MDM2-Recruiting PROTAC Offers Superior, Synergistic Antiproliferative Activity via Simultaneous Degradation of BRD4 and Stabilization of p53
Hines, John, Lartigue, Schan, Dong, Hanqing, Qian, Yimin, Crews, Craig M
Published in Cancer research (Chicago, Ill.) (01.01.2019)
Published in Cancer research (Chicago, Ill.) (01.01.2019)
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PROTAC-induced BET protein degradation as a therapy for castration-resistant prostate cancer
Raina, Kanak, Lu, Jing, Qian, Yimin, Altieri, Martha, Gordon, Deborah, Rossi, Ann Marie K., Wang, Jing, Chen, Xin, Dong, Hanqing, Siu, Kam, Winkler, James D., Crew, Andrew P., Crews, Craig M., Coleman, Kevin G.
Published in Proceedings of the National Academy of Sciences - PNAS (28.06.2016)
Published in Proceedings of the National Academy of Sciences - PNAS (28.06.2016)
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Androgen receptor degradation by the proteolysis-targeting chimera ARCC-4 outperforms enzalutamide in cellular models of prostate cancer drug resistance
Salami, Jemilat, Alabi, Shanique, Willard, Ryan R, Vitale, Nick J, Wang, Jing, Dong, Hanqing, Jin, Meizhong, McDonnell, Donald P, Crew, Andrew P, Neklesa, Taavi K, Crews, Craig M
Published in Communications biology (01.01.2018)
Published in Communications biology (01.01.2018)
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Identification and Characterization of Von Hippel-Lindau-Recruiting Proteolysis Targeting Chimeras (PROTACs) of TANK-Binding Kinase 1
Crew, Andrew P, Raina, Kanak, Dong, Hanqing, Qian, Yimin, Wang, Jing, Vigil, Dominico, Serebrenik, Yevgeniy V, Hamman, Brian D, Morgan, Alicia, Ferraro, Caterina, Siu, Kam, Neklesa, Taavi K, Winkler, James D, Coleman, Kevin G, Crews, Craig M
Published in Journal of medicinal chemistry (25.01.2018)
Published in Journal of medicinal chemistry (25.01.2018)
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Poly-ICLC, a TLR3 Agonist, Induces Transient Innate Immune Responses in Patients With Treated HIV-Infection: A Randomized Double-Blinded Placebo Controlled Trial
Saxena, Mansi, Sabado, Rachel L, La Mar, Melissa, Mohri, Hiroshi, Salazar, Andres M, Dong, Hanqing, Correa Da Rosa, Joel, Markowitz, Martin, Bhardwaj, Nina, Miller, Elizabeth
Published in Frontiers in immunology (09.04.2019)
Published in Frontiers in immunology (09.04.2019)
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ROCK1 and ROCK2 Are Required for Non-Small Cell Lung Cancer Anchorage-Independent Growth and Invasion
VIGIL, Dominico, TAI YOUNG KIM, DER, Channing J, PLACHCO, Ana, GARTON, Andrew J, CASTALDO, Linda, PACHTER, Jonathan A, HANQINGDONG, XIN CHEN, TOKAR, Brianna, CAMPBELL, Sharon L
Published in Cancer research (Chicago, Ill.) (15.10.2012)
Published in Cancer research (Chicago, Ill.) (15.10.2012)
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Cyclin-dependent Kinase 2 Negatively Regulates Human Pregnane X Receptor-mediated CYP3A4 Gene Expression in HepG2 Liver Carcinoma Cells
Lin, Wenwei, Wu, Jing, Dong, Hanqing, Bouck, David, Zeng, Fu-Yue, Chen, Taosheng
Published in The Journal of biological chemistry (07.11.2008)
Published in The Journal of biological chemistry (07.11.2008)
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Hijacking the E3 Ubiquitin Ligase Cereblon to Efficiently Target BRD4
Lu, Jing, Qian, Yimin, Altieri, Martha, Dong, Hanqing, Wang, Jing, Raina, Kanak, Hines, John, Winkler, James D., Crew, Andrew P., Coleman, Kevin, Crews, Craig M.
Published in Chemistry & biology (18.06.2015)
Published in Chemistry & biology (18.06.2015)
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Novel 2-phenylquinolin-7-yl-derived imidazo[1,5- a]pyrazines as potent insulin-like growth factor-I receptor (IGF-IR) inhibitors
Mulvihill, Mark J., Ji, Qun-Sheng, Coate, Heather R., Cooke, Andrew, Dong, Hanqing, Feng, Lixin, Foreman, Kenneth, Rosenfeld-Franklin, Maryland, Honda, Ayako, Mak, Gilda, Mulvihill, Kristen M., Nigro, Anthony I., O’Connor, Matthew, Pirrit, Caroline, Steinig, Arno G., Siu, Kam, Stolz, Kathryn M., Sun, Yingchuan, Tavares, Paula A.R., Yao, Yan, Gibson, Neil W.
Published in Bioorganic & medicinal chemistry (01.02.2008)
Published in Bioorganic & medicinal chemistry (01.02.2008)
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Imidazo[1,5- a]pyrazines: Orally efficacious inhibitors of mTORC1 and mTORC2
Crew, Andrew P., Bhagwat, Shripad V., Dong, Hanqing, Bittner, Mark A., Chan, Anna, Chen, Xin, Coate, Heather, Cooke, Andrew, Gokhale, Prafulla C., Honda, Ayako, Jin, Meizhong, Kahler, Jennifer, Mantis, Christine, Mulvihill, Mark J., Tavares-Greco, Paula A., Volk, Brian, Wang, Jing, Werner, Douglas S., Arnold, Lee D., Pachter, Jonathan A., Wild, Robert, Gibson, Neil W.
Published in Bioorganic & medicinal chemistry letters (01.04.2011)
Published in Bioorganic & medicinal chemistry letters (01.04.2011)
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Potent and selective cyclohexyl-derived imidazopyrazine insulin-like growth factor 1 receptor inhibitors with in vivo efficacy
Jin, Meizhong, Kleinberg, Andrew, Cooke, Andy, Gokhale, Prafulla C., Foreman, Kenneth, Dong, Hanqing, Siu, Kam W., Bittner, Mark A., Mulvihill, Kristen M., Yao, Yan, Landfair, Darla, O’Connor, Matthew, Mak, Gilda, Pachter, Jonathan A., Wild, Robert, Rosenfeld-Franklin, Maryland, Ji, Qunsheng, Mulvihill, Mark J.
Published in Bioorganic & medicinal chemistry letters (15.02.2011)
Published in Bioorganic & medicinal chemistry letters (15.02.2011)
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1,3-Disubstituted-imidazo[1,5- a]pyrazines as insulin-like growth-factor-I receptor (IGF-IR) inhibitors
Mulvihill, Mark J., Ji, Qun-Sheng, Werner, Doug, Beck, Patricia, Cesario, Cara, Cooke, Andrew, Cox, Matthew, Crew, Andrew, Dong, Hanqing, Feng, Lixin, Foreman, K.W., Mak, Gilda, Nigro, Anthony, O’Connor, Matthew, Saroglou, Lydia, Stolz, Kathryn M., Sujka, Izabela, Volk, Brian, Weng, Qinghua, Wilkes, Robin
Published in Bioorganic & medicinal chemistry letters (15.02.2007)
Published in Bioorganic & medicinal chemistry letters (15.02.2007)
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Journal Article
Glucokinase-activating ureas
Castelhano, Arlindo L., Dong, Hanqing, Fyfe, Matthew C.T., Gardner, Lisa S., Kamikozawa, Yukari, Kurabayashi, Satomi, Nawano, Masao, Ohashi, Rikiya, Procter, Martin J., Qiu, Li, Rasamison, Chrystelle M., Schofield, Karen L., Shah, Vilas K., Ueta, Kiichiro, Williams, Geoffrey M., Witter, David, Yasuda, Kosuke
Published in Bioorganic & medicinal chemistry letters (01.03.2005)
Published in Bioorganic & medicinal chemistry letters (01.03.2005)
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