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Published in Journal of medicinal chemistry (01.11.1995)
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Phosphodiesterase Type IV Inhibition. Structure-Activity Relationships of 1,3-Disubstituted Pyrrolidines
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Published in Journal of medicinal chemistry (01.04.1995)
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Introduction of a conformational switching element on a pyrrolidine ring. Synthesis and evaluation of methyl (R,R)-(.+-.)-3-acetyl-4-[3- (cyclopentyloxy)-4-methoxyphenyl]-3- methyl-1-pyrrolidinecarboxylate, a potent and selective inhibitor of cAMP-specific phosphodiesterase
Stafford, Jeffrey A, Veal, James M, Feldman, Paul L, Valvano, Nicole L, Baer, Philip G, Brackeen, Marcus F, Brawley, E. Sloan, Connolly, Kevin M, Domanico, Paul L
Published in Journal of medicinal chemistry (01.12.1995)
Published in Journal of medicinal chemistry (01.12.1995)
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Adenosine 5'-O-(3-thiotriphosphate) hydrolysis by dynein
Shimizu, Takashi, Katsura, Tatsuo, Domanico, Paul L, Marchese-Ragona, Silvio P, Johnson, Kenneth A
Published in Biochemistry (Easton) (22.08.1989)
Published in Biochemistry (Easton) (22.08.1989)
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Unambiguous stereochemical course of rabbit liver fructose bisphosphatase hydrolysis
Domanico, Paul L, Rahil, Jubrail F, Benkovic, Stephen J
Published in Biochemistry (Easton) (01.03.1985)
Published in Biochemistry (Easton) (01.03.1985)
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Dual Inhibition of Human Type 4 Phosphodiesterase Isostates by (R,R)-(±)-Methyl 3-Acetyl-4-[3-(cyclopentyloxy)-4-methoxyphenyl]-3- methyl-1-pyrrolidinecarboxylate
Tian, Gaochao, Rocque, Warren J, Wiseman, Jeffrey S, Thompson, Irene Z, Holmes, William D, Domanico, Paul L, Stafford, Jeffrey A, Feldman, Paul L, Luther, Michael A
Published in Biochemistry (Easton) (12.05.1998)
Published in Biochemistry (Easton) (12.05.1998)
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17β-(N-tert-butylcarbamoyl)-4-aza-5α-androstan-1-en-3-one is an active site-directed slow time-dependent inhibitor of human steroid 5α-reductase 1
GAOCHAO TIAN, STUART, J. D, FRYE, S. V, BATCHELOR, K. W, WISEMAN, J. S, MOSS, M. L, DOMANICO, P. L, BRAMSON, H. N, PATEL, I. R, KADWELL, S. H, OVERTON, L. K, KOST, T. A, MOOK, R. A
Published in Biochemistry (Easton) (01.03.1994)
Published in Biochemistry (Easton) (01.03.1994)
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17 beta-(N-tert-butylcarbamoyl)-4-aza-5 alpha-androstan-1-en-3-one is an active site-directed slow time-dependent inhibitor of human steroid 5 alpha-reductase 1
Tian, G, Stuart, J D, Moss, M L, Domanico, P L, Bramson, H N, Patel, I R, Kadwell, S H, Overton, L K, Kost, T A, Mook, Jr, R A
Published in Biochemistry (Easton) (01.03.1994)
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Published in Biochemistry (Easton) (01.03.1994)
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Experimental design for high-throughput screening
Lutz, Michael W., Menius, J. Alan, Choi, Tony D., Gooding Laskody, Rebecca, Domanico, Paul L., Goetz, Aaron S., Saussy, David L.
Published in Drug discovery today (01.07.1996)
Published in Drug discovery today (01.07.1996)
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Structure-activity relationships involving the catechol subunit of rolipram
Stafford, Jeffrey A., Feldman, Paul L., Marron, Brian E., Schoenen, Frank J., Valvano, Nicole L., Unwalla, Rayomand J., Domanico, Paul L., Brawley, E.Sloan, Leesnitzer, Michael A., Rose, Dudley A., Dougherty, Robert W.
Published in Bioorganic & medicinal chemistry letters (11.08.1994)
Published in Bioorganic & medicinal chemistry letters (11.08.1994)
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Phosphodiesterase type IV (PDE IV) inhibition. Synthesis and evaluation of a series of 1,3,4-trisubstituted pyrrolidines
Stafford, Jeffrey A, Valvano, Nicole L, Feldman, Paul L, Sloan Brawley, E, Cowan, David J, Domanico, Paul L, Leesnitzer, Michael A, Rose, Dudley A, Stimpson, Stephen A, Strickland, Alan B, Unwalla, Rayomand J, Verghese, Margrith W
Published in Bioorganic & medicinal chemistry letters (07.09.1995)
Published in Bioorganic & medicinal chemistry letters (07.09.1995)
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