4-Aryl-3-arylsulfonyl-quinolines as negative allosteric modulators of metabotropic GluR5 receptors: From HTS hit to development candidate
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Published in Bioorganic & medicinal chemistry letters (15.02.2016)
Published in Bioorganic & medicinal chemistry letters (15.02.2016)
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Thieno[2,3-b]pyridines as negative allosteric modulators of metabotropic GluR5 receptors: Lead optimization
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Published in Bioorganic & medicinal chemistry letters (15.04.2015)
Published in Bioorganic & medicinal chemistry letters (15.04.2015)
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Kynurenic acid amides as novel NR2B selective NMDA receptor antagonists
Borza, István, Kolok, Sándor, Galgóczy, Kornél, Gere, Anikó, Horváth, Csilla, Farkas, Sándor, Greiner, István, Domány, György
Published in Bioorganic & medicinal chemistry letters (15.01.2007)
Published in Bioorganic & medicinal chemistry letters (15.01.2007)
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Journal Article
Thieno[2,3-b]pyridines as negative allosteric modulators of metabotropic GluR5 receptors: Hit-to-lead optimization
Nógrádi, Katalin, Wágner, Gábor, Domány, György, Bobok, Amrita, Magdó, Ildikó, Kiss, Béla, Kolok, Sándor, Fónagy, Katalin, Gyertyán, István, Háda, Viktor, Kóti, János, Gál, Krisztina, Farkas, Sándor, Keserű, György M., Greiner, István, Szombathelyi, Zsolt
Published in Bioorganic & medicinal chemistry letters (15.08.2014)
Published in Bioorganic & medicinal chemistry letters (15.08.2014)
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Selective NR1/2B N-Methyl-d-aspartate Receptor Antagonists among Indole-2-carboxamides and Benzimidazole-2-carboxamides
Borza, István, Bozó, Éva, Barta-Szalai, Gizella, Kiss, Csilla, Tárkányi, Gábor, Demeter, Ádám, Gáti, Tamás, Háda, Viktor, Kolok, Sándor, Gere, Anikó, Fodor, László, Nagy, József, Galgóczy, Kornél, Magdó, Ildikó, Ágai, Béla, Fetter, József, Bertha, Ferenc, Keserü, György M, Horváth, Csilla, Farkas, Sándor, Greiner, István, Domány, György
Published in Journal of medicinal chemistry (08.03.2007)
Published in Journal of medicinal chemistry (08.03.2007)
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Effects of RGH-237 [ N -{4-[4-(3-Aminocarbonyl-phenyl)-piperazin-1-yl]-butyl}-4-bromo-benzamide], an Orally Active, Selective Dopamine D 3 Receptor Partial Agonist in Animal Models of Cocaine Abuse
Gyertyán, István, Kiss, Béla, Gál, Krisztina, Laszlovszky, István, Horváth, Attila, Gémesi, Larisza I., Sághy, Katalin, Pásztor, Gabriella, Zájer, Mária, Kapás, Margit, Csongor, Éva Ágai, Domány, György, Tihanyi, Károly, Szombathelyi, Zsolt
Published in The Journal of pharmacology and experimental therapeutics (01.03.2007)
Published in The Journal of pharmacology and experimental therapeutics (01.03.2007)
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Benzimidazole-2-carboxamides as novel NR2B selective NMDA receptor antagonists
Borza, István, Kolok, Sándor, Gere, Anikó, Nagy, József, Fodor, László, Galgóczy, Kornél, Fetter, József, Bertha, Ferenc, Ágai, Béla, Horváth, Csilla, Farkas, Sándor, Domány, György
Published in Bioorganic & medicinal chemistry letters (01.09.2006)
Published in Bioorganic & medicinal chemistry letters (01.09.2006)
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Cariprazine (RGH-188), a potent D3/D2 dopamine receptor partial agonist, binds to dopamine D3 receptors in vivo and shows antipsychotic-like and procognitive effects in rodents
GYERTYAN, Istvan, KISS, Béla, AGAI CSONGOR, Eva, DOMANY, György, TIHANYI, Károly, SZOMBATHELYI, Zsolt, SAGHY, Katalin, LASZY, Judit, SZABO, Györgyi, SZABADOS, Tamás, GEMESI, Larisza I, PASZTOR, Gabriella, ZAJER-BALAZS, Mária, KAPAS, Margit
Published in Neurochemistry international (01.11.2011)
Published in Neurochemistry international (01.11.2011)
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Quinolinyl- and phenantridinyl-acetamides as bradykinin B1 receptor antagonists
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Published in Bioorganic & medicinal chemistry letters (01.05.2012)
Published in Bioorganic & medicinal chemistry letters (01.05.2012)
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Carbamoyloximes as novel non-competitive mGlu5 receptor antagonists
Galambos, János, Wágner, Gábor, Nógrádi, Katalin, Bielik, Attila, Molnár, László, Bobok, Amrita, Horváth, Attila, Kiss, Béla, Kolok, Sándor, Nagy, József, Kurkó, Dalma, Bakk, Mónika L., Vastag, Mónika, Sághy, Katalin, Gyertyán, István, Gál, Krisztina, Greiner, István, Szombathelyi, Zsolt, Keserű, György M., Domány, György
Published in Bioorganic & medicinal chemistry letters (01.08.2010)
Published in Bioorganic & medicinal chemistry letters (01.08.2010)
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Discovery of cariprazine (RGH-188): A novel antipsychotic acting on dopamine D3/D2 receptors
Ágai-Csongor, Éva, Domány, György, Nógrádi, Katalin, Galambos, János, Vágó, István, Keserű, György Miklós, Greiner, István, Laszlovszky, István, Gere, Anikó, Schmidt, Éva, Kiss, Béla, Vastag, Mónika, Tihanyi, Károly, Sághy, Katalin, Laszy, Judit, Gyertyán, István, Zájer-Balázs, Mária, Gémesi, Larisza, Kapás, Margit, Szombathelyi, Zsolt
Published in Bioorganic & medicinal chemistry letters (15.05.2012)
Published in Bioorganic & medicinal chemistry letters (15.05.2012)
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Design of novel multiple-acting ligands towards SERT and 5-HT sub(2C) receptors
Elias, Oliver, Agai-Csongor, Eva, Domany, Gyorgy, Keserue, Gyorgy Miklos, Gere, Aniko, Kiss, Bela, Hellinger, Eva, Vastag, Monika, Gyertyan, Istvan
Published in Bioorganic & medicinal chemistry letters (01.05.2014)
Published in Bioorganic & medicinal chemistry letters (01.05.2014)
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The influence of 5-HT sub(2A) activity on a 5-HT sub(2C) specific in vivo assay used for early identification of multiple acting SERT and 5-HT sub(2C) receptor ligands
Elias, Oliver, Nogradi, Katalin, Domany, Gyorgy, Szakacs, Zoltan, Koti, Janos, Szantay, Csaba Jr, Tarcsay, Akos, Keserue, Gyorgy M, Gere, Aniko, Kiss, Bela, Kurko, Dalma, Kolok, Sandor, Nemethy, Zsolt, Kapui, Zoltan, Hellinger, Eva, Vastag, Monika, Saghy, Katalin, Kedves, Rita, Gyertyan, Istvan
Published in Bioorganic & medicinal chemistry letters (01.02.2016)
Published in Bioorganic & medicinal chemistry letters (01.02.2016)
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Novel sulfonamides having dual dopamine D2 and D3 receptor affinity show in vivo antipsychotic efficacy with beneficial cognitive and EPS profile
Ágai-Csongor, Éva, Nógrádi, Katalin, Galambos, János, Vágó, István, Bielik, Attila, Magdó, Ildikó, Ignácz-Szendrei, Györgyi, Keserű, György Miklós, Greiner, István, Laszlovszky, István, Béla Kiss, Éva Schmidt, Judit Laszy, Katalin Sághy, Gyertyán, István, Zájer-Balázs, Mária, Gémesi, Larisza, Domány, György
Published in Bioorganic & medicinal chemistry letters (01.10.2007)
Published in Bioorganic & medicinal chemistry letters (01.10.2007)
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Discovery and Preclinical Characterization of 3‑((4-(4-Chlorophenyl)-7-fluoroquinoline-3-yl)sulfonyl)benzonitrile, a Novel Non-acetylenic Metabotropic Glutamate Receptor 5 (mGluR5) Negative Allosteric Modulator for Psychiatric Indications
Galambos, János, Bielik, Attila, Krasavin, Mikhail, Orgován, Zoltán, Domány, György, Nógrádi, Katalin, Wágner, Gábor, Balogh, György T, Béni, Zoltán, Kóti, János, Szakács, Zoltán, Bobok, Amrita, Kolok, Sándor, Mikó-Bakk, Mónika L, Vastag, Mónika, Sághy, Katalin, Laszy, Judit, Halász, Attila Sándor, Balázs, Ottilia, Gál, Krisztina, Greiner, István, Szombathelyi, Zsolt, Keserű, György M
Published in Journal of medicinal chemistry (23.03.2017)
Published in Journal of medicinal chemistry (23.03.2017)
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Oxamides as novel NR2B selective NMDA receptor antagonists
Barta-Szalai, Gizella, Borza, István, Bozó, Éva, Kiss, Csilla, Ágai, Béla, Proszenyák, Ágnes, Keserű, György M, Gere, Anikó, Kolok, Sándor, Galgóczy, Kornél, Horváth, Csilla, Farkas, Sándor, Domány, György
Published in Bioorganic & medicinal chemistry letters (02.08.2004)
Published in Bioorganic & medicinal chemistry letters (02.08.2004)
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Indole-2-carboxamidines as novel NR2B selective NMDA receptor antagonists
Borza, István, Kolok, Sándor, Ignácz-Szendrei, Györgyi, Greiner, István, Tárkányi, Gábor, Galgóczy, Kornél, Horváth, Csilla, Farkas, Sándor, Domány, György
Published in Bioorganic & medicinal chemistry letters (15.12.2005)
Published in Bioorganic & medicinal chemistry letters (15.12.2005)
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Indole-2-carboxamides as novel NR2B selective NMDA receptor antagonists
BORZA, Istvan, KOLOK, Sandor, BIELIK, Attila, NAGY, Jozsef, FARKAS, Sandor, DOMANY, György, GERE, Aniko, AGAI-CSONGOR, Eva, AGAI, Béla, TARKANYI, Gabor, HORVATH, Csilla, BARTA-SZALAI, Gizella, BOZO, Eva, KISS, Csilla
Published in Bioorganic & medicinal chemistry letters (03.11.2003)
Published in Bioorganic & medicinal chemistry letters (03.11.2003)
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NOVEL PIPERAZINE SALTS AS D3/D2 ANTAGONISTS
DOMANY GYORGY, SEBOK FERENC, AGAINE CSONGOR EVA, CZIBULA LASZLO, GREINER ISTVAN
Year of Publication 05.08.2015
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Year of Publication 05.08.2015
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