, Saito, Kosuke, Kikura-Hanajiri, Rui, Saito, Yoshiro
Published in Drug metabolism and pharmacokinetics (01.06.2025)
Published in Drug metabolism and pharmacokinetics (01.06.2025)
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Drug-drug interaction between trastuzumab emtansine (T-DM1) and orally administered tacrolimus in a patient and in rats
Nakamura, Tomohiro, Shimada, Moeko, Takabayashi, Makiko, Fujita, Arimi, Kawakami, Takahiro, Maruyama, Hiroyuki, Terakawa, Hirofumi, Ishimoto, Takahiro, Shimada, Tsutomu, Miyamoto, Toshihiro, Sai, Yoshimichi
Published in Drug metabolism and pharmacokinetics (01.06.2025)
Published in Drug metabolism and pharmacokinetics (01.06.2025)
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Investigation in the predictive accuracy of brain KPUU across species using in vitro and in vivo methods
Zou, Ling, Chien, Huan-Chieh, Nguyen, Khoi, Pade, Devendra, Li, Yanfei, Enogieru, Jessica, Wahlstrom, Jan
Published in Drug metabolism and pharmacokinetics (01.06.2025)
Published in Drug metabolism and pharmacokinetics (01.06.2025)
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