Combined solution-phase and solid-phase synthesis of 2-amino-7,8-dihydropteridin-6(5 H)-ones
Metzger, Axel, Qin, Lan-Ying, Cole, Andrew G., Saionz, Kurt W., Brescia, Marc-Raleigh, Gstach, Hubert, Wareing, James R., Zimmermann, Juerg, Brill, Wolfgang K-D., Baldwin, John J., Dolle, Roland E., Henderson, Ian
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Published in Tetrahedron letters (16.12.2009)
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Novel pyridine derivatives as potent and selective CB sub(2) cannabinoid receptor agonists
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Published in Bioorganic & medicinal chemistry letters (01.09.2009)
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Synthesis and Pharmacological Evaluation of Novel Octahydro-1 H -pyrido[1,2-a]pyrazine as μ-Opioid Receptor Antagonists
Le Bourdonnec, Bertrand, Goodman, Allan J., Graczyk, Thomas M., Belanger, Serge, Seida, Pamela R., DeHaven, Robert N., Dolle, Roland E.
Published in Journal of medicinal chemistry (01.12.2006)
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Novel sulfamoyl benzamides as selective CB sub(2) agonists with improved in vitro metabolic stability
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Published in Bioorganic & medicinal chemistry letters (01.01.2010)
Published in Bioorganic & medicinal chemistry letters (01.01.2010)
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Novel sulfamoyl benzamides as selective CB 2 agonists with improved in vitro metabolic stability
Sellitto, Ian, Bourdonnec, Bertrand Le, Worm, Karin, Goodman, Allan, Savolainen, Markku A., Chu, Guo-Hua, Ajello, Christopher W., Saeui, Christopher T., Leister, Lara K., Cassel, Joel A., DeHaven, Robert N., LaBuda, Christopher J., Koblish, Michael, Little, Patrick J., Brogdon, Bernice L., Smith, Steven A., Dolle, Roland E.
Published in Bioorganic & medicinal chemistry letters (2010)
Published in Bioorganic & medicinal chemistry letters (2010)
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Discovery of N-(3-(morpholinomethyl)-phenyl)-amides as potent and selective CB 2 agonists
Worm, Karin, Weaver, Damian G., Green, Rosalyn C., Saeui, Christopher T., Dulay, Doreen-Marie S., Barker, William M., Cassel, Joel A., Stabley, Gabriel J., DeHaven, Robert N., LaBuda, Christopher J., Koblish, Michael, Brogdon, Bernice L., Smith, Steven A., Dolle, Roland E.
Published in Bioorganic & medicinal chemistry letters (2009)
Published in Bioorganic & medicinal chemistry letters (2009)
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Novel pyridine derivatives as potent and selective CB 2 cannabinoid receptor agonists
Chu, Guo-Hua, Saeui, Christopher T., Worm, Karin, Weaver, Damian G., Goodman, Allan J., Broadrup, Robert L., Cassel, Joel A., DeHaven, Robert N., LaBuda, Christopher J., Koblish, Michael, Brogdon, Bernice, Smith, Steve, Bourdonnec, Bertrand Le, Dolle, Roland E.
Published in Bioorganic & medicinal chemistry letters (2009)
Published in Bioorganic & medicinal chemistry letters (2009)
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Sulfamoyl benzamides as novel CB sub(2) cannabinoid receptor ligands
Worm, Karin, Zhou, QJean, Saeui, Christopher T, Green, Rosalyn C, Cassel, Joel A, Stabley, Gabriel J, DeHaven, Robert N, Conway-James, Nathalie, LaBuda, Christopher J, Koblish, Michael, Little, Patrick J, Dolle, Roland E
Published in Bioorganic & medicinal chemistry (01.05.2008)
Published in Bioorganic & medicinal chemistry (01.05.2008)
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CB 2 selective sulfamoyl benzamides: Optimization of the amide functionality
Goodman, Allan J., Ajello, Christopher W., Worm, Karin, Bourdonnec, Bertrand Le, Savolainen, Markku A., O’Hare, Heather, Cassel, Joel A., Stabley, Gabriel J., DeHaven, Robert N., LaBuda, Christopher J., Koblish, Michael, Little, Patrick J., Brogdon, Bernice L., Smith, Steven A., Dolle, Roland E.
Published in Bioorganic & medicinal chemistry letters (2009)
Published in Bioorganic & medicinal chemistry letters (2009)
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